MX2021004083A - Procedimiento para la preparacion de derivados de imidazol sustituidos. - Google Patents

Procedimiento para la preparacion de derivados de imidazol sustituidos.

Info

Publication number
MX2021004083A
MX2021004083A MX2021004083A MX2021004083A MX2021004083A MX 2021004083 A MX2021004083 A MX 2021004083A MX 2021004083 A MX2021004083 A MX 2021004083A MX 2021004083 A MX2021004083 A MX 2021004083A MX 2021004083 A MX2021004083 A MX 2021004083A
Authority
MX
Mexico
Prior art keywords
preparing substituted
imidazole derivatives
substituted imidazole
ivb
formula
Prior art date
Application number
MX2021004083A
Other languages
English (en)
Inventor
Rüdiger Fischer
Matthieu Willot
Dominik Hager
Laura Hoffmeister
Marc Mosrin
David Wilcke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of MX2021004083A publication Critical patent/MX2021004083A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F3/00Compounds containing elements of Groups 2 or 12 of the Periodic System
    • C07F3/06Zinc compounds

Abstract

La presente invención se refiere a un procedimiento para la preparación de derivados de imidazol sustituidos de la fórmula (II) (ver Fórmula) a partir de compuestos de la fórmula (I) (ver Fórmula) a través de etapas intermedias de la fórmula (IVa) o (IVb) (ver Fórmulas), en la que los elementos estructurales dados en las fórmulas (I), (II), (IVa) y (IVb) tienen los significados dados en la descripción. La invención también se refiere a las etapas intermedias de las fórmulas (IVa) y (IVb).
MX2021004083A 2018-10-11 2019-10-09 Procedimiento para la preparacion de derivados de imidazol sustituidos. MX2021004083A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP18199890 2018-10-11
PCT/EP2019/077307 WO2020074560A1 (de) 2018-10-11 2019-10-09 Verfahren zur herstellung substituierter imidazolderivate

Publications (1)

Publication Number Publication Date
MX2021004083A true MX2021004083A (es) 2021-06-04

Family

ID=63833927

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2021004083A MX2021004083A (es) 2018-10-11 2019-10-09 Procedimiento para la preparacion de derivados de imidazol sustituidos.

Country Status (12)

Country Link
US (1) US11479565B2 (es)
EP (1) EP3864016B1 (es)
JP (1) JP7448531B2 (es)
KR (1) KR20210075127A (es)
CN (1) CN112805286A (es)
BR (1) BR112021005368A2 (es)
DK (1) DK3864016T3 (es)
ES (1) ES2930222T3 (es)
IL (1) IL282034B2 (es)
MX (1) MX2021004083A (es)
TW (1) TWI820231B (es)
WO (1) WO2020074560A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPWO2022250069A1 (es) * 2021-05-26 2022-12-01

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4125726A (en) 1977-03-11 1978-11-14 Hoffmann-La Roche Inc. Imidazo[1,5-a][1,4]benzodiazepines
GB0310726D0 (en) 2003-05-09 2003-06-11 Merck Sharp & Dohme Therapeutic agents
US20080280926A1 (en) 2003-12-16 2008-11-13 Palle Venkata P Phosphodiesterase Inhibitors
GB0612428D0 (en) 2006-06-22 2006-08-02 Prolysis Ltd Antibacterial agents
JP2012144455A (ja) * 2011-01-07 2012-08-02 Idemitsu Kosan Co Ltd イミダゾール化合物の製造方法、およびイミダゾール化合物
CN103443081A (zh) * 2011-01-07 2013-12-11 出光兴产株式会社 咪唑化合物的制造方法、咪唑化合物、咪唑系化合物、有机金属络合物、有机电致发光元件用材料、有机电致发光元件、显示装置以及照明装置
KR101958177B1 (ko) 2011-04-21 2019-03-15 오리온 코포레이션 안드로겐 수용체 조절성 카복스아미드
BR112014018990A8 (pt) 2012-04-20 2017-07-11 Gilead Sciences Inc Derivados de ácido benzotiazol-6-il acético e seu uso para tratamento de uma infecção
EP2857396B1 (en) 2012-05-31 2018-11-21 Sumitomo Chemical Co., Ltd Fused heterocyclic compounds for pest control
ME03016B (me) 2012-11-14 2018-10-20 Teijin Pharma Ltd Derivat piridina
RU2659219C2 (ru) 2013-02-28 2018-06-29 Эйсай Ар Энд Ди Менеджмент Ко., Лтд. ТЕТРАГИДРОИМИДАЗО[1,5-d][1,4]ОКСАЗЕПИНОВОЕ ПРОИЗВОДНОЕ
WO2016039444A1 (ja) 2014-09-12 2016-03-17 日本農薬株式会社 イミダゾピリダジン化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法
BR112017009454B1 (pt) 2014-11-07 2022-05-03 Syngenta Participations Ag Composto, composição pesticida, método para controle de pragas e método para a proteção de material de propagação de plantas do ataque por pragas
US10351532B2 (en) 2014-12-29 2019-07-16 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Small molecule inhibitors of lactate dehydrogenase and methods of use thereof
FI3481805T3 (fi) 2016-07-05 2023-04-25 Bayer Cropscience Ag Menetelmä halogenoitujen pyridiinijohdannaisten valmistamiseksi
DK3500568T3 (da) * 2016-08-16 2020-12-14 Bayer Cropscience Ag Fremgangsmåde til fremstilling af 2-(3,6-dihalopyridin-2-yl)-3h-imidazol[4,5-c]pyridinderivater og beslægtede forbindelser ved hjælp af omsætning af 3h-imidazol[4,5-c]pyridinderivatet med en metalorganisk zink-amin base
KR102471278B1 (ko) * 2016-09-14 2022-11-25 바이엘 크롭사이언스 악티엔게젤샤프트 할로겐화 바이사이클릭 화합물의 제조 방법
JP7101177B2 (ja) 2017-01-10 2022-07-14 バイエル・アクチエンゲゼルシヤフト 有害生物防除剤としてのヘテロサイクレン誘導体
US11083199B2 (en) * 2017-01-10 2021-08-10 Bayer Aktiengesellschaft Heterocycle derivatives as pesticides
TWI762568B (zh) 2017-02-06 2022-05-01 德商拜耳作物科學股份有限公司 製備鹵化咪唑並吡啶衍生物之方法

Also Published As

Publication number Publication date
TW202028200A (zh) 2020-08-01
BR112021005368A2 (pt) 2021-06-15
TWI820231B (zh) 2023-11-01
IL282034B2 (en) 2024-02-01
JP2022512645A (ja) 2022-02-07
US11479565B2 (en) 2022-10-25
EP3864016A1 (de) 2021-08-18
EP3864016B1 (de) 2022-09-14
IL282034B1 (en) 2023-10-01
DK3864016T3 (da) 2022-10-31
ES2930222T3 (es) 2022-12-09
WO2020074560A1 (de) 2020-04-16
IL282034A (en) 2021-05-31
JP7448531B2 (ja) 2024-03-12
CN112805286A (zh) 2021-05-14
US20210380611A1 (en) 2021-12-09
KR20210075127A (ko) 2021-06-22

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