HU179443B - Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines - Google Patents

Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines

Info

Publication number
HU179443B
HU179443B HU79CI1932A HUCI001932A HU179443B HU 179443 B HU179443 B HU 179443B HU 79CI1932 A HU79CI1932 A HU 79CI1932A HU CI001932 A HUCI001932 A HU CI001932A HU 179443 B HU179443 B HU 179443B
Authority
HU
Hungary
Prior art keywords
square bracket
closed
square
pyrimidines
bracket
Prior art date
Application number
HU79CI1932A
Other languages
Hungarian (hu)
Inventor
Istvan Hermecz
Tibor Breining
Arpadne Vasvari
Agnes Horvath
Zoltan Meszaros
Istvan Bitter
Jozsef Koekoesi
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Priority to HU79CI1932A priority Critical patent/HU179443B/en
Priority to IL59967A priority patent/IL59967A/en
Priority to GR61852A priority patent/GR68518B/el
Priority to SU802920002A priority patent/SU1151210A3/en
Priority to DE19803017564 priority patent/DE3017564A1/en
Priority to CS803258A priority patent/CS241025B2/en
Priority to SE8003479A priority patent/SE441747B/en
Priority to LU82437A priority patent/LU82437A1/en
Priority to AT0247580A priority patent/AT377261B/en
Priority to NO801378A priority patent/NO152607C/en
Priority to CA000351662A priority patent/CA1141379A/en
Priority to GB8015469A priority patent/GB2051048B/en
Priority to IT67719/80A priority patent/IT1133085B/en
Priority to CH366380A priority patent/CH646971A5/en
Priority to DK204680A priority patent/DK204680A/en
Priority to FR8010481A priority patent/FR2456101A1/en
Priority to FI801512A priority patent/FI68825C/en
Priority to BE0/200550A priority patent/BE883217A/en
Priority to PT71213A priority patent/PT71213A/en
Priority to NL8002678A priority patent/NL8002678A/en
Priority to JP6161680A priority patent/JPS5615286A/en
Priority to PL1980224163A priority patent/PL124035B1/en
Priority to DD80221053A priority patent/DD150605A5/en
Priority to ES491896A priority patent/ES491896A0/en
Publication of HU179443B publication Critical patent/HU179443B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09BORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B62/00Reactive dyes, i.e. dyes which form covalent bonds with the substrates or which polymerise with themselves
HU79CI1932A 1979-05-11 1979-05-11 Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines HU179443B (en)

Priority Applications (24)

Application Number Priority Date Filing Date Title
HU79CI1932A HU179443B (en) 1979-05-11 1979-05-11 Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines
IL59967A IL59967A (en) 1979-05-11 1980-05-01 Geminal dihalogen derivatives of condensed pyrimidine-4-one compounds and a process for their preparation
GR61852A GR68518B (en) 1979-05-11 1980-05-03
SU802920002A SU1151210A3 (en) 1979-05-11 1980-05-08 Method of obtaining heminal dihalogen derivatives of condensed pyrimidin-4-ons,racemates or optically active antipodes
DE19803017564 DE3017564A1 (en) 1979-05-11 1980-05-08 COMMON DIHALOGEN DERIVATIVES OF CONDENSED PYRIMIDINE-4-ON COMPOUNDS, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS
CS803258A CS241025B2 (en) 1979-05-11 1980-05-08 Method of fussed pyrimidine-4-ons' dihalogenated derivatives production
SE8003479A SE441747B (en) 1979-05-11 1980-05-08 COMMON DIHALOGEN DERIVATIVES OF CONDENSED PYRIMIDIN-4-ON COMPOUNDS
LU82437A LU82437A1 (en) 1979-05-11 1980-05-09 GEMINED DIHALOGEN DERIVATIVES OF 4 CONDENSED PYRIMIDINE-ONE COMPOUNDS, METHOD OF PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
AT0247580A AT377261B (en) 1979-05-11 1980-05-09 METHOD FOR PRODUCING NEW CONDENSED PYRIMIDIN-4-ON DERIVATIVES AND THEIR SALTS AND OPTICAL ANTIPODES
NO801378A NO152607C (en) 1979-05-11 1980-05-09 OUTSTANDING MATERIALS FOR USE IN THE PREPARATION OF THERAPEUTIC ACTIVE PYRIMIDINE DERIVATIVES
CA000351662A CA1141379A (en) 1979-05-11 1980-05-09 Geminal dihalogen derivatives of condensed pyrimidine-4-one compounds, process for their preparation and pharmaceutical compositions containing them
GB8015469A GB2051048B (en) 1979-05-11 1980-05-09 Geminal dihalogen derivatives of condensed pyrimidin-4-one compounds their preparation and pharmaceutical compositions containing them
IT67719/80A IT1133085B (en) 1979-05-11 1980-05-09 GEMINAL DIALOGENATED DERIVATIVES OF CONDENSED COMPOUNDS OF PIRIMIDIN 4 ONE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
CH366380A CH646971A5 (en) 1979-05-11 1980-05-09 DIHALOGEN-SUBSTITUTED ANELATED PYRIMIDINE-4-ON DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF.
DK204680A DK204680A (en) 1979-05-11 1980-05-09 COMMON DIHALOGEN DERIVATIVES OF THEIR CONDENSED PYRIMIDIN-4-ONES OF THEIR PREPARATION AND USE
FR8010481A FR2456101A1 (en) 1979-05-11 1980-05-09 GEMINAL DIHALOGEN DERIVATIVES OF PYRIMIDIN-4-ONE CONDENSED, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FI801512A FI68825C (en) 1979-05-11 1980-05-09 GEMINALA DIHALOGENDERIV AV AVONDENSERADE PYRIMIDIN-4-ONER VILKA AER MELLANPRODUKTER VID FRAMSTAELLNING AV THERAPEUTIC ANAENDBARA 9-AMINOPYRIDO (1,2-A) PYRIMIDIN-OCH 9-HYDRATSONO-6,, 8,9-P-6,9-8,9-T -A) PYRIMIDINDERIVAT
BE0/200550A BE883217A (en) 1979-05-11 1980-05-09 GEMINAL DIHALOGEN DERIVATIVES OF PYRIMIDIN-4-ONE CONDENSED, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
PT71213A PT71213A (en) 1979-05-11 1980-05-09 Geminal dihalogen derivatives of condensed pyrimidine-4-one compounds process for their preparation and pharmaceutical compositions containing them
NL8002678A NL8002678A (en) 1979-05-11 1980-05-09 TWIN DIHALOGENE DERIVATIVES OF CONDENSED PYRIMIDINE 4 COMPOUNDS, METHOD FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE COMPOUNDS.
JP6161680A JPS5615286A (en) 1979-05-11 1980-05-09 Zwitter dihalogen derivative of condensed pyrimidinee44one compound* its manufacture and drug composition containing same
PL1980224163A PL124035B1 (en) 1979-05-11 1980-05-10 Process for preparing novel,substituted halo derivatives of pyrido/1,2-a/pyrimidines,pyrrol/1,2-a/pyrimidines and pyrimido/1,2-a/azepines
DD80221053A DD150605A5 (en) 1979-05-11 1980-05-12 PROCESS FOR PREPARING DIHALOGEN-SUBSTITUTED CONDENSED PYRIMIDIN-4-ON DERIVATIVES
ES491896A ES491896A0 (en) 1979-05-11 1980-05-12 PROCEDURE FOR PREPARING GEMINAL DIHALOGENIC DERIVATIVES

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU79CI1932A HU179443B (en) 1979-05-11 1979-05-11 Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines

Publications (1)

Publication Number Publication Date
HU179443B true HU179443B (en) 1982-10-28

Family

ID=10994747

Family Applications (1)

Application Number Title Priority Date Filing Date
HU79CI1932A HU179443B (en) 1979-05-11 1979-05-11 Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines

Country Status (24)

Country Link
JP (1) JPS5615286A (en)
AT (1) AT377261B (en)
BE (1) BE883217A (en)
CA (1) CA1141379A (en)
CH (1) CH646971A5 (en)
CS (1) CS241025B2 (en)
DD (1) DD150605A5 (en)
DE (1) DE3017564A1 (en)
DK (1) DK204680A (en)
ES (1) ES491896A0 (en)
FI (1) FI68825C (en)
FR (1) FR2456101A1 (en)
GB (1) GB2051048B (en)
GR (1) GR68518B (en)
HU (1) HU179443B (en)
IL (1) IL59967A (en)
IT (1) IT1133085B (en)
LU (1) LU82437A1 (en)
NL (1) NL8002678A (en)
NO (1) NO152607C (en)
PL (1) PL124035B1 (en)
PT (1) PT71213A (en)
SE (1) SE441747B (en)
SU (1) SU1151210A3 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178453B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydrazino-4-oxo-6,7,8,9-tetrahydro-4h-p-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
US4395549A (en) 1981-10-02 1983-07-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
US5158952A (en) * 1988-11-07 1992-10-27 Janssen Pharmaceutica N.V. 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use
UA72189C2 (en) 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Aqueous suspensions of 9-hydroxy-risperidone fatty acid esters provided in submicron form

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT302311B (en) * 1966-11-02 1972-09-15 Chinoin Gyogyszer Es Vegyeszet PROCESS FOR THE PREPARATION OF HOMOPYRIMIDAZOLE DERIVATIVES AND THEIR ACID-ADDITIONAL SALTS AND QUATERNAL AMMONIUM SALTS
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity

Also Published As

Publication number Publication date
NO801378L (en) 1980-11-12
CA1141379A (en) 1983-02-15
GB2051048A (en) 1981-01-14
DE3017564A1 (en) 1980-11-13
BE883217A (en) 1980-09-01
DD150605A5 (en) 1981-09-09
ES8102570A1 (en) 1981-02-16
GB2051048B (en) 1983-01-19
IT1133085B (en) 1986-07-09
CS241025B2 (en) 1986-03-13
CH646971A5 (en) 1984-12-28
NO152607C (en) 1985-10-23
PL224163A1 (en) 1981-02-13
FI68825C (en) 1985-11-11
LU82437A1 (en) 1980-07-31
JPS5615286A (en) 1981-02-14
FI68825B (en) 1985-07-31
SU1151210A3 (en) 1985-04-15
NL8002678A (en) 1980-11-13
AT377261B (en) 1985-02-25
PL124035B1 (en) 1982-12-31
PT71213A (en) 1980-06-01
GR68518B (en) 1982-01-11
FI801512A (en) 1980-11-12
IL59967A0 (en) 1980-07-31
SE8003479L (en) 1980-11-12
ES491896A0 (en) 1981-02-16
SE441747B (en) 1985-11-04
IL59967A (en) 1984-05-31
CS325880A2 (en) 1985-06-13
IT8067719A0 (en) 1980-05-09
DK204680A (en) 1980-11-12
FR2456101B1 (en) 1985-04-05
FR2456101A1 (en) 1980-12-05
NO152607B (en) 1985-07-15
ATA247580A (en) 1984-07-15

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