MX341082B - Formulaciones de pro-emulsion de taxano no acuosas y metodos para hacer y usar las mismas. - Google Patents

Formulaciones de pro-emulsion de taxano no acuosas y metodos para hacer y usar las mismas.

Info

Publication number
MX341082B
MX341082B MX2012012630A MX2012012630A MX341082B MX 341082 B MX341082 B MX 341082B MX 2012012630 A MX2012012630 A MX 2012012630A MX 2012012630 A MX2012012630 A MX 2012012630A MX 341082 B MX341082 B MX 341082B
Authority
MX
Mexico
Prior art keywords
emulsion formulations
pro
making
methods
same
Prior art date
Application number
MX2012012630A
Other languages
English (en)
Other versions
MX2012012630A (es
Inventor
Nabeta Kiichiro
Original Assignee
Teikoku Pharma Usa Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teikoku Pharma Usa Inc filed Critical Teikoku Pharma Usa Inc
Publication of MX2012012630A publication Critical patent/MX2012012630A/es
Publication of MX341082B publication Critical patent/MX341082B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44—Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Dispersion Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se proporcionan formulaciones de pro-emulsión de taxano no acuosas. Las formulaciones de pro-emulsión de las modalidades de la invención incluyen un taxano, un componente de aceite, un componente tensoactivo y, opcionalmente, un componente de solvente no acuoso. También se proporcionan métodos para hacer y usar las formulaciones de pro-emulsión, así como también kits que incluyen las formulaciones de pro-emulsión.
MX2012012630A 2010-05-03 2011-04-29 Formulaciones de pro-emulsion de taxano no acuosas y metodos para hacer y usar las mismas. MX341082B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33070510P 2010-05-03 2010-05-03
PCT/US2011/034586 WO2011139899A2 (en) 2010-05-03 2011-04-29 Non-aqueous taxane pro-emulsion formulations and methods of making and using the same

Publications (2)

Publication Number Publication Date
MX2012012630A MX2012012630A (es) 2013-05-20
MX341082B true MX341082B (es) 2016-08-08

Family

ID=44858719

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012012630A MX341082B (es) 2010-05-03 2011-04-29 Formulaciones de pro-emulsion de taxano no acuosas y metodos para hacer y usar las mismas.

Country Status (21)

Country Link
US (2) US10842770B2 (es)
EP (1) EP2566474B1 (es)
JP (1) JP5824511B2 (es)
KR (1) KR101752944B1 (es)
CN (2) CN102970990A (es)
AP (1) AP3552A (es)
AU (1) AU2011248449B2 (es)
BR (1) BR112012028037A2 (es)
CA (1) CA2798180A1 (es)
CO (1) CO6640232A2 (es)
EA (1) EA027666B1 (es)
ES (1) ES2652509T3 (es)
IL (1) IL222785A0 (es)
MX (1) MX341082B (es)
MY (1) MY167224A (es)
NZ (1) NZ603828A (es)
SG (2) SG10201503234SA (es)
TW (2) TW201526889A (es)
UA (1) UA109275C2 (es)
WO (1) WO2011139899A2 (es)
ZA (1) ZA201208229B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011139899A2 (en) 2010-05-03 2011-11-10 Teikoku Pharma Usa, Inc. Non-aqueous taxane pro-emulsion formulations and methods of making and using the same
ES2687705T3 (es) * 2012-07-19 2018-10-26 Fujifilm Corporation Composición líquida que contiene un principio activo a base de taxano, proceso de producción de la misma y preparación medicinal líquida
JO3685B1 (ar) * 2012-10-01 2020-08-27 Teikoku Pharma Usa Inc صيغ التشتيت الجسيمي للتاكسين غير المائي وطرق استخدامها
CN104720070A (zh) * 2013-12-20 2015-06-24 财团法人食品工业发展研究所 微乳液预浓缩物和微乳液及其制备方法
TWI531318B (zh) 2013-12-20 2016-05-01 財團法人食品工業發展研究所 微乳液預濃縮物和微乳液暨其製備方法
CN106176599A (zh) * 2015-05-06 2016-12-07 江苏天士力帝益药业有限公司 一种卡巴他赛脂肪乳注射剂及其制备方法
JP6292267B2 (ja) * 2016-09-13 2018-03-14 ニプロ株式会社 ドセタキセル製剤
WO2018182039A1 (ja) * 2017-03-31 2018-10-04 テクノガード株式会社 薬物を保持した非水系組成物およびその製造方法
JP2018115178A (ja) * 2018-03-15 2018-07-26 ニプロ株式会社 ドセタキセル製剤

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