MX2021004081A - Procedimiento para la preparacion de derivados de imidazol. - Google Patents

Procedimiento para la preparacion de derivados de imidazol.

Info

Publication number
MX2021004081A
MX2021004081A MX2021004081A MX2021004081A MX2021004081A MX 2021004081 A MX2021004081 A MX 2021004081A MX 2021004081 A MX2021004081 A MX 2021004081A MX 2021004081 A MX2021004081 A MX 2021004081A MX 2021004081 A MX2021004081 A MX 2021004081A
Authority
MX
Mexico
Prior art keywords
sup
imidazole derivatives
preparing imidazole
iiib
iiia
Prior art date
Application number
MX2021004081A
Other languages
English (en)
Inventor
Rüdiger Fischer
Matthieu Willot
Dominik Hager
Laura Hoffmeister
Marc Mosrin
David Wilcke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of MX2021004081A publication Critical patent/MX2021004081A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Epoxy Resins (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

La presente invención se refiere a un procedimiento para la preparación de derivados de imidazol de la fórmula (II) a partir de compuestos de estructura Q-H a través de intermedios de la fórmula (IIIa) o (IIIb) (ver Fórmulas) en donde Q representa un elemento estructural (ver Fórmula) en donde el símbolo # indica el enlace con el resto de la molécula y A, Q1, Q2, Q3, Q4, Q5, Q6 y Q7, y R2, W, V e Y tienen los significados dados en la descripción.
MX2021004081A 2018-10-11 2019-10-09 Procedimiento para la preparacion de derivados de imidazol. MX2021004081A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP18199885 2018-10-11
PCT/EP2019/077304 WO2020074558A1 (de) 2018-10-11 2019-10-09 Verfahren zur herstellung von imidazolderivaten

Publications (1)

Publication Number Publication Date
MX2021004081A true MX2021004081A (es) 2021-06-04

Family

ID=63833924

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2021004081A MX2021004081A (es) 2018-10-11 2019-10-09 Procedimiento para la preparacion de derivados de imidazol.

Country Status (13)

Country Link
US (1) US20220009930A1 (es)
EP (1) EP3864015B1 (es)
JP (1) JP2022512640A (es)
KR (1) KR20210074318A (es)
CN (1) CN112867713B (es)
BR (1) BR112021005723A2 (es)
DK (1) DK3864015T3 (es)
ES (1) ES2951539T3 (es)
FI (1) FI3864015T3 (es)
IL (1) IL282036B2 (es)
MX (1) MX2021004081A (es)
TW (1) TWI820232B (es)
WO (1) WO2020074558A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112022026904A2 (pt) 2020-07-02 2023-01-24 Bayer Ag Derivados de heterocicleno como agentes de controle de pragas

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0212048D0 (en) 2002-05-24 2002-07-03 Merck Sharp & Dohme Therapeutic agents
US7858649B2 (en) 2005-10-14 2010-12-28 Neurosearch A/S Imidazole derivatives and their use for modulating the GABAA receptor complex
WO2010083145A1 (en) 2009-01-16 2010-07-22 Merck Sharp & Dohme Corp. IMIDAZO[1,2-a]PYRIDINES AND IMIDAZO[1,2-b]PYRIDAZINES AS MARK INHIBITORS
WO2013066729A1 (en) 2011-10-31 2013-05-10 Merck Sharp & Dohme Corp. Aminopyrimidinones as interleukin receptor-associated kinase inhibitors
ES2707305T3 (es) 2012-12-20 2019-04-03 Merck Sharp & Dohme Imidazopiridinas sustituidas como inhibidores de HDM2
BR112016001954A2 (pt) 2013-07-31 2017-08-01 Gilead Sciences Inc composto, composição farmacêutica, e, método para tratar uma doença ou condição
MX2019001917A (es) * 2016-08-16 2019-07-15 Bayer Cropscience Ag Metodo para producir derivados de piridina 2-(3,6-dihalopyridin-2- yl)-3h-imidazol[4,5-c] y compuestos relacionados por reaccion del derivado de piridina 3h-imidazol[4,5-c] con una base organometalica de zinc-amina.
GB201614314D0 (en) 2016-08-22 2016-10-05 Discuva Ltd Antibiotic compounds
MX2019008229A (es) * 2017-01-10 2019-10-24 Bayer Ag Derivados heterociclicos como agentes de control de plagas.
CN110312718B (zh) * 2017-01-10 2023-02-28 拜耳公司 作为害虫防治剂的杂环烯衍生物

Also Published As

Publication number Publication date
EP3864015A1 (de) 2021-08-18
TWI820232B (zh) 2023-11-01
FI3864015T3 (fi) 2023-07-26
EP3864015B1 (de) 2023-05-10
IL282036A (en) 2021-05-31
JP2022512640A (ja) 2022-02-07
IL282036B2 (en) 2024-03-01
ES2951539T3 (es) 2023-10-23
KR20210074318A (ko) 2021-06-21
DK3864015T3 (da) 2023-07-31
IL282036B1 (en) 2023-11-01
US20220009930A1 (en) 2022-01-13
CN112867713A (zh) 2021-05-28
BR112021005723A2 (pt) 2021-06-22
WO2020074558A1 (de) 2020-04-16
TW202028201A (zh) 2020-08-01
CN112867713B (zh) 2023-05-05

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