MX9304868A - 27-hidroxirapamicina, derivados de la misma y composicion farmaceutica que la contiene. - Google Patents

27-hidroxirapamicina, derivados de la misma y composicion farmaceutica que la contiene.

Info

Publication number
MX9304868A
MX9304868A MX9304868A MX9304868A MX9304868A MX 9304868 A MX9304868 A MX 9304868A MX 9304868 A MX9304868 A MX 9304868A MX 9304868 A MX9304868 A MX 9304868A MX 9304868 A MX9304868 A MX 9304868A
Authority
MX
Mexico
Prior art keywords
hydroxyrapamicine
derived
same
pharmaceutical composition
hydroxyrapamycin
Prior art date
Application number
MX9304868A
Other languages
English (en)
Spanish (es)
Inventor
Frances Christy Nelson
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/009,605 external-priority patent/US5256790A/en
Application filed by American Home Prod filed Critical American Home Prod
Publication of MX9304868A publication Critical patent/MX9304868A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Transplantation (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
MX9304868A 1992-08-13 1993-08-11 27-hidroxirapamicina, derivados de la misma y composicion farmaceutica que la contiene. MX9304868A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US93012492A 1992-08-13 1992-08-13
US08/009,605 US5256790A (en) 1992-08-13 1993-01-27 27-hydroxyrapamycin and derivatives thereof

Publications (1)

Publication Number Publication Date
MX9304868A true MX9304868A (es) 1994-05-31

Family

ID=26679675

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9304868A MX9304868A (es) 1992-08-13 1993-08-11 27-hidroxirapamicina, derivados de la misma y composicion farmaceutica que la contiene.

Country Status (12)

Country Link
EP (1) EP0655065B1 (enExample)
JP (1) JPH08501084A (enExample)
AT (1) ATE146179T1 (enExample)
AU (1) AU5007193A (enExample)
CA (1) CA2142288A1 (enExample)
DE (1) DE69306585T2 (enExample)
DK (1) DK0655065T3 (enExample)
ES (1) ES2096941T3 (enExample)
GR (1) GR3022730T3 (enExample)
HU (1) HU221499B (enExample)
MX (1) MX9304868A (enExample)
WO (1) WO1994004540A1 (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5527907A (en) * 1993-11-19 1996-06-18 Abbott Laboratories Macrolide immunomodulators
CA2175215C (en) * 1993-11-19 2008-06-03 Yat Sun Or Semisynthetic analogs of rapamycin (macrolides) being immunomodulators
US6187757B1 (en) 1995-06-07 2001-02-13 Ariad Pharmaceuticals, Inc. Regulation of biological events using novel compounds
KR100400620B1 (ko) * 1995-06-09 2004-02-18 노파르티스 아게 라파마이신유도체
CA2383451A1 (en) 1999-08-24 2001-03-01 Ariad Gene Therapeutics, Inc. 28-epirapalogs
US7067526B1 (en) 1999-08-24 2006-06-27 Ariad Gene Therapeutics, Inc. 28-epirapalogs
PT1478648E (pt) 2002-02-01 2014-07-15 Ariad Pharma Inc Compostos contendo fósforo e suas utilizações
US20040225077A1 (en) 2002-12-30 2004-11-11 Angiotech International Ag Drug delivery from rapid gelling polymer composition
US20110104186A1 (en) 2004-06-24 2011-05-05 Nicholas Valiante Small molecule immunopotentiators and assays for their detection
WO2008060546A2 (en) 2006-11-14 2008-05-22 Ariad Pharmaceuticals, Inc. Oral formulations
US8921642B2 (en) 2008-01-11 2014-12-30 Massachusetts Eye And Ear Infirmary Conditional-stop dimerizable caspase transgenic animals
JP6525971B2 (ja) 2013-06-11 2019-06-05 タカラ バイオ ユーエスエー, インコーポレイテッド タンパク質富化微細小胞、タンパク質富化微細小胞の作製方法及び使用方法
IL278335B2 (en) 2018-05-01 2024-09-01 Revolution Medicines Inc C26-linked rapamycin analogs as mtor inhibitors
FI3788049T3 (fi) 2018-05-01 2023-05-30 Revolution Medicines Inc C40-, c28- ja c-32-liittyneitä rapamysiinianalogeja mtor-estäjinä
AU2022253019A1 (en) * 2021-04-09 2023-11-16 Revolution Medicines, Inc. Synthesis of rapamycin analog compounds
CA3256390A1 (en) 2022-05-25 2023-11-30 Revolution Medicines Inc CANCER TREATMENT METHODS USING AN MTOR INHIBITOR

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH04230389A (ja) * 1990-07-16 1992-08-19 American Home Prod Corp ラパマイシン誘導体
US5102876A (en) * 1991-05-07 1992-04-07 American Home Products Corporation Reduction products of rapamycin

Also Published As

Publication number Publication date
DE69306585D1 (de) 1997-01-23
AU5007193A (en) 1994-03-15
HU9500432D0 (en) 1995-04-28
HUT71614A (en) 1996-01-29
JPH08501084A (ja) 1996-02-06
EP0655065B1 (en) 1996-12-11
ES2096941T3 (es) 1997-03-16
DE69306585T2 (de) 1997-04-17
DK0655065T3 (enExample) 1997-02-24
HU221499B (en) 2002-10-28
WO1994004540A1 (en) 1994-03-03
GR3022730T3 (en) 1997-06-30
EP0655065A1 (en) 1995-05-31
ATE146179T1 (de) 1996-12-15
CA2142288A1 (en) 1994-03-03

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Legal Events

Date Code Title Description
FG Grant or registration
HC Change of company name or juridical status

Owner name: SILGAN TUBES CORPORATION

MM Annulment or lapse due to non-payment of fees