FI801512A - GEMINAL DIHALOGENDER AV AV CONDENSERS PYRIMIDIN-4-ON-FOERENINGAR FOERFARANDE FOER DERAS FRAMSTAELLNING OCH PHARMACEUTICAL COMPOSITION INNEHAOLLANDE DESSA - Google Patents

GEMINAL DIHALOGENDER AV AV CONDENSERS PYRIMIDIN-4-ON-FOERENINGAR FOERFARANDE FOER DERAS FRAMSTAELLNING OCH PHARMACEUTICAL COMPOSITION INNEHAOLLANDE DESSA

Info

Publication number
FI801512A
FI801512A FI801512A FI801512A FI801512A FI 801512 A FI801512 A FI 801512A FI 801512 A FI801512 A FI 801512A FI 801512 A FI801512 A FI 801512A FI 801512 A FI801512 A FI 801512A
Authority
FI
Finland
Prior art keywords
dihalogender
foereningar
geminal
condensers
pyrimidin
Prior art date
Application number
FI801512A
Other languages
Finnish (fi)
Other versions
FI68825C (en
FI68825B (en
Inventor
Istvan Hermecz
Tibor Breining
Debreczy Lelle Vasvari
Agnes Horvath
Zoltan Meszaros
Istvan Bitter
Jozsef Koekoesi
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of FI801512A publication Critical patent/FI801512A/en
Application granted granted Critical
Publication of FI68825B publication Critical patent/FI68825B/en
Publication of FI68825C publication Critical patent/FI68825C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09BORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B62/00Reactive dyes, i.e. dyes which form covalent bonds with the substrates or which polymerise with themselves

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
FI801512A 1979-05-11 1980-05-09 GEMINALA DIHALOGENDERIV AV AVONDENSERADE PYRIMIDIN-4-ONER VILKA AER MELLANPRODUKTER VID FRAMSTAELLNING AV THERAPEUTIC ANAENDBARA 9-AMINOPYRIDO (1,2-A) PYRIMIDIN-OCH 9-HYDRATSONO-6,, 8,9-P-6,9-8,9-T -A) PYRIMIDINDERIVAT FI68825C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU79CI1932A HU179443B (en) 1979-05-11 1979-05-11 Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines
HUCI001932 1979-05-11

Publications (3)

Publication Number Publication Date
FI801512A true FI801512A (en) 1980-11-12
FI68825B FI68825B (en) 1985-07-31
FI68825C FI68825C (en) 1985-11-11

Family

ID=10994747

Family Applications (1)

Application Number Title Priority Date Filing Date
FI801512A FI68825C (en) 1979-05-11 1980-05-09 GEMINALA DIHALOGENDERIV AV AVONDENSERADE PYRIMIDIN-4-ONER VILKA AER MELLANPRODUKTER VID FRAMSTAELLNING AV THERAPEUTIC ANAENDBARA 9-AMINOPYRIDO (1,2-A) PYRIMIDIN-OCH 9-HYDRATSONO-6,, 8,9-P-6,9-8,9-T -A) PYRIMIDINDERIVAT

Country Status (24)

Country Link
JP (1) JPS5615286A (en)
AT (1) AT377261B (en)
BE (1) BE883217A (en)
CA (1) CA1141379A (en)
CH (1) CH646971A5 (en)
CS (1) CS241025B2 (en)
DD (1) DD150605A5 (en)
DE (1) DE3017564A1 (en)
DK (1) DK204680A (en)
ES (1) ES491896A0 (en)
FI (1) FI68825C (en)
FR (1) FR2456101A1 (en)
GB (1) GB2051048B (en)
GR (1) GR68518B (en)
HU (1) HU179443B (en)
IL (1) IL59967A (en)
IT (1) IT1133085B (en)
LU (1) LU82437A1 (en)
NL (1) NL8002678A (en)
NO (1) NO152607C (en)
PL (1) PL124035B1 (en)
PT (1) PT71213A (en)
SE (1) SE441747B (en)
SU (1) SU1151210A3 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178453B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydrazino-4-oxo-6,7,8,9-tetrahydro-4h-p-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
US4395549A (en) 1981-10-02 1983-07-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones
ES8501397A1 (en) * 1982-08-05 1984-11-16 Erba Farmitalia Amino derivatives of benzylidene-pyrrolo[2,1-b]quinazolines useful for treating conditions of allergic origin
US5158952A (en) * 1988-11-07 1992-10-27 Janssen Pharmaceutica N.V. 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use
UA72189C2 (en) 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Aqueous suspensions of 9-hydroxy-risperidone fatty acid esters provided in submicron form

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT299212B (en) * 1966-11-02 1972-06-12 Chinoin Gyogyszer Es Vegyeszet Process for the preparation of new homopyrimidazole derivatives and their salts
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity

Also Published As

Publication number Publication date
CS325880A2 (en) 1985-06-13
DE3017564A1 (en) 1980-11-13
CA1141379A (en) 1983-02-15
ES8102570A1 (en) 1981-02-16
BE883217A (en) 1980-09-01
DD150605A5 (en) 1981-09-09
IL59967A0 (en) 1980-07-31
PT71213A (en) 1980-06-01
NL8002678A (en) 1980-11-13
FR2456101B1 (en) 1985-04-05
ATA247580A (en) 1984-07-15
CH646971A5 (en) 1984-12-28
NO152607C (en) 1985-10-23
GB2051048A (en) 1981-01-14
SE441747B (en) 1985-11-04
PL224163A1 (en) 1981-02-13
JPS5615286A (en) 1981-02-14
SE8003479L (en) 1980-11-12
IT1133085B (en) 1986-07-09
GB2051048B (en) 1983-01-19
IT8067719A0 (en) 1980-05-09
NO152607B (en) 1985-07-15
GR68518B (en) 1982-01-11
DK204680A (en) 1980-11-12
PL124035B1 (en) 1982-12-31
SU1151210A3 (en) 1985-04-15
AT377261B (en) 1985-02-25
FI68825C (en) 1985-11-11
FR2456101A1 (en) 1980-12-05
FI68825B (en) 1985-07-31
LU82437A1 (en) 1980-07-31
CS241025B2 (en) 1986-03-13
ES491896A0 (en) 1981-02-16
IL59967A (en) 1984-05-31
NO801378L (en) 1980-11-12
HU179443B (en) 1982-10-28

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MM Patent lapsed

Owner name: CHINOIN GYOGUSZER ES VEGYESZETI TERMEKEK