AR001314A1 - Compuesto de ciclohexapeptidil bis-amina, composiciones que lo contienen y metodos de uso. - Google Patents

Compuesto de ciclohexapeptidil bis-amina, composiciones que lo contienen y metodos de uso.

Info

Publication number
AR001314A1
AR001314A1 ARP960105124A AR001314A1 AR 001314 A1 AR001314 A1 AR 001314A1 AR P960105124 A ARP960105124 A AR P960105124A AR 001314 A1 AR001314 A1 AR 001314A1
Authority
AR
Argentina
Prior art keywords
cyclohexapeptidyl
bis
methods
compositions containing
amine compound
Prior art date
Application number
Other languages
English (en)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9603241.2A external-priority patent/GB9603241D0/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of AR001314A1 publication Critical patent/AR001314A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Se describe un compuesto de fórmula (I) que es útil para el tratamiento de infecciones micóticas y para el tratamiento de infecciones causadas porpneumocystis carinii.
ARP960105124 1995-11-09 1996-11-08 Compuesto de ciclohexapeptidil bis-amina, composiciones que lo contienen y metodos de uso. AR001314A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US650595P 1995-11-09 1995-11-09
GBGB9603241.2A GB9603241D0 (en) 1996-02-16 1996-02-16 Cyclohexapeptidyl bisamine compound, compositions containing said compound and methods of use

Publications (1)

Publication Number Publication Date
AR001314A1 true AR001314A1 (es) 1997-10-22

Family

ID=26308720

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP960105124 AR001314A1 (es) 1995-11-09 1996-11-08 Compuesto de ciclohexapeptidil bis-amina, composiciones que lo contienen y metodos de uso.

Country Status (9)

Country Link
EP (1) EP0862579A1 (es)
JP (1) JP2000501076A (es)
AR (1) AR001314A1 (es)
AU (1) AU707664B2 (es)
CA (1) CA2235824A1 (es)
CO (1) CO4770984A1 (es)
HR (1) HRP960521A2 (es)
PE (1) PE16198A1 (es)
WO (1) WO1997017365A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2189500A (en) * 1998-12-16 2000-07-03 Eli Lilly And Company Cyclic peptide antifungal agents having a sugar substituent

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6030944A (en) * 1991-10-01 2000-02-29 Merck & Co., Inc. Cyclohexapeptidyl bisamine compounds
US5378804A (en) * 1993-03-16 1995-01-03 Merck & Co., Inc. Aza cyclohexapeptide compounds
IL109615A (en) * 1993-05-17 2000-12-06 Fujisawa Pharmaceutical Co Cyclic polypeptide derivatives processes for the preparation thereof and pharmaceutical compositions containing the same

Also Published As

Publication number Publication date
PE16198A1 (es) 1998-04-11
WO1997017365A1 (en) 1997-05-15
HRP960521A2 (en) 1998-04-30
JP2000501076A (ja) 2000-02-02
EP0862579A1 (en) 1998-09-09
AU7554096A (en) 1997-05-29
CO4770984A1 (es) 1999-04-30
AU707664B2 (en) 1999-07-15
CA2235824A1 (en) 1997-05-15

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