MX9803599A - Procedimientos e intermedios para preparar 3-(1-piperazinil)-1,2-benzodisotiazol. - Google Patents

Procedimientos e intermedios para preparar 3-(1-piperazinil)-1,2-benzodisotiazol.

Info

Publication number
MX9803599A
MX9803599A MX9803599A MX9803599A MX9803599A MX 9803599 A MX9803599 A MX 9803599A MX 9803599 A MX9803599 A MX 9803599A MX 9803599 A MX9803599 A MX 9803599A MX 9803599 A MX9803599 A MX 9803599A
Authority
MX
Mexico
Prior art keywords
benzisothiazole
piperazinyl
processes
intermediates
preparing
Prior art date
Application number
MX9803599A
Other languages
English (en)
Inventor
Darrell E Fox
John F Lambert
Terry G Sinay Jr
Stanley W Walinsky
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX9803599A publication Critical patent/MX9803599A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

La presente invencion se refiera a procedimientos para preparacion de 3-(1-piperazinil) -1,2-benzoisotiazol o sus sales farmacéuticamente aceptables y a nuevos intermedios usados en el procedimiento; el 3-(1-piperazinil) -1,2-benzoisotiazol es un intermedio clave util para la preparacion de ziprasidona.
MX9803599A 1995-11-07 1998-05-06 Procedimientos e intermedios para preparar 3-(1-piperazinil)-1,2-benzodisotiazol. MX9803599A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US630195P 1995-11-07 1995-11-07

Publications (1)

Publication Number Publication Date
MX9803599A true MX9803599A (es) 1998-09-30

Family

ID=21720240

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9803599A MX9803599A (es) 1995-11-07 1998-05-06 Procedimientos e intermedios para preparar 3-(1-piperazinil)-1,2-benzodisotiazol.

Country Status (29)

Country Link
US (1) US6111105A (es)
EP (1) EP0874834B1 (es)
JP (1) JP3152938B2 (es)
KR (1) KR100315939B1 (es)
CN (1) CN1071324C (es)
AR (2) AR004279A1 (es)
AT (1) ATE198071T1 (es)
AU (1) AU698443B2 (es)
BR (1) BR9611366A (es)
CA (1) CA2236940C (es)
CO (1) CO4480028A1 (es)
CZ (1) CZ290600B6 (es)
DE (1) DE69611253T2 (es)
DK (1) DK0874834T3 (es)
ES (1) ES2152564T3 (es)
GR (1) GR3035215T3 (es)
HU (1) HU225921B1 (es)
MX (1) MX9803599A (es)
MY (1) MY116579A (es)
NO (1) NO309811B1 (es)
NZ (1) NZ318844A (es)
PE (1) PE17298A1 (es)
PL (1) PL185048B1 (es)
PT (1) PT874834E (es)
RU (1) RU2147302C1 (es)
TR (1) TR199800814T2 (es)
TW (1) TW358807B (es)
WO (1) WO1997017336A1 (es)
ZA (1) ZA969315B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY27668A1 (es) 2002-02-20 2003-10-31 Pfizer Prod Inc Composición de ziprasidona y controles sintéticos
US20040048876A1 (en) * 2002-02-20 2004-03-11 Pfizer Inc. Ziprasidone composition and synthetic controls
EP1628973A2 (en) 2003-10-24 2006-03-01 Teva Pharmaceutical Industries Ltd. Processes for preparation of ziprasidone
US7777037B2 (en) * 2004-10-27 2010-08-17 Dr. Reddy's Laboratories Limited Ziprasidone process
CN105891392A (zh) * 2016-03-29 2016-08-24 北京万全德众医药生物技术有限公司 一种用液相色谱法分离测定盐酸鲁拉西酮中间体有关物质的方法
CN107064323A (zh) * 2016-12-05 2017-08-18 北京万全德众医药生物技术有限公司 一种用液相色谱法分离测定盐酸鲁拉西酮及其有关物质的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4590196A (en) * 1984-08-23 1986-05-20 Bristol-Myers Company Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives
JPH06220030A (ja) * 1993-01-22 1994-08-09 Sumitomo Pharmaceut Co Ltd ３−アミノ−１，２−ベンズイソチアゾール誘導体の製造法
JP3701044B2 (ja) * 1995-04-24 2005-09-28 住友精化株式会社 シアノベンゼンスルフェニルハライドおよびそれを用いる３−置換ベンゾイソチアゾールの製造方法
JP3996228B2 (ja) * 1996-10-11 2007-10-24 住友精化株式会社 ３−ピペラジニルベンズイソチアゾール類の製造法

Also Published As

Publication number Publication date
NO309811B1 (no) 2001-04-02
AR004279A1 (es) 1998-11-04
MY116579A (en) 2004-02-28
HU225921B1 (en) 2008-01-28
HUP9903765A2 (hu) 2000-03-28
CN1071324C (zh) 2001-09-19
CA2236940A1 (en) 1997-05-15
PT874834E (pt) 2001-04-30
US6111105A (en) 2000-08-29
AU698443B2 (en) 1998-10-29
HUP9903765A3 (en) 2001-12-28
KR100315939B1 (ko) 2002-01-16
CZ137898A3 (cs) 1999-03-17
NZ318844A (en) 1999-04-29
CN1201457A (zh) 1998-12-09
KR19990067381A (ko) 1999-08-16
AR032373A2 (es) 2003-11-05
DE69611253D1 (de) 2001-01-18
GR3035215T3 (en) 2001-04-30
ATE198071T1 (de) 2000-12-15
DE69611253T2 (de) 2001-04-05
ES2152564T3 (es) 2001-02-01
JPH10512595A (ja) 1998-12-02
WO1997017336A1 (en) 1997-05-15
EP0874834B1 (en) 2000-12-13
BR9611366A (pt) 1999-02-23
ZA969315B (en) 1998-05-06
NO982051D0 (no) 1998-05-06
CA2236940C (en) 2001-08-21
PL185048B1 (pl) 2003-02-28
NO982051L (no) 1998-07-03
CZ290600B6 (cs) 2002-08-14
AU7092696A (en) 1997-05-29
PE17298A1 (es) 1998-04-16
TW358807B (en) 1999-05-21
CO4480028A1 (es) 1997-07-09
TR199800814T2 (xx) 1998-07-21
EP0874834A1 (en) 1998-11-04
PL326630A1 (en) 1998-10-12
JP3152938B2 (ja) 2001-04-03
RU2147302C1 (ru) 2000-04-10
DK0874834T3 (da) 2001-02-19

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Legal Events

Date Code Title Description
FG Grant or registration
MM Annulment or lapse due to non-payment of fees