JPS54112882A - Preparation of pyrimidine derivative - Google Patents

Preparation of pyrimidine derivative

Info

Publication number
JPS54112882A
JPS54112882A JP2014478A JP2014478A JPS54112882A JP S54112882 A JPS54112882 A JP S54112882A JP 2014478 A JP2014478 A JP 2014478A JP 2014478 A JP2014478 A JP 2014478A JP S54112882 A JPS54112882 A JP S54112882A
Authority
JP
Japan
Prior art keywords
pyrimidine derivative
hydrocarbon group
formula
preparation
trithiocyclopropenium
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2014478A
Other languages
Japanese (ja)
Other versions
JPS5512016B2 (en
Inventor
Zenichi Yoshida
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mitsubishi Kasei Corp
Original Assignee
Mitsubishi Kasei Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Kasei Corp filed Critical Mitsubishi Kasei Corp
Priority to JP2014478A priority Critical patent/JPS54112882A/en
Publication of JPS54112882A publication Critical patent/JPS54112882A/en
Publication of JPS5512016B2 publication Critical patent/JPS5512016B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Plural Heterocyclic Compounds (AREA)

Abstract

PURPOSE: To prepare a pyrimidine derivative useful as pesticides, pharmaceuticals, etc., by reacting trithiocyclopropenium salt with an amine selected from urea, thiourea and amidines.
CONSTITUTION: A pyrimidine derivative of formula III (R1 is hydrocarbon group, heterocyclic group; R3 is H, hydrocarbon group, amino, alkoxy, thioalkoxy, OH, mercapto) is prepared by reacting a trithiocyclopropenium salt of formula I (X- is anion) with an amine selected from urea, thiourea, and amidines of formula II (R2 is H, hydrocarbon group, amino, alkoxy, thioalkoxy), in a solvent such as CH2Cl2, CHCl3, etc., in the presence of metal alkoxide such as t-butoxy potassium, etc., at 0W100°C for 0.5W5 hours.
COPYRIGHT: (C)1979,JPO&Japio
JP2014478A 1978-02-23 1978-02-23 Preparation of pyrimidine derivative Granted JPS54112882A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2014478A JPS54112882A (en) 1978-02-23 1978-02-23 Preparation of pyrimidine derivative

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2014478A JPS54112882A (en) 1978-02-23 1978-02-23 Preparation of pyrimidine derivative

Publications (2)

Publication Number Publication Date
JPS54112882A true JPS54112882A (en) 1979-09-04
JPS5512016B2 JPS5512016B2 (en) 1980-03-29

Family

ID=12018945

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014478A Granted JPS54112882A (en) 1978-02-23 1978-02-23 Preparation of pyrimidine derivative

Country Status (1)

Country Link
JP (1) JPS54112882A (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992006965A1 (en) * 1990-10-19 1992-04-30 Ici Australia Operations Proprietary Limited Herbicidal sulfonylurea derivatives
WO1993010103A1 (en) * 1990-05-17 1993-05-27 Ici Australia Operations Proprietary Limited Herbicidal sulfonyluria derivatives
JP2015205871A (en) * 2009-11-20 2015-11-19 シムライズ アーゲー Use of physiological cold sense active ingredient, and agent containing such active ingredient
US11434220B2 (en) 2017-08-31 2022-09-06 Basf Se Use of physiological cooling active ingredients, and compositions comprising such active ingredients

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57164236U (en) * 1981-04-09 1982-10-16

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1993010103A1 (en) * 1990-05-17 1993-05-27 Ici Australia Operations Proprietary Limited Herbicidal sulfonyluria derivatives
WO1992006965A1 (en) * 1990-10-19 1992-04-30 Ici Australia Operations Proprietary Limited Herbicidal sulfonylurea derivatives
JP2015205871A (en) * 2009-11-20 2015-11-19 シムライズ アーゲー Use of physiological cold sense active ingredient, and agent containing such active ingredient
US9718839B2 (en) 2009-11-20 2017-08-01 Symrise Ag Use of physiological cooling active ingredients, and agents containing such active ingredients
US10584134B2 (en) 2009-11-20 2020-03-10 Symrise Ag Use of physiological cooling active ingredients, and agents containing such active ingredients
US11434220B2 (en) 2017-08-31 2022-09-06 Basf Se Use of physiological cooling active ingredients, and compositions comprising such active ingredients

Also Published As

Publication number Publication date
JPS5512016B2 (en) 1980-03-29

Similar Documents

Publication Publication Date Title
JPS57203072A (en) 4-anilinopyrimidine derivative, its preparation, antidepressant comprising it as active ingredient
JPS5444660A (en) Heterocyclic compound and its preparation
JPS54112882A (en) Preparation of pyrimidine derivative
IE41052B1 (en) Crop protection composition and method of application, whereby the drift of spraying liquids may be reduced
JPS57136579A (en) Thiazolylurea derivative, its preparation, and pharmaceutical composition containing the same
JPS57165387A (en) Prparation of fluoran derivative
JPS5762254A (en) Preparation of sulfur-containing compound
JPS5655359A (en) Halogenated alpha-amino acid, and its preparation
JPS5535067A (en) Novel urea derivative and its preparation
JPS57146786A (en) Optically active borane compound and preparation of optically active compound using the same
JPS57120600A (en) Nitrosourea derivative and its preparation
JPS57197256A (en) Novel cyclohexanecarboxamide derivative and its preparation
JPS56120662A (en) Novel nitrosourea derivative and its preparation
JPS5587777A (en) Pyrimidine derivative, its preparation and antitumorigenic agent
JPS562951A (en) Preparation of 2-cyanophenol derivative
JPS54145631A (en) Preparation of 2-cyanophenol derivative
JPS5759858A (en) Substituted thiobiuret derivative
JPS5444632A (en) Novel compound with immunization activity and its preparation and application
JPS54145634A (en) Preparation of 2,6-dicyanophenol derivative
JPS57203047A (en) Preparation of amino derivative of cyclopentenone
JPS54145633A (en) Preparation of 2,6-dicyanophenol derivative
JPS567782A (en) Novel pyridinecarboxamide derivative and its preparation
JPS56122338A (en) Preparation of isocyanic acid ester
JPS57158770A (en) Thiadiazole derivative and its preparation
JPS5793954A (en) Phenoxybenzylthiol carbamate derivative, its preparaion and acaricide comprising it as active ingredient