MX9100345A - Procedimiento para la preparacion de derivados 6-(aminopropionil sustituidos)de forscolina - Google Patents

Procedimiento para la preparacion de derivados 6-(aminopropionil sustituidos)de forscolina

Info

Publication number
MX9100345A
MX9100345A MX9100345A MX9100345A MX9100345A MX 9100345 A MX9100345 A MX 9100345A MX 9100345 A MX9100345 A MX 9100345A MX 9100345 A MX9100345 A MX 9100345A MX 9100345 A MX9100345 A MX 9100345A
Authority
MX
Mexico
Prior art keywords
derivatives
forscolina
aminopropionil
substituted
procedure
Prior art date
Application number
MX9100345A
Other languages
English (en)
Inventor
Noel John De Souza Adolf D Sa
Samba Laximinarayan Kattige
Gulab Bajirao Padwal
Jurgen Blumbach
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of MX9100345A publication Critical patent/MX9100345A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78Ring systems having three or more relevant rings
    • C07D311/92Naphthopyrans; Hydrogenated naphthopyrans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
MX9100345A 1990-07-24 1991-07-23 Procedimiento para la preparacion de derivados 6-(aminopropionil sustituidos)de forscolina MX9100345A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP90114124 1990-07-24

Publications (1)

Publication Number Publication Date
MX9100345A true MX9100345A (es) 1992-02-28

Family

ID=8204249

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9100345A MX9100345A (es) 1990-07-24 1991-07-23 Procedimiento para la preparacion de derivados 6-(aminopropionil sustituidos)de forscolina

Country Status (23)

Country Link
US (1) US5869523A (es)
EP (1) EP0468445B1 (es)
JP (1) JPH04279577A (es)
KR (1) KR0173317B1 (es)
CN (1) CN1033583C (es)
AT (1) ATE132863T1 (es)
AU (1) AU642754B2 (es)
CA (1) CA2047617A1 (es)
CZ (1) CZ281393B6 (es)
DE (1) DE69116251T2 (es)
DK (1) DK0468445T3 (es)
ES (1) ES2082890T3 (es)
FI (1) FI913506A (es)
GR (1) GR3018642T3 (es)
HU (1) HU208966B (es)
IE (1) IE74140B1 (es)
IL (1) IL98914A (es)
MX (1) MX9100345A (es)
MY (1) MY106512A (es)
PL (1) PL167626B1 (es)
RU (1) RU2045523C1 (es)
YU (1) YU48634B (es)
ZA (1) ZA915763B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL98913A0 (en) * 1990-07-24 1992-07-15 Hoechst Ag Process for the preparation of 6-(3-substituted aminopropionyl)7-deacetylforskolin derivatives
PL170900B1 (pl) * 1990-11-01 1997-02-28 Nippon Kayaku Kk Sposób wytwarzania 6-(3-dwumetyloaminopropionylo)-forskolinu PL PL PL
US7334636B2 (en) * 2005-02-08 2008-02-26 Halliburton Energy Services, Inc. Methods of creating high-porosity propped fractures using reticulated foam
US20220079915A1 (en) * 2018-12-29 2022-03-17 Shanghai Archeus Biotech Co., Ltd. Immunosuppressive pharmaceutical composition and application thereof
CN117586217B (zh) * 2024-01-17 2024-03-19 云南省药物研究所 一种基于国产毛喉鞘蕊花的佛司可林制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3623300A1 (de) * 1986-07-11 1988-01-21 Hoechst Ag 7-acyloxy-6-aminoacyloxypolyoxylabdane, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
FR2614891B1 (fr) * 1987-05-04 1991-05-24 Roussel Uclaf Nouveaux derives de la forskoline, leur procede de preparation, leur application comme medicaments, les compositions pharmaceutiques les renfermant ainsi que des intermediaires de leur procede de preparation
EP0447962A1 (en) * 1990-03-17 1991-09-25 Hoechst Aktiengesellschaft Labdanes and process for their preparation
IL98913A0 (en) * 1990-07-24 1992-07-15 Hoechst Ag Process for the preparation of 6-(3-substituted aminopropionyl)7-deacetylforskolin derivatives

Also Published As

Publication number Publication date
YU48634B (sh) 1999-03-04
DK0468445T3 (da) 1996-05-20
ATE132863T1 (de) 1996-01-15
IL98914A0 (en) 1992-07-15
IE912592A1 (en) 1992-01-29
HUT58715A (en) 1992-03-30
US5869523A (en) 1999-02-09
PL291199A1 (en) 1992-03-09
JPH04279577A (ja) 1992-10-05
ZA915763B (en) 1992-04-29
IL98914A (en) 1997-01-10
KR0173317B1 (ko) 1999-02-01
CN1058403A (zh) 1992-02-05
HU912489D0 (en) 1991-12-30
ES2082890T3 (es) 1996-04-01
YU128591A (sh) 1994-09-09
AU642754B2 (en) 1993-10-28
GR3018642T3 (en) 1996-04-30
CA2047617A1 (en) 1992-01-25
DE69116251D1 (de) 1996-02-22
CN1033583C (zh) 1996-12-18
KR920002573A (ko) 1992-02-28
CZ281393B6 (cs) 1996-09-11
FI913506A0 (fi) 1991-07-22
FI913506A (fi) 1992-01-25
AU8120891A (en) 1992-07-02
MY106512A (en) 1995-06-30
HU208966B (en) 1994-02-28
CS231391A3 (en) 1992-02-19
EP0468445B1 (en) 1996-01-10
RU2045523C1 (ru) 1995-10-10
IE74140B1 (en) 1997-07-02
PL167626B1 (pl) 1995-10-31
EP0468445A1 (en) 1992-01-29
DE69116251T2 (de) 1996-07-04

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Legal Events

Date Code Title Description
FG Grant or registration
MM Annulment or lapse due to non-payment of fees