NL8601043A - Anti-psychotische benzisothiazool-s-oxide-verbinding. - Google Patents

Anti-psychotische benzisothiazool-s-oxide-verbinding. Download PDF

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Publication number
NL8601043A
NL8601043A NL8601043A NL8601043A NL8601043A NL 8601043 A NL8601043 A NL 8601043A NL 8601043 A NL8601043 A NL 8601043A NL 8601043 A NL8601043 A NL 8601043A NL 8601043 A NL8601043 A NL 8601043A
Authority
NL
Netherlands
Prior art keywords
compound
psychotic
bmy
formula
acid addition
Prior art date
Application number
NL8601043A
Other languages
English (en)
Dutch (nl)
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of NL8601043A publication Critical patent/NL8601043A/nl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NL8601043A 1985-04-24 1986-04-23 Anti-psychotische benzisothiazool-s-oxide-verbinding. NL8601043A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72644985 1985-04-24
US06/726,449 US4656173A (en) 1985-04-24 1985-04-24 Antipsychotic benzisothiazole S-oxide compound

Publications (1)

Publication Number Publication Date
NL8601043A true NL8601043A (nl) 1986-11-17

Family

ID=24918649

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8601043A NL8601043A (nl) 1985-04-24 1986-04-23 Anti-psychotische benzisothiazool-s-oxide-verbinding.

Country Status (26)

Country Link
US (1) US4656173A (da)
JP (1) JPH0764842B2 (da)
KR (1) KR900000372B1 (da)
CN (1) CN1017528B (da)
AT (1) AT394719B (da)
AU (1) AU592787B2 (da)
BE (1) BE904662A (da)
CA (1) CA1247102A (da)
CH (1) CH666034A5 (da)
DE (1) DE3613739C2 (da)
DK (1) DK187686A (da)
EG (1) EG18002A (da)
ES (1) ES8708228A1 (da)
FI (1) FI84604C (da)
FR (1) FR2581064B1 (da)
GB (1) GB2174393B (da)
GR (1) GR861063B (da)
HU (1) HU195654B (da)
IE (1) IE59182B1 (da)
IT (1) IT1208600B (da)
LU (1) LU86405A1 (da)
MY (1) MY102041A (da)
NL (1) NL8601043A (da)
PT (1) PT82450B (da)
SE (1) SE462163B (da)
ZA (1) ZA861531B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4780466A (en) * 1988-03-17 1988-10-25 Hoechst-Roussel Pharmaceuticals, Inc. Arylpiperazinylalkoxy derivatives of cyclic imides
EP0350145A3 (en) * 1988-04-28 1990-07-04 Yamanouchi Pharmaceutical Co. Ltd. Pyridylthiazolidine carboxamide derivatives and their intermediates and production of both
HUT61760A (en) * 1988-09-16 1993-03-01 Pfizer Process for producing bridged, bicyclic imides comprising 4-/4-(3-benzisothiazolyl)-1-piperazinyl/-butyl group and pharmaceutical compositions comprising such compounds
US4956368A (en) * 1989-07-24 1990-09-11 Bristol-Myers Company Metabolites and prodrug formulations of 8-[4-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]butyl]-8-azaspiro[4.5]decane-7,9-dione
US4968792A (en) * 1989-09-25 1990-11-06 American Home Products Corporation Psychotropic benzisothiazole derivatives
US5162321A (en) * 1989-12-20 1992-11-10 Adir Et Compagnie 1-naphthyl piperazines useful as 5-HT1A receptor ligands
JP2800953B2 (ja) * 1990-07-06 1998-09-21 住友製薬株式会社 新規なイミド誘導体
EP2919788A4 (en) 2012-11-14 2016-05-25 Univ Johns Hopkins METHODS AND COMPOSITIONS FOR THE TREATMENT OF SCHIZOPHRENIA

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE759371A (fr) * 1969-11-24 1971-05-24 Bristol Myers Co Azaspirodecanediones heterocycliques et procedes pour leur preparation
US3976776A (en) * 1972-12-06 1976-08-24 Mead Johnson & Company Tranquilizer process employing N-(heteroarcyclic)piperazinylalkylazaspiroalkanediones
CH582699A5 (da) * 1973-03-26 1976-12-15 Sandoz Ag
AT342057B (de) * 1974-04-25 1978-03-10 Thomae Gmbh Dr K Verfahren zur herstellung von neuen 3-piperazino-isochinolinen und deren salzen
FI753625A (da) * 1975-01-06 1976-07-07 Spofa Vereinigte Pharma Werke
JPS51144735A (en) * 1975-06-06 1976-12-13 Nippon Nohyaku Co Ltd A remedy for hepatic failure
US4411901A (en) * 1981-12-23 1983-10-25 Mead Johnson & Company Benzisothiazole and benzisoxazole piperazine derivatives
US4452799A (en) * 1981-12-23 1984-06-05 Mead Johnson & Company Benzisothiazole and benzisoxazole piperazine derivatives
US4524206A (en) * 1983-09-12 1985-06-18 Mead Johnson & Company 1-Heteroaryl-4-(2,5-pyrrolidinedion-1-yl)alkyl)piperazine derivatives

Also Published As

Publication number Publication date
FR2581064A1 (fr) 1986-10-31
DE3613739C2 (de) 1993-12-09
JPS61251683A (ja) 1986-11-08
HU195654B (en) 1988-06-28
CN86102742A (zh) 1987-02-04
PT82450A (en) 1986-05-01
AT394719B (de) 1992-06-10
CH666034A5 (de) 1988-06-30
IT8620187A0 (it) 1986-04-23
BE904662A (fr) 1986-10-23
DE3613739A1 (de) 1986-11-20
FI861668A0 (fi) 1986-04-21
FI861668A (fi) 1986-10-25
SE462163B (sv) 1990-05-14
FI84604C (fi) 1991-12-27
FI84604B (fi) 1991-09-13
CN1017528B (zh) 1992-07-22
SE8601883L (sv) 1986-10-25
AU592787B2 (en) 1990-01-25
GR861063B (en) 1986-09-01
PT82450B (pt) 1988-11-30
CA1247102A (en) 1988-12-20
MY102041A (en) 1992-02-29
ES8708228A1 (es) 1987-10-01
HUT42088A (en) 1987-06-29
FR2581064B1 (fr) 1988-09-16
ATA110486A (de) 1991-11-15
KR900000372B1 (ko) 1990-01-25
DK187686D0 (da) 1986-04-23
IT1208600B (it) 1989-07-10
IE861083L (en) 1986-10-24
GB2174393B (en) 1989-02-01
AU5612186A (en) 1986-10-30
US4656173A (en) 1987-04-07
GB8609932D0 (en) 1986-05-29
IE59182B1 (en) 1994-01-26
DK187686A (da) 1986-10-25
GB2174393A (en) 1986-11-05
ZA861531B (en) 1986-10-29
LU86405A1 (fr) 1986-11-05
EG18002A (en) 1991-08-30
JPH0764842B2 (ja) 1995-07-12
KR860008174A (ko) 1986-11-12
ES554284A0 (es) 1987-10-01
SE8601883D0 (sv) 1986-04-23

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Legal Events

Date Code Title Description
DNT Communications of changes of names of applicants whose applications have been laid open to public inspection

Free format text: BRISTOL-MYERS SQUIBB COMPANY

BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
BN A decision not to publish the application has become irrevocable