NL7908398A - Aminederivaten met farmaceutische werking, werkwijzen ter bereiding daarvan alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten. - Google Patents

Aminederivaten met farmaceutische werking, werkwijzen ter bereiding daarvan alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten. Download PDF

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Publication number
NL7908398A
NL7908398A NL7908398A NL7908398A NL7908398A NL 7908398 A NL7908398 A NL 7908398A NL 7908398 A NL7908398 A NL 7908398A NL 7908398 A NL7908398 A NL 7908398A NL 7908398 A NL7908398 A NL 7908398A
Authority
NL
Netherlands
Prior art keywords
formula
methyl
compounds according
compounds
alk
Prior art date
Application number
NL7908398A
Other languages
English (en)
Dutch (nl)
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NL7908398A publication Critical patent/NL7908398A/nl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/28Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to cyano groups, e.g. cyanoguanidines, dicyandiamides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/40Radicals substituted by oxygen atoms
    • C07D307/42Singly bound oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14Radicals substituted by singly bound hetero atoms other than halogen

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Furan Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NL7908398A 1978-11-16 1979-11-16 Aminederivaten met farmaceutische werking, werkwijzen ter bereiding daarvan alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten. NL7908398A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7844777 1978-11-16
GB7844777 1978-11-16

Publications (1)

Publication Number Publication Date
NL7908398A true NL7908398A (nl) 1980-05-20

Family

ID=10501093

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7908398A NL7908398A (nl) 1978-11-16 1979-11-16 Aminederivaten met farmaceutische werking, werkwijzen ter bereiding daarvan alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.

Country Status (13)

Country Link
US (3) US4264614A (de)
JP (1) JPS5581838A (de)
AU (1) AU538513B2 (de)
BE (1) BE880066A (de)
CH (1) CH644347A5 (de)
DE (1) DE2946332A1 (de)
DK (1) DK489279A (de)
ES (1) ES486071A1 (de)
FR (1) FR2446829A1 (de)
IT (1) IT1164761B (de)
NL (1) NL7908398A (de)
SE (1) SE7909507L (de)
ZA (1) ZA796169B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5021429A (en) * 1977-05-17 1991-06-04 Allen & Hansburys Limited Pharmacologically active aminoalkylphenyl compounds and their use
JPS5681578A (en) * 1979-12-07 1981-07-03 Shionogi & Co Ltd Novel thioalkyl amide derivative
YU53681A (en) * 1980-03-08 1983-12-31 Smith Kline French Lab Process for obtaining 5-dimethylamino-methyl-2-furane methanol
DE3168031D1 (en) * 1980-07-30 1985-02-14 Ici Plc Guanidine derivatives
JPS57102852A (en) * 1980-12-19 1982-06-26 Shionogi & Co Ltd Dicarboxylic acid diamide
DE3245482A1 (de) * 1982-12-08 1984-06-14 Byk-Mallinckrodt Chemische Produkte Gmbh, 4230 Wesel Entschaeumer und verfahren zu ihrer herstellung
US4665172A (en) * 1983-01-28 1987-05-12 Ube Industries, Ltd. Process for producing heterocyclic compound having nitromethylene group as the side chain group
AU581324B2 (en) * 1985-07-05 1989-02-16 Smith Kline & French Laboratories Limited Substituted 6-phenyl-4,5-dihydro pyradazin-3-ones
US4950789A (en) * 1989-01-25 1990-08-21 The Dow Chemical Company Aromatic polyalkyleneoxy polyamines containing amioncarbonyl or aminothiocarbonyl moieties and a compatible mixture of high and low molecular weight polyols made therefrom
CA2349575A1 (en) 1998-11-17 2000-05-25 Nitromed, Inc. Nitrosated and nitrosylated h2 receptor antagonist compounds, compositions and methods of use
EP4196793A1 (de) 2020-08-11 2023-06-21 Université de Strasbourg Auf lebermakrophagen abzielende h2-blocker zur prävention und behandlung von lebererkrankungen und krebs

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1493931A (en) 1974-02-07 1977-11-30 Smith Kline French Lab Guanidines isothioureas and thioureas
ZA774221B (en) 1976-07-28 1978-06-28 Smith Kline French Lab Pharmacologically active compounds
ZA774220B (en) 1976-07-28 1978-06-28 Smith Kline French Lab Pharmacologically active compounds
IL52544A0 (en) * 1976-07-28 1977-10-31 Smith Kline French Lab Alpha,omega-bis (heterocyclicguanidino) alkane derivative
GB1565966A (en) * 1976-08-04 1980-04-23 Allen & Hanburys Ltd Aminoalkyl furan derivatives
DE2719798A1 (de) 1977-05-03 1978-11-16 Uniroyal Ag Hochbelastbarer stahlkord-guertelreifen, insbesondere fuer lastkraftwagen, schwer- und/oder grossfahrzeuge mit einer mindestens einlagigen radialkarkasse, vorzugsweise aus stahlkord, und einer mehrlagigen guertelartigen verstaerkung, welche wenigstens eine faltlage aus stahlkord und wenigstens eine weitere ungefaltete lage aus textilkord aufweist

Also Published As

Publication number Publication date
JPS5581838A (en) 1980-06-20
AU538513B2 (en) 1984-08-16
FR2446829A1 (fr) 1980-08-14
DE2946332A1 (de) 1980-05-29
US4264614A (en) 1981-04-28
AU5291279A (en) 1980-05-22
ES486071A1 (es) 1980-09-01
IT1164761B (it) 1987-04-15
CH644347A5 (fr) 1984-07-31
IT7950847A0 (it) 1979-11-16
FR2446829B1 (de) 1983-04-29
ZA796169B (en) 1981-04-29
US4317819A (en) 1982-03-02
DK489279A (da) 1980-05-17
BE880066A (fr) 1980-03-17
US4366164A (en) 1982-12-28
SE7909507L (sv) 1980-05-17

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BV The patent application has lapsed