MX2021004081A - Procedimiento para la preparacion de derivados de imidazol. - Google Patents
Procedimiento para la preparacion de derivados de imidazol.Info
- Publication number
- MX2021004081A MX2021004081A MX2021004081A MX2021004081A MX2021004081A MX 2021004081 A MX2021004081 A MX 2021004081A MX 2021004081 A MX2021004081 A MX 2021004081A MX 2021004081 A MX2021004081 A MX 2021004081A MX 2021004081 A MX2021004081 A MX 2021004081A
- Authority
- MX
- Mexico
- Prior art keywords
- sup
- imidazole derivatives
- preparing imidazole
- iiib
- iiia
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Epoxy Resins (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
La presente invención se refiere a un procedimiento para la preparación de derivados de imidazol de la fórmula (II) a partir de compuestos de estructura Q-H a través de intermedios de la fórmula (IIIa) o (IIIb) (ver Fórmulas) en donde Q representa un elemento estructural (ver Fórmula) en donde el símbolo # indica el enlace con el resto de la molécula y A, Q1, Q2, Q3, Q4, Q5, Q6 y Q7, y R2, W, V e Y tienen los significados dados en la descripción.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP18199885 | 2018-10-11 | ||
PCT/EP2019/077304 WO2020074558A1 (de) | 2018-10-11 | 2019-10-09 | Verfahren zur herstellung von imidazolderivaten |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2021004081A true MX2021004081A (es) | 2021-06-04 |
Family
ID=63833924
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2021004081A MX2021004081A (es) | 2018-10-11 | 2019-10-09 | Procedimiento para la preparacion de derivados de imidazol. |
Country Status (13)
Country | Link |
---|---|
US (1) | US20220009930A1 (es) |
EP (1) | EP3864015B1 (es) |
JP (1) | JP2022512640A (es) |
KR (1) | KR20210074318A (es) |
CN (1) | CN112867713B (es) |
BR (1) | BR112021005723A2 (es) |
DK (1) | DK3864015T3 (es) |
ES (1) | ES2951539T3 (es) |
FI (1) | FI3864015T3 (es) |
IL (1) | IL282036B2 (es) |
MX (1) | MX2021004081A (es) |
TW (1) | TWI820232B (es) |
WO (1) | WO2020074558A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR112022026904A2 (pt) | 2020-07-02 | 2023-01-24 | Bayer Ag | Derivados de heterocicleno como agentes de controle de pragas |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0212048D0 (en) | 2002-05-24 | 2002-07-03 | Merck Sharp & Dohme | Therapeutic agents |
US7858649B2 (en) | 2005-10-14 | 2010-12-28 | Neurosearch A/S | Imidazole derivatives and their use for modulating the GABAA receptor complex |
WO2010083145A1 (en) | 2009-01-16 | 2010-07-22 | Merck Sharp & Dohme Corp. | IMIDAZO[1,2-a]PYRIDINES AND IMIDAZO[1,2-b]PYRIDAZINES AS MARK INHIBITORS |
WO2013066729A1 (en) | 2011-10-31 | 2013-05-10 | Merck Sharp & Dohme Corp. | Aminopyrimidinones as interleukin receptor-associated kinase inhibitors |
ES2707305T3 (es) | 2012-12-20 | 2019-04-03 | Merck Sharp & Dohme | Imidazopiridinas sustituidas como inhibidores de HDM2 |
BR112016001954A2 (pt) | 2013-07-31 | 2017-08-01 | Gilead Sciences Inc | composto, composição farmacêutica, e, método para tratar uma doença ou condição |
MX2019001917A (es) * | 2016-08-16 | 2019-07-15 | Bayer Cropscience Ag | Metodo para producir derivados de piridina 2-(3,6-dihalopyridin-2- yl)-3h-imidazol[4,5-c] y compuestos relacionados por reaccion del derivado de piridina 3h-imidazol[4,5-c] con una base organometalica de zinc-amina. |
GB201614314D0 (en) | 2016-08-22 | 2016-10-05 | Discuva Ltd | Antibiotic compounds |
MX2019008229A (es) * | 2017-01-10 | 2019-10-24 | Bayer Ag | Derivados heterociclicos como agentes de control de plagas. |
CN110312718B (zh) * | 2017-01-10 | 2023-02-28 | 拜耳公司 | 作为害虫防治剂的杂环烯衍生物 |
-
2019
- 2019-10-09 KR KR1020217013665A patent/KR20210074318A/ko unknown
- 2019-10-09 DK DK19780272.1T patent/DK3864015T3/da active
- 2019-10-09 WO PCT/EP2019/077304 patent/WO2020074558A1/de unknown
- 2019-10-09 EP EP19780272.1A patent/EP3864015B1/de active Active
- 2019-10-09 TW TW108136617A patent/TWI820232B/zh active
- 2019-10-09 ES ES19780272T patent/ES2951539T3/es active Active
- 2019-10-09 CN CN201980066392.2A patent/CN112867713B/zh active Active
- 2019-10-09 FI FIEP19780272.1T patent/FI3864015T3/fi active
- 2019-10-09 US US17/283,661 patent/US20220009930A1/en active Pending
- 2019-10-09 MX MX2021004081A patent/MX2021004081A/es unknown
- 2019-10-09 JP JP2021519568A patent/JP2022512640A/ja active Pending
- 2019-10-09 BR BR112021005723-4A patent/BR112021005723A2/pt unknown
- 2019-10-09 IL IL282036A patent/IL282036B2/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP3864015A1 (de) | 2021-08-18 |
TWI820232B (zh) | 2023-11-01 |
FI3864015T3 (fi) | 2023-07-26 |
EP3864015B1 (de) | 2023-05-10 |
IL282036A (en) | 2021-05-31 |
JP2022512640A (ja) | 2022-02-07 |
IL282036B2 (en) | 2024-03-01 |
ES2951539T3 (es) | 2023-10-23 |
KR20210074318A (ko) | 2021-06-21 |
DK3864015T3 (da) | 2023-07-31 |
IL282036B1 (en) | 2023-11-01 |
US20220009930A1 (en) | 2022-01-13 |
CN112867713A (zh) | 2021-05-28 |
BR112021005723A2 (pt) | 2021-06-22 |
WO2020074558A1 (de) | 2020-04-16 |
TW202028201A (zh) | 2020-08-01 |
CN112867713B (zh) | 2023-05-05 |
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