CZ281393B6 - Způsob výroby 6-(substituovaných amino)-propionyl derivátů forskolinu - Google Patents

Způsob výroby 6-(substituovaných amino)-propionyl derivátů forskolinu

Info

Publication number
CZ281393B6
CZ281393B6 CS912313A CS231391A CZ281393B6 CZ 281393 B6 CZ281393 B6 CZ 281393B6 CS 912313 A CS912313 A CS 912313A CS 231391 A CS231391 A CS 231391A CZ 281393 B6 CZ281393 B6 CZ 281393B6
Authority
CZ
Czechia
Prior art keywords
derivatives
propionyloxyforskolin
intermediates
preparing
substituted amino
Prior art date
Application number
CS912313A
Other languages
English (en)
Inventor
Souza Noel John Dr. De
Adolf Dr. D`Sa
Samba Laxminarayan Kattige
Gulab Bajirao Padwal
Jürgen Dr. Blumbach
Original Assignee
Hoechst Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Aktiengesellschaft filed Critical Hoechst Aktiengesellschaft
Publication of CS231391A3 publication Critical patent/CS231391A3/cs
Publication of CZ281393B6 publication Critical patent/CZ281393B6/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/92—Naphthopyrans; Hydrogenated naphthopyrans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Investigating Or Analysing Biological Materials (AREA)

Abstract

Způsob výroby 6-(3-substituovanýchamino)propionyloxyforskoli- nových derivátů obecného vzorce I.ŕ
CS912313A 1990-07-24 1991-07-23 Způsob výroby 6-(substituovaných amino)-propionyl derivátů forskolinu CZ281393B6 (cs)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP90114124 1990-07-24

Publications (2)

Publication Number Publication Date
CS231391A3 CS231391A3 (en) 1992-02-19
CZ281393B6 true CZ281393B6 (cs) 1996-09-11

Family

ID=8204249

Family Applications (1)

Application Number Title Priority Date Filing Date
CS912313A CZ281393B6 (cs) 1990-07-24 1991-07-23 Způsob výroby 6-(substituovaných amino)-propionyl derivátů forskolinu

Country Status (23)

Country Link
US (1) US5869523A (cs)
EP (1) EP0468445B1 (cs)
JP (1) JPH04279577A (cs)
KR (1) KR0173317B1 (cs)
CN (1) CN1033583C (cs)
AT (1) ATE132863T1 (cs)
AU (1) AU642754B2 (cs)
CA (1) CA2047617A1 (cs)
CZ (1) CZ281393B6 (cs)
DE (1) DE69116251T2 (cs)
DK (1) DK0468445T3 (cs)
ES (1) ES2082890T3 (cs)
FI (1) FI913506A7 (cs)
GR (1) GR3018642T3 (cs)
HU (1) HU208966B (cs)
IE (1) IE74140B1 (cs)
IL (1) IL98914A (cs)
MX (1) MX9100345A (cs)
MY (1) MY106512A (cs)
PL (1) PL167626B1 (cs)
RU (1) RU2045523C1 (cs)
YU (1) YU48634B (cs)
ZA (1) ZA915763B (cs)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL98913A0 (en) * 1990-07-24 1992-07-15 Hoechst Ag Process for the preparation of 6-(3-substituted aminopropionyl)7-deacetylforskolin derivatives
PL170900B1 (pl) * 1990-11-01 1997-02-28 Nippon Kayaku Kk Sposób wytwarzania 6-(3-dwumetyloaminopropionylo)-forskolinu PL PL PL
US7334636B2 (en) * 2005-02-08 2008-02-26 Halliburton Energy Services, Inc. Methods of creating high-porosity propped fractures using reticulated foam
EP3903778B1 (en) * 2018-12-29 2025-07-30 Shanghai Archeus Biotech Co., Ltd. Immunosuppressive pharmaceutical composition and application thereof
CN117586217B (zh) * 2024-01-17 2024-03-19 云南省药物研究所 一种基于国产毛喉鞘蕊花的佛司可林制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3623300A1 (de) * 1986-07-11 1988-01-21 Hoechst Ag 7-acyloxy-6-aminoacyloxypolyoxylabdane, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
FR2614891B1 (fr) * 1987-05-04 1991-05-24 Roussel Uclaf Nouveaux derives de la forskoline, leur procede de preparation, leur application comme medicaments, les compositions pharmaceutiques les renfermant ainsi que des intermediaires de leur procede de preparation
EP0447962A1 (en) * 1990-03-17 1991-09-25 Hoechst Aktiengesellschaft Labdanes and process for their preparation
IL98913A0 (en) * 1990-07-24 1992-07-15 Hoechst Ag Process for the preparation of 6-(3-substituted aminopropionyl)7-deacetylforskolin derivatives

Also Published As

Publication number Publication date
HU912489D0 (en) 1991-12-30
KR0173317B1 (ko) 1999-02-01
PL167626B1 (pl) 1995-10-31
CN1058403A (zh) 1992-02-05
IE912592A1 (en) 1992-01-29
EP0468445B1 (en) 1996-01-10
YU48634B (sh) 1999-03-04
FI913506A0 (fi) 1991-07-22
HUT58715A (en) 1992-03-30
EP0468445A1 (en) 1992-01-29
DE69116251D1 (de) 1996-02-22
KR920002573A (ko) 1992-02-28
US5869523A (en) 1999-02-09
ES2082890T3 (es) 1996-04-01
RU2045523C1 (ru) 1995-10-10
GR3018642T3 (en) 1996-04-30
MY106512A (en) 1995-06-30
CA2047617A1 (en) 1992-01-25
PL291199A1 (en) 1992-03-09
FI913506A7 (fi) 1992-01-25
AU8120891A (en) 1992-07-02
ATE132863T1 (de) 1996-01-15
YU128591A (sh) 1994-09-09
DE69116251T2 (de) 1996-07-04
IL98914A0 (en) 1992-07-15
IE74140B1 (en) 1997-07-02
DK0468445T3 (da) 1996-05-20
JPH04279577A (ja) 1992-10-05
CN1033583C (zh) 1996-12-18
HU208966B (en) 1994-02-28
MX9100345A (es) 1992-02-28
CS231391A3 (en) 1992-02-19
ZA915763B (en) 1992-04-29
IL98914A (en) 1997-01-10
AU642754B2 (en) 1993-10-28

Similar Documents

Publication Publication Date Title
DK0553202T3 (da) Fremgangsmåde til fremstilling af imidazo(4,5-c)quinolin-4-aminer
BG41820A3 (en) Method for preparing n- (3- hydroxy- 4- piperidinyl) benzamide derivatives
FI914905L (fi) Menetelmä uusien terapeuttisesti käyttökelpoisten merkaptoasetyyliamidopyrrolo- ja -pyridobentsatsepiinijohdannaisten valmistamiseksi
YU25497A (sh) Postupak za dobijanje sildenafila
ATE269290T1 (de) Benzoylderivate
ES525122A0 (es) Procedimiento para preparar derivados de piridina
MX9603050A (es) Derivados de la 1-h-3-aril-pirrolidin-2,4-diona como agentes pesticidas.
PT723538E (pt) Compostos triciclicos de carbamato uteis para a ainibicao da funcao da proteina g e para o tratamento de doencas proliferativas
PL285248A1 (en) Method of obtaining novel aminophenol derivatives
NO911600D0 (no) Fremgangsmaate for fremstilling av n-(3-fluor-2-fosfonyl-metoksypropyl)-derivater av heterocykliske purin- og pyrimidinbaser.
FI101376B1 (fi) Menetelmä 3-bentsyyliamino-2-fenyylipiperidiinijohdannaisten valmistamiseksi
NO930035L (no) Eksitatoriske aminosyreantagonister
FI915231A7 (fi) Mikrobiologinen menetelmä hydroksyloitujen pyratsiinijohdannaisten valmistamiseksi
CZ282732B6 (cs) Substituované 1,2,3,4-tetrahydrocyklopent/b/indoly, 1,2,3,3a,4,8a-hexahydrocyklopent/b/indoly a příbuzné sloučeniny, meziprodukty a způsob jejich přípravy a jejich použití jako léčiv
YU78092A (sh) Postupak za dobijanje derivata beta-fenilizoserina i njihova primena
DK0526529T3 (da) "Forbedret fremgangsmåde til fremstilling af substituerede indolonderivater"
GR1000156B (el) ΜΕΘΟΔΟΣ ΠΑΡΑΣΚΕΥΗΣ ΝΕΩΝ ΠΑΡΑΓΩΓΩΝ ΤΡΙΚΥΚΛΙΚΩΝ ΑΜΙΝΩΝ ΤΗΣ ΤΕΤΡΑΥΔΡΟ-5,6,7,8ΝΑΦΘΟ[2,3b] ΔΙΥΔΡΟ-2,3 ΦΟΥΡΑΝΗΣ & ΤΗΣ ΤΕΤΡΑΥΔΡΟ-6,7,8,9 5Η-ΒΕΝΖΟΚΥΚΛΟΕΠΤΑ[2,3Β] ΔΙΥΔΡΟ-2,3 ΦΟΥΡΑΝΗΣ.
CZ281393B6 (cs) Způsob výroby 6-(substituovaných amino)-propionyl derivátů forskolinu
AP8800109A0 (en) "Heterocyclic insecticides".
ES2080332T3 (es) Derivados de 2'-fluorofuranosil y nuevo procedimiento de preparacion de nucleosidos de 2'-fluoropirimidina y 2'-fluoropurina.
EE03027B1 (et) Meetod 8-klorokinolooni derivaatide valmistamiseks
BG34610A3 (en) Method for preparating 2', 6'- dialkyl- n- (alkoxymethyl)- 2- chloracetanylides
GR1001309B (el) Μεθοδος παρασκευης παραγωγου ενωσεως της διχλωροανιλινης.
FI97388B (fi) Menetelmä heterosyklisten NMDA-antagonistien valmistamiseksi
FI910159A7 (fi) Menetelmä uusien, terapeuttisesti käyttökelpoisten 9a-hydroksi-3-okso- 4,24(25)-stigmastadieeni-26-happojohdannaisten valmistamiseksi