MX3055E - Procedimiento para la preparacion de derivados de histidina - Google Patents
Procedimiento para la preparacion de derivados de histidinaInfo
- Publication number
- MX3055E MX3055E MX000050U MX5076U MX3055E MX 3055 E MX3055 E MX 3055E MX 000050 U MX000050 U MX 000050U MX 5076 U MX5076 U MX 5076U MX 3055 E MX3055 E MX 3055E
- Authority
- MX
- Mexico
- Prior art keywords
- hydrogen
- alkyl
- compound
- formula
- preparation
- Prior art date
Links
- 150000002410 histidine derivatives Chemical class 0.000 title abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 5
- 239000001257 hydrogen Substances 0.000 abstract 5
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 5
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 3
- 125000006239 protecting group Chemical group 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 108010016626 Dipeptides Proteins 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
- C07K5/0825—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Glp-amino acid; Derivatives thereof
Abstract
La presente invención se refiere a procedimiento para la preparación de derivados de histidina de la fórmula: (VER FIGURA) en la cual R es hidrógeno o alquilo C1-3'R1 es alquilo o alcoxi(ver gaceta ), C1-3'R2 es hidrógeno, alquilo o alcoxi, C1-3'R3 es higrógeno, alquilo C1-6 o cicloalquilo, C3-6 y R4 es hidrógeno o alquilo, C1-6' caracterizado porque un compuesto de la fórmula II: en donde A e Y son respectivamente un grupo protector o un grupo capaz de formar un enlace de péptido, en primer lugar se acopla con (VER FIGURA) (a) un copuesto de la fórmula III, en donde B es hidrógeno o un grupo protector y X es un grupo capaz de formar un enlace de péptido; o bien (b) un compuesto de la fórmula IV; y en segundo término, el dipéptido resultante se acopla con el otro compuesto, y en seguida se remueven los grupos protectores.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB10144/75A GB1523598A (en) | 1975-03-08 | 1975-03-08 | Tripeptides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX3055E true MX3055E (es) | 1980-03-10 |
Family
ID=9962321
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX000050U MX3055E (es) | 1975-03-08 | 1976-03-08 | Procedimiento para la preparacion de derivados de histidina |
Country Status (32)
| Country | Link |
|---|---|
| US (1) | US4060603A (es) |
| JP (1) | JPS5940144B2 (es) |
| AR (1) | AR208361A1 (es) |
| AT (1) | AT352918B (es) |
| BE (1) | BE839187A (es) |
| CA (1) | CA1059994A (es) |
| CH (1) | CH608484A5 (es) |
| CS (1) | CS197268B2 (es) |
| DE (1) | DE2609154C2 (es) |
| DK (1) | DK97376A (es) |
| EG (1) | EG13624A (es) |
| ES (1) | ES445763A1 (es) |
| FI (1) | FI62823C (es) |
| FR (1) | FR2303559A1 (es) |
| GB (1) | GB1523598A (es) |
| GR (1) | GR59891B (es) |
| HU (1) | HU175652B (es) |
| IE (1) | IE42784B1 (es) |
| IL (1) | IL49122A (es) |
| LU (1) | LU74483A1 (es) |
| MX (1) | MX3055E (es) |
| NL (1) | NL7602257A (es) |
| NO (1) | NO144604C (es) |
| OA (1) | OA05260A (es) |
| PH (1) | PH11727A (es) |
| PL (1) | PL101401B1 (es) |
| PT (1) | PT64853B (es) |
| SE (1) | SE411671B (es) |
| SU (1) | SU619101A3 (es) |
| YU (1) | YU58176A (es) |
| ZA (1) | ZA761062B (es) |
| ZM (1) | ZM2576A1 (es) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5920647B2 (ja) * | 1976-10-01 | 1984-05-15 | 武田薬品工業株式会社 | 注射剤 |
| US4182856A (en) * | 1978-04-25 | 1980-01-08 | Miles Laboratories, Inc. | Reagents for use in binding assays to determine diphenylhydantoin |
| CA1256650A (en) * | 1983-03-25 | 1989-06-27 | Toshinari Tamura | Process of producing 2-azetidinone-4-substituted compounds, and medicaments containing the compounds |
| JPS59195037U (ja) * | 1983-06-14 | 1984-12-25 | 株式会社村上開明堂 | バツクミラ− |
| JPS59195038U (ja) * | 1983-06-14 | 1984-12-25 | 株式会社村上開明堂 | バツクミラ− |
| GB2146026A (en) * | 1983-09-07 | 1985-04-11 | Tanabe Seiyaku Co | Peptides and process for preparing the same |
| FR2622581B1 (fr) * | 1987-11-03 | 1990-02-16 | Inorgan Sa Rech Develop Pharm | Nouveaux derives de l-proline, leur preparation et leurs applications biologiques |
| FR2649110B1 (fr) * | 1989-06-29 | 1994-10-21 | Adir | Nouveaux derives peptidiques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| DK437289D0 (da) * | 1989-09-04 | 1989-09-04 | Hans Bundgaard | Prodrug derivatives of thyrotropin-releasing hormone (trh) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2343035C2 (de) * | 1973-08-25 | 1982-04-01 | Hoechst Ag, 6000 Frankfurt | Pyroglutamyl-histidyl-prolinamide, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel |
| US3959248A (en) * | 1974-04-03 | 1976-05-25 | Merck & Co., Inc. | Analogs of thyrotropin-releasing hormone |
-
1975
- 1975-03-08 GB GB10144/75A patent/GB1523598A/en not_active Expired
-
1976
- 1976-01-01 AR AR262475A patent/AR208361A1/es active
- 1976-02-20 US US05/659,913 patent/US4060603A/en not_active Expired - Lifetime
- 1976-02-20 CA CA246,250A patent/CA1059994A/en not_active Expired
- 1976-02-23 SE SE7602165A patent/SE411671B/xx not_active IP Right Cessation
- 1976-02-24 ZA ZA761062A patent/ZA761062B/xx unknown
- 1976-02-27 PT PT64853A patent/PT64853B/pt unknown
- 1976-02-29 IL IL49122A patent/IL49122A/xx unknown
- 1976-03-02 FI FI760538A patent/FI62823C/fi not_active IP Right Cessation
- 1976-03-02 PH PH18163A patent/PH11727A/en unknown
- 1976-03-03 GR GR50233A patent/GR59891B/el unknown
- 1976-03-03 ZM ZM25/76A patent/ZM2576A1/xx unknown
- 1976-03-03 JP JP51023063A patent/JPS5940144B2/ja not_active Expired
- 1976-03-04 BE BE164854A patent/BE839187A/xx not_active IP Right Cessation
- 1976-03-04 NL NL7602257A patent/NL7602257A/xx not_active Application Discontinuation
- 1976-03-04 ES ES445763A patent/ES445763A1/es not_active Expired
- 1976-03-04 NO NO760741A patent/NO144604C/no unknown
- 1976-03-05 DK DK97376*#A patent/DK97376A/da not_active Application Discontinuation
- 1976-03-05 FR FR7606369A patent/FR2303559A1/fr active Granted
- 1976-03-05 DE DE2609154A patent/DE2609154C2/de not_active Expired
- 1976-03-05 OA OA55754A patent/OA05260A/xx unknown
- 1976-03-05 SU SU762331353A patent/SU619101A3/ru active
- 1976-03-05 LU LU74483A patent/LU74483A1/xx unknown
- 1976-03-05 CH CH282376A patent/CH608484A5/xx not_active IP Right Cessation
- 1976-03-05 PL PL1976187742A patent/PL101401B1/pl unknown
- 1976-03-08 CS CS761513A patent/CS197268B2/cs unknown
- 1976-03-08 IE IE477/76A patent/IE42784B1/en unknown
- 1976-03-08 YU YU00581/76A patent/YU58176A/xx unknown
- 1976-03-08 HU HU76RE580A patent/HU175652B/hu unknown
- 1976-03-08 AT AT169776A patent/AT352918B/de not_active IP Right Cessation
- 1976-03-08 MX MX000050U patent/MX3055E/es unknown
- 1976-03-09 EG EG139/76A patent/EG13624A/xx active
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