DK437289D0 - Prodrug derivatives of thyrotropin-releasing hormone (trh) - Google Patents

Prodrug derivatives of thyrotropin-releasing hormone (trh)

Info

Publication number
DK437289D0
DK437289D0 DK437289A DK437289A DK437289D0 DK 437289 D0 DK437289 D0 DK 437289D0 DK 437289 A DK437289 A DK 437289A DK 437289 A DK437289 A DK 437289A DK 437289 D0 DK437289 D0 DK 437289D0
Authority
DK
Denmark
Prior art keywords
trh
thyrotropin
releasing hormone
product derivatives
derivatives
Prior art date
Application number
DK437289A
Other languages
English (en)
Inventor
Hans Bundgaard
Judi Moess
Original Assignee
Hans Bundgaard
Judi Moess
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hans Bundgaard, Judi Moess filed Critical Hans Bundgaard
Priority to DK437289A priority Critical patent/DK437289D0/da
Publication of DK437289D0 publication Critical patent/DK437289D0/da
Priority to US07/842,181 priority patent/US5405834A/en
Priority to CA002066449A priority patent/CA2066449A1/en
Priority to KR1019920700492A priority patent/KR920703628A/ko
Priority to EP90913468A priority patent/EP0490947A1/en
Priority to JP2512601A priority patent/JPH05500061A/ja
Priority to PCT/DK1990/000228 priority patent/WO1991003487A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • C07K5/0825—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Glp-amino acid; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/10—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH
    • A61P5/12—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH for decreasing, blocking or antagonising the activity of the posterior pituitary hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
DK437289A 1989-09-04 1989-09-04 Prodrug derivatives of thyrotropin-releasing hormone (trh) DK437289D0 (da)

Priority Applications (7)

Application Number Priority Date Filing Date Title
DK437289A DK437289D0 (da) 1989-09-04 1989-09-04 Prodrug derivatives of thyrotropin-releasing hormone (trh)
US07/842,181 US5405834A (en) 1989-09-04 1990-09-03 Prodrug derivatives of thyrotropin-releasing hormone (TRH)
CA002066449A CA2066449A1 (en) 1989-09-04 1990-09-03 Prodrug derivatives of thyrotropin-releasing hormone (trh)
KR1019920700492A KR920703628A (ko) 1989-09-04 1990-09-03 티로트로핀-방출 호르몬(trh)의 프로드러그 유도체
EP90913468A EP0490947A1 (en) 1989-09-04 1990-09-03 Prodrug derivatives of thyrotropin-releasing hormone (trh)
JP2512601A JPH05500061A (ja) 1989-09-04 1990-09-03 甲状腺刺激ホルモン放出ホルモンのプロドラッグ誘導体
PCT/DK1990/000228 WO1991003487A1 (en) 1989-09-04 1990-09-03 Prodrug derivatives of thyrotropin-releasing hormone (trh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK437289A DK437289D0 (da) 1989-09-04 1989-09-04 Prodrug derivatives of thyrotropin-releasing hormone (trh)

Publications (1)

Publication Number Publication Date
DK437289D0 true DK437289D0 (da) 1989-09-04

Family

ID=8132949

Family Applications (1)

Application Number Title Priority Date Filing Date
DK437289A DK437289D0 (da) 1989-09-04 1989-09-04 Prodrug derivatives of thyrotropin-releasing hormone (trh)

Country Status (7)

Country Link
US (1) US5405834A (da)
EP (1) EP0490947A1 (da)
JP (1) JPH05500061A (da)
KR (1) KR920703628A (da)
CA (1) CA2066449A1 (da)
DK (1) DK437289D0 (da)
WO (1) WO1991003487A1 (da)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5543390A (en) * 1990-11-01 1996-08-06 State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University Covalent microparticle-drug conjugates for biological targeting
US5827819A (en) * 1990-11-01 1998-10-27 Oregon Health Sciences University Covalent polar lipid conjugates with neurologically active compounds for targeting
US7045543B2 (en) 2001-11-05 2006-05-16 Enzrel Inc. Covalent conjugates of biologically-active compounds with amino acids and amino acid derivatives for targeting to physiologically-protected sites
WO2003089459A2 (en) * 2002-04-19 2003-10-30 University Of Florida Thyrotropin-releasing hormone analogues and their therapeutic applications
AU2003285200A1 (en) * 2002-11-09 2004-06-03 Nobex Corporation Modified carbamate-containing prodrugs and methods of synthesizing same
US7414076B2 (en) * 2003-06-23 2008-08-19 Neurochem (International) Limited Methods and compositions for treating amyloid-related diseases
US7244764B2 (en) * 2003-06-23 2007-07-17 Neurochem (International) Limited Methods and compositions for treating amyloid-related diseases
US20070010573A1 (en) * 2003-06-23 2007-01-11 Xianqi Kong Methods and compositions for treating amyloid-related diseases
US7462595B2 (en) * 2004-09-17 2008-12-09 Prange Jr Arthur Jergen Methods for treating cancer-related fatigue
BRPI0517790A (pt) * 2004-11-12 2008-10-21 Neurochem Int Ltd métodos e composições fluoradas para tratar doenças relacionadas à amilóide
EP1817305A2 (en) * 2004-11-16 2007-08-15 Neurochem (International) Limited Compounds for the treatment of cns and amyloid associated diseases
EP1836161B1 (en) 2004-12-22 2016-07-20 BHI Limited Partnership Methods and compositions for treating amyloid-related diseases
EP1901763A4 (en) * 2005-03-09 2009-10-21 Roger Williams Hospital THYROTROPIN RELEASE HORMONE ANALOGUES AND METHODS OF USE
US20070232556A1 (en) * 2006-03-31 2007-10-04 Montine Thomas J Methods and compositions for the treatment of neurological diseases and disorders
US20100316626A1 (en) * 2006-08-11 2010-12-16 The Government Of The United States Of America As Represented By The Secretary Methods for treatment and diagnosis of psychiatric disorders
PT3851447T (pt) 2006-10-12 2023-12-11 Bellus Health Inc Métodos, compostos, composições e veículos para administrar ácido 3-amino-1-propanossulfónico
US20110178024A1 (en) 2008-09-29 2011-07-21 Ben Gurion University Of The Negev Research And Development Authority Amyloid beta-peptides and methods of use thereof
JP2020523035A (ja) 2017-06-07 2020-08-06 エーディーアールエックス， インコーポレイテッド タウ凝集阻害剤
US11453701B2 (en) 2017-08-18 2022-09-27 Adrx, Inc. Tau aggregation peptide inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3959248A (en) * 1974-04-03 1976-05-25 Merck & Co., Inc. Analogs of thyrotropin-releasing hormone
GB1523598A (en) * 1975-03-08 1978-09-06 Reckitt & Colmann Prod Ltd Tripeptides
CA1256650A (en) * 1983-03-25 1989-06-27 Toshinari Tamura Process of producing 2-azetidinone-4-substituted compounds, and medicaments containing the compounds

Also Published As

Publication number Publication date
WO1991003487A1 (en) 1991-03-21
US5405834A (en) 1995-04-11
KR920703628A (ko) 1992-12-18
CA2066449A1 (en) 1991-03-05
EP0490947A1 (en) 1992-06-24
JPH05500061A (ja) 1993-01-14

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