NL8002685A - 9-hydrazono-6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyri- midin-4-on derivaten en werkwijze voor de bereiding daarvan. - Google Patents

9-hydrazono-6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyri- midin-4-on derivaten en werkwijze voor de bereiding daarvan. Download PDF

Info

Publication number
NL8002685A
NL8002685A NL8002685A NL8002685A NL8002685A NL 8002685 A NL8002685 A NL 8002685A NL 8002685 A NL8002685 A NL 8002685A NL 8002685 A NL8002685 A NL 8002685A NL 8002685 A NL8002685 A NL 8002685A
Authority
NL
Netherlands
Prior art keywords
group
hydrogen
optionally substituted
short chain
formula
Prior art date
Application number
NL8002685A
Other languages
English (en)
Dutch (nl)
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of NL8002685A publication Critical patent/NL8002685A/nl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pulmonology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NL8002685A 1979-05-11 1980-05-09 9-hydrazono-6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyri- midin-4-on derivaten en werkwijze voor de bereiding daarvan. NL8002685A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU79CI1934A HU178453B (en) 1979-05-11 1979-05-11 Process for producing 9-hydrazino-4-oxo-6,7,8,9-tetrahydro-4h-p-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
HUCI001934 1979-05-11

Publications (1)

Publication Number Publication Date
NL8002685A true NL8002685A (nl) 1980-11-13

Family

ID=10994749

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8002685A NL8002685A (nl) 1979-05-11 1980-05-09 9-hydrazono-6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyri- midin-4-on derivaten en werkwijze voor de bereiding daarvan.

Country Status (25)

Country Link
US (1) US4456752A (no)
JP (1) JPS5622785A (no)
AT (1) AT375937B (no)
AU (1) AU550521B2 (no)
BE (1) BE883219A (no)
CA (1) CA1153371A (no)
CH (1) CH648847A5 (no)
DE (1) DE3017719A1 (no)
DK (1) DK205080A (no)
ES (1) ES8105003A1 (no)
FI (1) FI68826C (no)
FR (1) FR2456099B1 (no)
GB (1) GB2051783B (no)
GR (1) GR68519B (no)
HU (1) HU178453B (no)
IL (1) IL60027A (no)
IT (1) IT1133088B (no)
LU (1) LU82438A1 (no)
NL (1) NL8002685A (no)
NO (2) NO151464C (no)
PL (1) PL127345B1 (no)
PT (1) PT71215A (no)
SE (1) SE441749B (no)
SU (1) SU980622A3 (no)
YU (1) YU122280A (no)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178453B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydrazino-4-oxo-6,7,8,9-tetrahydro-4h-p-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
US4395549A (en) 1981-10-02 1983-07-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3141043A (en) * 1961-03-24 1964-07-14 Purdue Research Foundation Cyclopentadienylimines, process for their production and condensation products thereof
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity
HU178452B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 9-substituted amino-4-oxo-6,7-dihydro-4h-pyrido/1,2-a/pyrimidine derivatives
HU179443B (en) * 1979-05-11 1982-10-28 Chinoin Gyogyszer Es Vegyeszet Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines
HU178453B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydrazino-4-oxo-6,7,8,9-tetrahydro-4h-p-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives

Also Published As

Publication number Publication date
SU980622A3 (ru) 1982-12-07
DK205080A (da) 1980-11-12
NO151464C (no) 1985-04-17
NO801380L (no) 1980-11-12
IT8067739A0 (it) 1980-05-09
NO151464B (no) 1985-01-02
IL60027A0 (en) 1980-07-31
SE8003481L (sv) 1980-11-12
LU82438A1 (de) 1980-07-31
AU550521B2 (en) 1986-03-27
CA1153371A (en) 1983-09-06
ES491769A0 (es) 1981-06-01
NO152750B (no) 1985-08-05
CH648847A5 (de) 1985-04-15
SE441749B (sv) 1985-11-04
ES8105003A1 (es) 1981-06-01
BE883219A (fr) 1980-09-01
DE3017719A1 (de) 1981-02-05
PT71215A (en) 1980-06-01
YU122280A (en) 1983-02-28
FI68826B (fi) 1985-07-31
HU178453B (en) 1982-05-28
AT375937B (de) 1984-09-25
FR2456099A1 (fr) 1980-12-05
GB2051783A (en) 1981-01-21
AU5828080A (en) 1980-11-13
IT1133088B (it) 1986-07-09
GB2051783B (en) 1983-04-27
JPS5622785A (en) 1981-03-03
FR2456099B1 (fr) 1985-07-05
GR68519B (no) 1982-01-11
FI68826C (fi) 1985-11-11
NO801379L (no) 1980-11-12
FI801513A (fi) 1980-11-12
PL127345B1 (en) 1983-10-31
US4456752A (en) 1984-06-26
IL60027A (en) 1984-05-31
ATA247680A (de) 1984-02-15
PL224162A1 (no) 1981-02-13
NO152750C (no) 1985-11-13

Similar Documents

Publication Publication Date Title
US7256195B2 (en) Preparation of risperidone
SE446337B (sv) Nya 4-anilinokinazolinderivat till anvendning som analgetiska och antiinflammatoriska medel samt farmaceutisk komposition derav
EP3013815B1 (en) Carbazole carboxamide compounds useful as kinase inhibitors
JPH054983A (ja) イソキノリノン誘導体、その製造方法およびその誘導体を有効成分として含有する5−ht3 レセプター拮抗剤
PL125321B1 (en) Process for preparing novel,condensed derivatives of pyrimidines
KR20130046436A (ko) 안드로겐 수용체 길항제, 항암제로서 사이클릭 n,n''-다이아릴티오우레아 및 n,n''-다이아릴우레아, 이의 제조방법 및 이의 용도
CN109111426B (zh) 一类稠合双环杂芳基或芳基化合物,及其用途
CN103813793A (zh) 4-叔丁基-n-[4-氯-2-(1-氧基-吡啶-4-羰基)-苯基]-苯磺酰胺钠盐的多晶型
US3681360A (en) Antiviral substituted acridanones
NL8002685A (nl) 9-hydrazono-6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyri- midin-4-on derivaten en werkwijze voor de bereiding daarvan.
JPS6345279A (ja) 新規ピリド〔2,3−d〕ピリミジン誘導体、その製造方法並びに該化合物を含有する医薬組成物
JPS5831351B2 (ja) 6−フエニル−S−トリアゾロ−(4,3−a)−ピリド−(2,3−f)−(1,4)−ジアゼピン及びその製造方法
WO2002012200A9 (en) Preparation of risperidone
LU86421A1 (fr) Derives de piperazine 1,4-disubstitues,composition pharmaceutique les contenant;leur procede d'obtention
CA1209994A (en) 2-piperazinyl-quinazoline derivatives, their production and pharmaceutical compositions containing them
CA1242201A (en) Asymeticl 1,4-dihydropyridine-3,5-dicarboxylic acid esters having moieties facilitating separation and useful as intermediates for preparing therapeutically active analogues
US4452982A (en) Process for the preparation of nitrogen-bridgehead condensed pyrimidine compounds, and pharmaceutical compositions containing them
EP3484872B1 (en) Crystalline forms of 4-cyano-n-(2-(4,4-dimethylcyclohex-1-en-1-yl)-6-(2,2,6,6-tetramethyltetrahydro-2h-pyran-4-yl)pyridin-3-yl)-1h-imidazole-2-carboxamide
JPS6024794B2 (ja) オキサジアゾロピリミジン誘導体
JPH06505017A (ja) 三環式イソインドリノンの抗ウイルス医薬としての使用、ならびに新規な光学活性イソインドリノン
US3047571A (en) Derivatives of oxopiperidinyl phenthiazines
JPS5989666A (ja) 5H−ジベンゾ〔b,f〕アゼピン−5−カルボキサミド、その製造方法、及びそれを含む医薬用調製物
GB2128190A (en) Chemical compounds
NZ202351A (en) Imidazole carboxamines
EA041321B1 (ru) Кристаллические формы 4-циано-n-(2-(4,4-диметилциклогекс-1-ен-1-ил)-6-(2,2,6,6-тетраметилтетрагидро-2h-пиран-4-ил)пиридин-3-ил)-1h-имидазол-2-карбоксамида

Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BV The patent application has lapsed