NL8300934A - Gesubstitueerde 1h-pyrazolo1,5-a-pyrimidinen, werkwijzen ter bereiding ervan, alsmede farmaceutische preparaten, die deze verbindingen bevatten. - Google Patents

Gesubstitueerde 1h-pyrazolo1,5-a-pyrimidinen, werkwijzen ter bereiding ervan, alsmede farmaceutische preparaten, die deze verbindingen bevatten. Download PDF

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Publication number
NL8300934A
NL8300934A NL8300934A NL8300934A NL8300934A NL 8300934 A NL8300934 A NL 8300934A NL 8300934 A NL8300934 A NL 8300934A NL 8300934 A NL8300934 A NL 8300934A NL 8300934 A NL8300934 A NL 8300934A
Authority
NL
Netherlands
Prior art keywords
pyrazolo1
pyrimidines
substituted
preparing
compounds
Prior art date
Application number
NL8300934A
Other languages
English (en)
Dutch (nl)
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838303089A external-priority patent/GB8303089D0/en
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of NL8300934A publication Critical patent/NL8300934A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NL8300934A 1982-03-16 1983-03-15 Gesubstitueerde 1h-pyrazolo1,5-a-pyrimidinen, werkwijzen ter bereiding ervan, alsmede farmaceutische preparaten, die deze verbindingen bevatten. NL8300934A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8207637 1982-03-16
GB838303089A GB8303089D0 (en) 1983-02-04 1983-02-04 Substituted 1h-pyrazolo 1,5-a pyrimidines

Publications (1)

Publication Number Publication Date
NL8300934A true NL8300934A (nl) 1983-10-17

Family

ID=26282260

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8300934A NL8300934A (nl) 1982-03-16 1983-03-15 Gesubstitueerde 1h-pyrazolo1,5-a-pyrimidinen, werkwijzen ter bereiding ervan, alsmede farmaceutische preparaten, die deze verbindingen bevatten.

Country Status (13)

Country Link
US (1) US4482555A (fr)
AU (1) AU557300B2 (fr)
CA (1) CA1192546A (fr)
CH (1) CH654306A5 (fr)
DE (1) DE3309432A1 (fr)
DK (1) DK120783A (fr)
FI (1) FI74469C (fr)
FR (1) FR2523582B1 (fr)
IL (1) IL68133A (fr)
IT (1) IT1194555B (fr)
NL (1) NL8300934A (fr)
SE (1) SE450573B (fr)
SU (1) SU1366060A3 (fr)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6245759B1 (en) * 1999-03-11 2001-06-12 Merck & Co., Inc. Tyrosine kinase inhibitors
MY125533A (en) 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
WO2004089471A2 (fr) * 2003-04-11 2004-10-21 Novo Nordisk A/S Utilisation pharmaceutique de pyrazolo[1,5-a]pyrimidines substituees
EP1782859A3 (fr) * 2003-04-11 2009-09-30 High Point Pharmaceuticals, LLC Utilisation thérapeutique de pyrazolo [1,5- a] pyrimidines
US7772232B2 (en) 2004-04-15 2010-08-10 Bristol-Myers Squibb Company Quinazolinyl compounds as inhibitors of potassium channel function
EP1802623A1 (fr) * 2004-10-12 2007-07-04 Novo Nordisk A/S Composes spiro actifs du type a- hydroxysteroide deshydrogenase de type 1
AU2006310519A1 (en) * 2005-11-01 2007-05-10 High Point Pharmaceuticals, Llc Pharmaceutical use of substituted amides
AU2006310518A1 (en) * 2005-11-01 2007-05-10 High Point Pharmaceuticals, Llc Pharmaceutical use of substituted amides
JP2009530346A (ja) * 2006-03-21 2009-08-27 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー メタボリックシンドロームの治療用のアダマンタン誘導体
EP2010479A1 (fr) 2006-04-07 2009-01-07 High Point Pharmaceuticals, LLC COMPOSÉS ACTIFS de 11 BETA -HYDROXYSTÉROÏDE DÉSHYDROGÉNASE DE TYPE 1
EP2038255A2 (fr) * 2006-06-16 2009-03-25 High Point Pharmaceuticals, LLC Utilisation pharmaceutique de piperidines carboxamides substitués
US8048908B2 (en) * 2006-07-13 2011-11-01 High Point Pharmaceuticals, Llc 11β-hydroxysteroid dehydrogenase type 1 active compounds
EP1878721A1 (fr) * 2006-07-13 2008-01-16 Novo Nordisk A/S 4-Piperidylbenzamides en tant qu'inhibiteurs de la 11-beta-hydroxysteroid dehydrogenase type 1
BRPI0806847A2 (pt) 2007-02-23 2014-04-29 High Point Pharmaceuticals Llc N-adamantil benzamidas como inibidores de 11-beta-hidroxiesteróide desidrogenase
US20110003856A1 (en) * 2007-02-23 2011-01-06 Soren Ebdrup N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
JP2010519242A (ja) * 2007-02-23 2010-06-03 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー 新規化合物
JP2010519239A (ja) * 2007-02-23 2010-06-03 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー １１−ベータ−ヒドロキシステロイドデヒドロゲナーゼの阻害因子としてのｎ−アドマンチルベンザミド
KR20100015414A (ko) * 2007-03-09 2010-02-12 하이 포인트 파마슈티칼스, 엘엘씨 히드록시스테로이드 탈수소효소 억제제로서 인돌- 및 벤즈이미다졸 아미드
EP2141990A4 (fr) * 2007-03-28 2011-07-06 High Point Pharmaceuticals Llc Composés actifs sur 11bêta-hsd1
EP2152081B1 (fr) * 2007-04-11 2012-10-24 High Point Pharmaceuticals, LLC Nouveaux composés
CN101711106B (zh) * 2007-04-24 2013-02-06 高点制药有限责任公司 取代的酰胺类的药物应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE786611A (fr) * 1971-08-16 1973-01-22 Int Chem & Nuclear Corp Nouveaux inhibiteurs de xanthine-oxydase et leur procede de preparatio
US3907799A (en) * 1971-08-16 1975-09-23 Icn Pharmaceuticals Xanthine oxidase inhibitors
BE792533A (fr) * 1971-12-09 1973-06-08 Int Chem & Nuclear Corp Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation
US3925385A (en) * 1972-04-20 1975-12-09 Icn Pharmaceuticals 6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines
US4093617A (en) * 1974-11-12 1978-06-06 Icn Pharmaceuticals, Inc. 3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines
US4048184A (en) * 1976-11-15 1977-09-13 E. R. Squibb & Sons, Inc. 6-Phenyl-2H-pyrazolo[3,4-b]pyridines
US4281000A (en) * 1979-07-09 1981-07-28 American Cyanamid Company Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents

Also Published As

Publication number Publication date
IT1194555B (it) 1988-09-22
SE8301412L (sv) 1983-09-17
IL68133A0 (en) 1983-06-15
US4482555A (en) 1984-11-13
SE8301412D0 (sv) 1983-03-15
CA1192546A (fr) 1985-08-27
SU1366060A3 (ru) 1988-01-07
FI830864L (fi) 1983-09-17
DK120783A (da) 1983-09-17
CH654306A5 (de) 1986-02-14
AU1230483A (en) 1983-09-22
IT8320024A0 (it) 1983-03-11
DK120783D0 (da) 1983-03-15
FI830864A0 (fi) 1983-03-15
AU557300B2 (en) 1986-12-18
FI74469B (fi) 1987-10-30
IL68133A (en) 1985-12-31
FR2523582B1 (fr) 1985-12-06
SE450573B (sv) 1987-07-06
FI74469C (fi) 1988-02-08
FR2523582A1 (fr) 1983-09-23
DE3309432A1 (de) 1983-09-22

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BV The patent application has lapsed
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
BN A decision not to publish the application has become irrevocable