MX2020002347A - Uso de principios activos refrescantes fisiologicos y agentes que contienen dichos principios activos. - Google Patents

Uso de principios activos refrescantes fisiologicos y agentes que contienen dichos principios activos.

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Publication number
MX2020002347A
MX2020002347A MX2020002347A MX2020002347A MX2020002347A MX 2020002347 A MX2020002347 A MX 2020002347A MX 2020002347 A MX2020002347 A MX 2020002347A MX 2020002347 A MX2020002347 A MX 2020002347A MX 2020002347 A MX2020002347 A MX 2020002347A
Authority
MX
Mexico
Prior art keywords
active ingredients
compositions
physiological cooling
modulation
compounds
Prior art date
Application number
MX2020002347A
Other languages
English (en)
Inventor
Martin Weisel
Thomas Subkowski
Claus Bollschweiler
Michael Backes
Arnold Machinek
Benoît Join
Jekaterina Ongouta
Rahim Brodhage
Hubert Loges
Susanne Mundt
Tom Somers
Jens Wittenberg
Wolfgang Siegel
Ralf Pelzer
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of MX2020002347A publication Critical patent/MX2020002347A/es

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    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
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    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
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    • A23G3/00—Sweetmeats; Confectionery; Marzipan; Coated or filled products
    • A23G3/34—Sweetmeats, confectionery or marzipan; Processes for the preparation thereof
    • A23G3/36—Sweetmeats, confectionery or marzipan; Processes for the preparation thereof characterised by the composition containing organic or inorganic compounds
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    • A23L27/88—Taste or flavour enhancing agents
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    • A23L29/00—Foods or foodstuffs containing additives; Preparation or treatment thereof
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    • A61K31/36—Compounds containing methylenedioxyphenyl groups, e.g. sesamin
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • C07C323/39—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
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    • C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract

La invención se refiere principalmente a procedimientos para la modulación, preferentemente para la modulación in vitro y/o in vivo, del receptor de mentol frío TRPM8, en donde el receptor se pone en contacto con al menos un modulador que se selecciona del grupo que consiste en los compuestos de tipo estructural 1 descritos en el presente documento. La presente invención se refiere, además, a usos y composiciones correspondientes que comprenden tales compuestos.
MX2020002347A 2017-08-31 2018-08-31 Uso de principios activos refrescantes fisiologicos y agentes que contienen dichos principios activos. MX2020002347A (es)

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EP3675809A1 (de) 2020-07-08
ES2967435T3 (es) 2024-04-30
US11434220B2 (en) 2022-09-06
CN111343963B (zh) 2023-09-12
CN111343963A (zh) 2020-06-26
WO2019043164A1 (de) 2019-03-07
US20200190052A1 (en) 2020-06-18
JP2020531552A (ja) 2020-11-05
JP7231617B2 (ja) 2023-03-01
BR112020003942A2 (pt) 2020-09-08

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