MX2020001434A - Analogos de insulina acilados novedosos y usos de estos. - Google Patents
Analogos de insulina acilados novedosos y usos de estos.Info
- Publication number
- MX2020001434A MX2020001434A MX2020001434A MX2020001434A MX2020001434A MX 2020001434 A MX2020001434 A MX 2020001434A MX 2020001434 A MX2020001434 A MX 2020001434A MX 2020001434 A MX2020001434 A MX 2020001434A MX 2020001434 A MX2020001434 A MX 2020001434A
- Authority
- MX
- Mexico
- Prior art keywords
- insulin analogues
- acylated insulin
- novel acylated
- novel
- analogues
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/62—Insulins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
- G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
- G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K2319/00—Fusion polypeptide
- C07K2319/90—Fusion polypeptide containing a motif for post-translational modification
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N2440/00—Post-translational modifications [PTMs] in chemical analysis of biological material
- G01N2440/14—Post-translational modifications [PTMs] in chemical analysis of biological material phosphorylation
Abstract
La presente invención se refiere a análogos de insulina novedosos y derivados de estos, tales como análogos de insulina acilados, y su uso farmacéutico, en particular en el tratamiento o prevención de afecciones médicas relacionadas con la diabetes, la obesidad y enfermedades cardiovasculares.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP17186612 | 2017-08-17 | ||
EP17204872 | 2017-12-01 | ||
PCT/EP2018/072191 WO2019034726A1 (en) | 2017-08-17 | 2018-08-16 | NOVEL ACYLATED INSULIN ANALOGUES AND USES THEREOF |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2020001434A true MX2020001434A (es) | 2020-03-20 |
Family
ID=63165388
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2020001434A MX2020001434A (es) | 2017-08-17 | 2018-08-16 | Analogos de insulina acilados novedosos y usos de estos. |
Country Status (19)
Country | Link |
---|---|
US (2) | US10919949B2 (es) |
EP (1) | EP3668892A1 (es) |
JP (2) | JP2020531451A (es) |
KR (1) | KR20200038502A (es) |
CN (1) | CN111032685A (es) |
AU (1) | AU2018317810A1 (es) |
BR (1) | BR112020002364A2 (es) |
CA (1) | CA3071686A1 (es) |
CL (1) | CL2020000310A1 (es) |
CO (1) | CO2020002500A2 (es) |
IL (1) | IL272394A (es) |
MA (1) | MA49896A (es) |
MX (1) | MX2020001434A (es) |
PE (1) | PE20211264A1 (es) |
PH (1) | PH12020550050A1 (es) |
RU (1) | RU2020108281A (es) |
SG (1) | SG11202001077UA (es) |
TW (1) | TW201917134A (es) |
WO (1) | WO2019034726A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PT1969004E (pt) | 2005-12-28 | 2011-11-25 | Novo Nordisk As | Composições que compreendem uma insulina acilada e zinco e método para criar tais composições |
MX2023008330A (es) | 2021-01-20 | 2024-01-18 | Viking Therapeutics Inc | Agonistas del receptor dual gip/glp-1 de molécula pequeña, composiciones farmacéuticas y preparación de las mismas para usarse en el tratamiento de trastornos metabólicos y hepáticos. |
Family Cites Families (56)
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US4343898A (en) | 1980-02-11 | 1982-08-10 | Novo Industri A/S | Process for preparing esters of human insulin |
DK58285D0 (da) | 1984-05-30 | 1985-02-08 | Novo Industri As | Peptider samt fremstilling og anvendelse deraf |
PH25772A (en) | 1985-08-30 | 1991-10-18 | Novo Industri As | Insulin analogues, process for their preparation |
US5616729A (en) | 1986-07-17 | 1997-04-01 | Board Of Governors Of Wayne State University | Enhanced chemiluminescence from 1,2-dioxetanes through energy transfer to tethered fluorescers |
DK105489D0 (da) | 1989-03-03 | 1989-03-03 | Novo Nordisk As | Polypeptid |
DK155690D0 (da) | 1990-06-28 | 1990-06-28 | Novo Nordisk As | Nye peptider |
DK10191D0 (da) | 1991-01-22 | 1991-01-22 | Novo Nordisk As | Hidtil ukendte peptider |
DK33591D0 (es) | 1991-02-27 | 1991-02-27 | Novo Nordisk As | |
IL114160A (en) | 1994-06-17 | 2006-12-31 | Novo Nordisk As | Dna constructs encoding heterologous proteins and processes for the heterologous protein production in yeast |
US6500645B1 (en) | 1994-06-17 | 2002-12-31 | Novo Nordisk A/S | N-terminally extended proteins expressed in yeast |
US5693609A (en) | 1994-11-17 | 1997-12-02 | Eli Lilly And Company | Acylated insulin analogs |
US6451970B1 (en) | 1996-02-21 | 2002-09-17 | Novo Nordisk A/S | Peptide derivatives |
DE69735242T2 (de) | 1996-12-20 | 2006-09-21 | Novo Nordisk A/S | N-terminal verlängerte proteine exprimiert in hefe |
AU2624400A (en) | 1999-01-26 | 2000-08-07 | Eli Lilly And Company | Monodisperse hexameric acylated insulin analog formulations |
JP2003518917A (ja) * | 1999-05-19 | 2003-06-17 | ゼンコー | 糖尿病の処置に有用なインシュリン様活性を有する新規タンパク質 |
RU2283846C2 (ru) | 1999-12-29 | 2006-09-20 | Ново Нордиск А/С | Предшественник инсулина, способ его получения и применение |
EP1692168B1 (en) | 2003-12-03 | 2011-07-20 | Novo Nordisk A/S | Single-chain insulin |
WO2006008238A1 (en) * | 2004-07-16 | 2006-01-26 | Novo Nordisk A/S | Method for selective acylation |
JP4933455B2 (ja) | 2005-02-02 | 2012-05-16 | ノヴォ ノルディスク アー/エス | 新規のインスリン誘導体 |
EP1991576B1 (en) * | 2006-02-27 | 2010-09-29 | Novo Nordisk A/S | Insulin derivatives |
RU2524150C2 (ru) | 2006-09-22 | 2014-07-27 | Ново Нордиск А/С | Аналоги инсулина, устойчивые к протеазам |
AU2008288413B2 (en) | 2007-08-15 | 2013-09-26 | Novo Nordisk A/S | Insulin analogues with an acyl and aklylene glycol moiety |
US9260502B2 (en) | 2008-03-14 | 2016-02-16 | Novo Nordisk A/S | Protease-stabilized insulin analogues |
RU2571857C2 (ru) | 2008-03-18 | 2015-12-20 | Ново Нордиск А/С | Стабилизированные по отношению к протеазам ацилированные аналоги инсулина |
WO2010080609A1 (en) | 2008-12-19 | 2010-07-15 | Indiana University Research And Technology Corporation | Amide-based insulin prodrugs |
JP5789515B2 (ja) | 2008-12-19 | 2015-10-07 | インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションIndiana University Research And Technology Corporation | インスリン類似体 |
US20110245164A1 (en) | 2008-12-19 | 2011-10-06 | Indiana University Research And Technology Corporation | Yl-based insulin-like growth factors exhibiting high activity at the insulin receptor |
JP2012532177A (ja) | 2009-07-06 | 2012-12-13 | サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | 熱及び振動安定性インスリン製剤 |
WO2011159882A2 (en) | 2010-06-16 | 2011-12-22 | Indiana University Research And Technology Corporation | Novel stabilized insulin agonists |
WO2011159895A2 (en) | 2010-06-16 | 2011-12-22 | Indiana University Research And Technology Corporation | Single chain insulin agonists exhibiting high activity at the insulin receptor |
JP5973427B2 (ja) | 2010-06-23 | 2016-08-23 | ノヴォ ノルディスク アー/エス | 追加のジスルフィド結合を含有するインスリン類似体 |
EP2585102B1 (en) | 2010-06-24 | 2015-05-06 | Indiana University Research and Technology Corporation | Amide-based insulin prodrugs |
WO2011163460A1 (en) | 2010-06-24 | 2011-12-29 | Indiana University Research And Technology Corporation | Yl-based insulin-like growth factors exhibiting high activity at the insulin receptor |
WO2012015692A2 (en) | 2010-07-28 | 2012-02-02 | Smartcells, Inc. | Recombinantly expressed insulin polypeptides and uses thereof |
WO2012049307A2 (en) | 2010-10-15 | 2012-04-19 | Novo Nordisk A/S | Novel n-terminally modified insulin derivatives |
AR087433A1 (es) | 2011-08-08 | 2014-03-26 | Merck Sharp & Dohme | Analogos de insulina n-glicosilados |
EP2793932B1 (en) | 2011-12-20 | 2018-10-03 | Indiana University Research and Technology Corporation | Ctp-based insulin analogs for treatment of diabetes |
WO2013093009A1 (en) | 2011-12-21 | 2013-06-27 | Novo Nordisk A/S | N -terminally modified insulin derivatives |
JP6387008B2 (ja) | 2012-09-26 | 2018-09-05 | インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションIndiana University Research And Technology Corporation | インスリンアナローグダイマー |
EP2925345B1 (en) | 2012-12-03 | 2018-09-05 | Merck Sharp & Dohme Corp. | Method for making o-glycosylated carboxy terminal portion (ctp) peptide-based insulin and insulin analogues |
US10421795B2 (en) | 2012-12-17 | 2019-09-24 | Merck Sharp & Dohme Corp. | Process for purifying insulin and analogues thereof |
US20160024169A1 (en) | 2013-03-14 | 2016-01-28 | Indiana University Research And Technology Corporation | Insulin-incretin conjugates |
US20160193154A1 (en) | 2013-07-24 | 2016-07-07 | Novo Nordisk A/S | Pharmaceutical Composition for Oral Insulin Administration Comprising a Tablet Core and an Anionic Copolymer Coating |
MX366852B (es) | 2013-10-04 | 2019-07-25 | Merck Sharp & Dohme | Conjugados de insulina sensibles a glucosa. |
AR099569A1 (es) * | 2014-02-28 | 2016-08-03 | Novo Nordisk As | Derivados de insulina y los usos médicos de estos |
CN108271356A (zh) | 2014-09-24 | 2018-07-10 | 印第安纳大学研究及科技有限公司 | 肠降血糖素-胰岛素缀合物 |
EP3197912B1 (en) | 2014-09-24 | 2023-01-04 | Indiana University Research & Technology Corporation | Lipidated amide-based insulin prodrugs |
CA2966765C (en) | 2014-11-21 | 2020-04-14 | Merck Sharp & Dohme Corp. | Insulin receptor partial agonists |
EP3250225A1 (en) | 2015-01-29 | 2017-12-06 | Novo Nordisk A/S | Pharmaceutical composition for oral insulin administration comprising a tablet core and a polyvinyl alcohol coating |
WO2016144658A1 (en) | 2015-03-10 | 2016-09-15 | Merck Sharp & Dohme Corp. | Process for preparing recombinant insulin using microfiltration |
US20180110863A1 (en) | 2015-04-08 | 2018-04-26 | Merck Sharp & Dohme Corp. | Glucose-responsive insulin conjugates |
WO2016172269A2 (en) | 2015-04-20 | 2016-10-27 | University Of Utah Research Foundation | Insulin analogs having shortened b chain peptides and associated methods |
WO2017032798A1 (en) | 2015-08-25 | 2017-03-02 | Novo Nordisk A/S | Novel insulin derivatives and the medical uses hereof |
EP3341402A1 (en) * | 2015-08-25 | 2018-07-04 | Novo Nordisk A/S | Novel insulin derivatives and the medical uses hereof |
US20190010206A1 (en) * | 2015-08-25 | 2019-01-10 | Novo Nordisk A/S | Novel Insulin Derivatives and the Medical Uses Hereof |
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-
2018
- 2018-08-16 AU AU2018317810A patent/AU2018317810A1/en not_active Withdrawn
- 2018-08-16 CA CA3071686A patent/CA3071686A1/en not_active Withdrawn
- 2018-08-16 US US15/998,755 patent/US10919949B2/en active Active
- 2018-08-16 KR KR1020207006535A patent/KR20200038502A/ko not_active Application Discontinuation
- 2018-08-16 TW TW107128618A patent/TW201917134A/zh unknown
- 2018-08-16 EP EP18752779.1A patent/EP3668892A1/en not_active Withdrawn
- 2018-08-16 BR BR112020002364-7A patent/BR112020002364A2/pt not_active Application Discontinuation
- 2018-08-16 PE PE2020000179A patent/PE20211264A1/es unknown
- 2018-08-16 MX MX2020001434A patent/MX2020001434A/es unknown
- 2018-08-16 MA MA049896A patent/MA49896A/fr unknown
- 2018-08-16 SG SG11202001077UA patent/SG11202001077UA/en unknown
- 2018-08-16 RU RU2020108281A patent/RU2020108281A/ru unknown
- 2018-08-16 WO PCT/EP2018/072191 patent/WO2019034726A1/en active Application Filing
- 2018-08-16 JP JP2020508562A patent/JP2020531451A/ja not_active Withdrawn
- 2018-08-16 CN CN201880052683.1A patent/CN111032685A/zh not_active Withdrawn
-
2020
- 2020-01-31 IL IL272394A patent/IL272394A/en unknown
- 2020-02-05 CL CL2020000310A patent/CL2020000310A1/es unknown
- 2020-02-07 PH PH12020550050A patent/PH12020550050A1/en unknown
- 2020-03-04 CO CONC2020/0002500A patent/CO2020002500A2/es unknown
- 2020-11-05 US US17/089,993 patent/US20210094999A1/en not_active Abandoned
-
2022
- 2022-04-25 JP JP2022071578A patent/JP2022105082A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
TW201917134A (zh) | 2019-05-01 |
US20210094999A1 (en) | 2021-04-01 |
JP2022105082A (ja) | 2022-07-12 |
MA49896A (fr) | 2020-06-24 |
BR112020002364A2 (pt) | 2020-09-01 |
CL2020000310A1 (es) | 2020-07-10 |
JP2020531451A (ja) | 2020-11-05 |
RU2020108281A (ru) | 2021-08-26 |
SG11202001077UA (en) | 2020-03-30 |
CO2020002500A2 (es) | 2020-06-09 |
KR20200038502A (ko) | 2020-04-13 |
PH12020550050A1 (en) | 2020-10-19 |
PE20211264A1 (es) | 2021-07-15 |
RU2020108281A3 (es) | 2022-03-09 |
IL272394A (en) | 2020-03-31 |
EP3668892A1 (en) | 2020-06-24 |
US10919949B2 (en) | 2021-02-16 |
WO2019034726A1 (en) | 2019-02-21 |
CA3071686A1 (en) | 2019-02-21 |
CN111032685A (zh) | 2020-04-17 |
US20190194285A1 (en) | 2019-06-27 |
AU2018317810A1 (en) | 2020-03-19 |
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