CO4480028A1 - Procedimientos e intermedios para preparar 3-(1-piperazinil)-1,2-benzoisotiazol - Google Patents

Procedimientos e intermedios para preparar 3-(1-piperazinil)-1,2-benzoisotiazol

Info

Publication number
CO4480028A1
CO4480028A1 CO96058758A CO96058758A CO4480028A1 CO 4480028 A1 CO4480028 A1 CO 4480028A1 CO 96058758 A CO96058758 A CO 96058758A CO 96058758 A CO96058758 A CO 96058758A CO 4480028 A1 CO4480028 A1 CO 4480028A1
Authority
CO
Colombia
Prior art keywords
procedures
benzoisotiazol
piperazinil
intermediates
prepare
Prior art date
Application number
CO96058758A
Other languages
English (en)
Inventor
E Fox Darrel
John F Lambert
Terry G Signay
W Walinsky Stanley
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CO4480028A1 publication Critical patent/CO4480028A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms

Abstract

LA PRESENTE INVENCION SE REFIERE A PROCEDIMIENTOS PARA LA PREPARACION DE 3-(1-PIPERAZINIL)-1,2-BEN- ZOISOTIAZOL O SUS SALES FARMACEUTICAMENTE ACEPTA- BLES Y A NUEVOS INTERMEDIOS USADOS EN EL PROCEDI- MIENTO. EL 3-(1-PIPERAZINIL)-1,2-BENZOISOTIAZOL ES UN INTERMEDIO CLAVE UTIL PARA LA PREPARACION DE ZIPRASIDONA. FIGURA 1
CO96058758A 1995-11-07 1996-11-07 Procedimientos e intermedios para preparar 3-(1-piperazinil)-1,2-benzoisotiazol CO4480028A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US630195P 1995-11-07 1995-11-07

Publications (1)

Publication Number Publication Date
CO4480028A1 true CO4480028A1 (es) 1997-07-09

Family

ID=21720240

Family Applications (1)

Application Number Title Priority Date Filing Date
CO96058758A CO4480028A1 (es) 1995-11-07 1996-11-07 Procedimientos e intermedios para preparar 3-(1-piperazinil)-1,2-benzoisotiazol

Country Status (29)

Country Link
US (1) US6111105A (es)
EP (1) EP0874834B1 (es)
JP (1) JP3152938B2 (es)
KR (1) KR100315939B1 (es)
CN (1) CN1071324C (es)
AR (2) AR004279A1 (es)
AT (1) ATE198071T1 (es)
AU (1) AU698443B2 (es)
BR (1) BR9611366A (es)
CA (1) CA2236940C (es)
CO (1) CO4480028A1 (es)
CZ (1) CZ290600B6 (es)
DE (1) DE69611253T2 (es)
DK (1) DK0874834T3 (es)
ES (1) ES2152564T3 (es)
GR (1) GR3035215T3 (es)
HU (1) HU225921B1 (es)
MX (1) MX9803599A (es)
MY (1) MY116579A (es)
NO (1) NO309811B1 (es)
NZ (1) NZ318844A (es)
PE (1) PE17298A1 (es)
PL (1) PL185048B1 (es)
PT (1) PT874834E (es)
RU (1) RU2147302C1 (es)
TR (1) TR199800814T2 (es)
TW (1) TW358807B (es)
WO (1) WO1997017336A1 (es)
ZA (1) ZA969315B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY27668A1 (es) 2002-02-20 2003-10-31 Pfizer Prod Inc Composición de ziprasidona y controles sintéticos
US20040048876A1 (en) * 2002-02-20 2004-03-11 Pfizer Inc. Ziprasidone composition and synthetic controls
EP1628973A2 (en) 2003-10-24 2006-03-01 Teva Pharmaceutical Industries Ltd. Processes for preparation of ziprasidone
US7777037B2 (en) * 2004-10-27 2010-08-17 Dr. Reddy's Laboratories Limited Ziprasidone process
CN105891392A (zh) * 2016-03-29 2016-08-24 北京万全德众医药生物技术有限公司 一种用液相色谱法分离测定盐酸鲁拉西酮中间体有关物质的方法
CN107064323A (zh) * 2016-12-05 2017-08-18 北京万全德众医药生物技术有限公司 一种用液相色谱法分离测定盐酸鲁拉西酮及其有关物质的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4590196A (en) * 1984-08-23 1986-05-20 Bristol-Myers Company Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives
JPH06220030A (ja) * 1993-01-22 1994-08-09 Sumitomo Pharmaceut Co Ltd ３−アミノ−１，２−ベンズイソチアゾール誘導体の製造法
JP3701044B2 (ja) * 1995-04-24 2005-09-28 住友精化株式会社 シアノベンゼンスルフェニルハライドおよびそれを用いる３−置換ベンゾイソチアゾールの製造方法
JP3996228B2 (ja) * 1996-10-11 2007-10-24 住友精化株式会社 ３−ピペラジニルベンズイソチアゾール類の製造法

Also Published As

Publication number Publication date
NO309811B1 (no) 2001-04-02
AR004279A1 (es) 1998-11-04
MY116579A (en) 2004-02-28
HU225921B1 (en) 2008-01-28
MX9803599A (es) 1998-09-30
HUP9903765A2 (hu) 2000-03-28
CN1071324C (zh) 2001-09-19
CA2236940A1 (en) 1997-05-15
PT874834E (pt) 2001-04-30
US6111105A (en) 2000-08-29
AU698443B2 (en) 1998-10-29
HUP9903765A3 (en) 2001-12-28
KR100315939B1 (ko) 2002-01-16
CZ137898A3 (cs) 1999-03-17
NZ318844A (en) 1999-04-29
CN1201457A (zh) 1998-12-09
KR19990067381A (ko) 1999-08-16
AR032373A2 (es) 2003-11-05
DE69611253D1 (de) 2001-01-18
GR3035215T3 (en) 2001-04-30
ATE198071T1 (de) 2000-12-15
DE69611253T2 (de) 2001-04-05
ES2152564T3 (es) 2001-02-01
JPH10512595A (ja) 1998-12-02
WO1997017336A1 (en) 1997-05-15
EP0874834B1 (en) 2000-12-13
BR9611366A (pt) 1999-02-23
ZA969315B (en) 1998-05-06
NO982051D0 (no) 1998-05-06
CA2236940C (en) 2001-08-21
PL185048B1 (pl) 2003-02-28
NO982051L (no) 1998-07-03
CZ290600B6 (cs) 2002-08-14
AU7092696A (en) 1997-05-29
PE17298A1 (es) 1998-04-16
TW358807B (en) 1999-05-21
TR199800814T2 (xx) 1998-07-21
EP0874834A1 (en) 1998-11-04
PL326630A1 (en) 1998-10-12
JP3152938B2 (ja) 2001-04-03
RU2147302C1 (ru) 2000-04-10
DK0874834T3 (da) 2001-02-19

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