IT1133085B - GEMINAL DIALOGENATED DERIVATIVES OF CONDENSED COMPOUNDS OF PIRIMIDIN 4 ONE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

GEMINAL DIALOGENATED DERIVATIVES OF CONDENSED COMPOUNDS OF PIRIMIDIN 4 ONE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number
IT1133085B
IT1133085B IT67719/80A IT6771980A IT1133085B IT 1133085 B IT1133085 B IT 1133085B IT 67719/80 A IT67719/80 A IT 67719/80A IT 6771980 A IT6771980 A IT 6771980A IT 1133085 B IT1133085 B IT 1133085B
Authority
IT
Italy
Prior art keywords
dialogenated
pirimidin
geminal
derivatives
procedure
Prior art date
Application number
IT67719/80A
Other languages
Italian (it)
Other versions
IT8067719A0 (en
Inventor
Istvan Hermecz
Tibor Breining
Lelle Vasvari
Nata Debreczy
Agnes Horvath
Zoltan Meszaros
Istvan Bitter
Jozsef Kokosi
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of IT8067719A0 publication Critical patent/IT8067719A0/en
Application granted granted Critical
Publication of IT1133085B publication Critical patent/IT1133085B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09BORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B62/00Reactive dyes, i.e. dyes which form covalent bonds with the substrates or which polymerise with themselves

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
IT67719/80A 1979-05-11 1980-05-09 GEMINAL DIALOGENATED DERIVATIVES OF CONDENSED COMPOUNDS OF PIRIMIDIN 4 ONE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IT1133085B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU79CI1932A HU179443B (en) 1979-05-11 1979-05-11 Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines

Publications (2)

Publication Number Publication Date
IT8067719A0 IT8067719A0 (en) 1980-05-09
IT1133085B true IT1133085B (en) 1986-07-09

Family

ID=10994747

Family Applications (1)

Application Number Title Priority Date Filing Date
IT67719/80A IT1133085B (en) 1979-05-11 1980-05-09 GEMINAL DIALOGENATED DERIVATIVES OF CONDENSED COMPOUNDS OF PIRIMIDIN 4 ONE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (24)

Country Link
JP (1) JPS5615286A (en)
AT (1) AT377261B (en)
BE (1) BE883217A (en)
CA (1) CA1141379A (en)
CH (1) CH646971A5 (en)
CS (1) CS241025B2 (en)
DD (1) DD150605A5 (en)
DE (1) DE3017564A1 (en)
DK (1) DK204680A (en)
ES (1) ES491896A0 (en)
FI (1) FI68825C (en)
FR (1) FR2456101A1 (en)
GB (1) GB2051048B (en)
GR (1) GR68518B (en)
HU (1) HU179443B (en)
IL (1) IL59967A (en)
IT (1) IT1133085B (en)
LU (1) LU82437A1 (en)
NL (1) NL8002678A (en)
NO (1) NO152607C (en)
PL (1) PL124035B1 (en)
PT (1) PT71213A (en)
SE (1) SE441747B (en)
SU (1) SU1151210A3 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178453B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydrazino-4-oxo-6,7,8,9-tetrahydro-4h-p-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
US4395549A (en) 1981-10-02 1983-07-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
US5158952A (en) * 1988-11-07 1992-10-27 Janssen Pharmaceutica N.V. 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use
UA72189C2 (en) 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Aqueous suspensions of 9-hydroxy-risperidone fatty acid esters provided in submicron form

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1795769C3 (en) * 1966-11-02 1978-11-02 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt, Budapest 6,7,8,9-Tetrahydro-2H-pyrido [Ua] pyrimidine derivatives, their salts with acids and quaternary methosalts, processes for their preparation and medicaments containing these compounds
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity

Also Published As

Publication number Publication date
IT8067719A0 (en) 1980-05-09
ES8102570A1 (en) 1981-02-16
AT377261B (en) 1985-02-25
SU1151210A3 (en) 1985-04-15
DK204680A (en) 1980-11-12
NO152607C (en) 1985-10-23
BE883217A (en) 1980-09-01
DD150605A5 (en) 1981-09-09
PL224163A1 (en) 1981-02-13
CH646971A5 (en) 1984-12-28
SE441747B (en) 1985-11-04
CA1141379A (en) 1983-02-15
ATA247580A (en) 1984-07-15
CS241025B2 (en) 1986-03-13
JPS5615286A (en) 1981-02-14
SE8003479L (en) 1980-11-12
FR2456101B1 (en) 1985-04-05
GB2051048B (en) 1983-01-19
PT71213A (en) 1980-06-01
NO152607B (en) 1985-07-15
FI68825C (en) 1985-11-11
CS325880A2 (en) 1985-06-13
IL59967A0 (en) 1980-07-31
IL59967A (en) 1984-05-31
GR68518B (en) 1982-01-11
LU82437A1 (en) 1980-07-31
PL124035B1 (en) 1982-12-31
FR2456101A1 (en) 1980-12-05
NL8002678A (en) 1980-11-13
FI801512A7 (en) 1980-11-12
DE3017564A1 (en) 1980-11-13
NO801378L (en) 1980-11-12
GB2051048A (en) 1981-01-14
ES491896A0 (en) 1981-02-16
FI68825B (en) 1985-07-31
HU179443B (en) 1982-10-28

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