MX2018000418A - Derivados de amida que tienen actividad multimodal contra el dolor. - Google Patents
Derivados de amida que tienen actividad multimodal contra el dolor.Info
- Publication number
- MX2018000418A MX2018000418A MX2018000418A MX2018000418A MX2018000418A MX 2018000418 A MX2018000418 A MX 2018000418A MX 2018000418 A MX2018000418 A MX 2018000418A MX 2018000418 A MX2018000418 A MX 2018000418A MX 2018000418 A MX2018000418 A MX 2018000418A
- Authority
- MX
- Mexico
- Prior art keywords
- amide derivatives
- activity against
- against pain
- multimodal activity
- pain
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/09—Geometrical isomers
Abstract
La presente invención se refiere a compuestos que tienen actividad farmacológica dual hacia el receptor sigma (s) y el receptor opioide µ, a procesos de preparación de dichos compuestos, a composiciones farmacéuticas que los comprenden y a su uso en terapia, en particular para el tratamiento del dolor.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP15382391 | 2015-07-29 | ||
PCT/EP2016/001309 WO2017016668A1 (en) | 2015-07-29 | 2016-07-28 | Amide derivatives having multimodal activity against pain |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2018000418A true MX2018000418A (es) | 2018-08-14 |
Family
ID=54056149
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2018000418A MX2018000418A (es) | 2015-07-29 | 2016-07-28 | Derivados de amida que tienen actividad multimodal contra el dolor. |
Country Status (9)
Country | Link |
---|---|
US (1) | US10351549B2 (es) |
EP (1) | EP3328847B1 (es) |
JP (1) | JP2018521090A (es) |
CN (1) | CN107922384A (es) |
CA (1) | CA2992054A1 (es) |
ES (1) | ES2760625T3 (es) |
HK (1) | HK1255248A1 (es) |
MX (1) | MX2018000418A (es) |
WO (1) | WO2017016668A1 (es) |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1585165A (en) | 1976-06-29 | 1981-02-25 | Leo Pharm Prod Ltd | Derivatives of 6-amidino penicillanic acid |
EP0252670B1 (en) | 1986-06-30 | 1992-01-15 | Toyo Jozo Kabushiki Kaisha | 2-substituted alkoxy-3-substituted-pyrazines |
JPH11130761A (ja) * | 1997-10-24 | 1999-05-18 | Otsuka Pharmaceut Co Ltd | ベンゾチアゾール誘導体 |
US20030022891A1 (en) * | 2000-12-01 | 2003-01-30 | Anandan Palani | MCH antagonists and their use in the treatment of obesity |
FI110636B (fi) * | 2001-06-29 | 2003-02-28 | Teknoware Oy | Järjestely valaisimen yhteydessä ja valaisin |
NZ534046A (en) * | 2001-12-04 | 2006-02-24 | Actelion Pharmaceuticals Ltd | 4-(piperidyl-and pyrrolidyl-alkyl-ureido) -quinolines as urotensin II receptor antagonists |
US7521457B2 (en) * | 2004-08-20 | 2009-04-21 | Boehringer Ingelheim International Gmbh | Pyrimidines as PLK inhibitors |
TN2016000203A1 (en) * | 2013-12-20 | 2017-10-06 | Esteve Labor Dr | Piperazine derivatives having multimodal activity against pain. |
MX2016006604A (es) | 2013-12-20 | 2016-09-08 | Esteve Labor Dr | Derivados de piperidina con actividad multimodal contra el dolor. |
-
2016
- 2016-07-28 CN CN201680043614.5A patent/CN107922384A/zh active Pending
- 2016-07-28 EP EP16744665.7A patent/EP3328847B1/en active Active
- 2016-07-28 CA CA2992054A patent/CA2992054A1/en not_active Abandoned
- 2016-07-28 JP JP2018503652A patent/JP2018521090A/ja active Pending
- 2016-07-28 ES ES16744665T patent/ES2760625T3/es active Active
- 2016-07-28 US US15/747,220 patent/US10351549B2/en not_active Expired - Fee Related
- 2016-07-28 MX MX2018000418A patent/MX2018000418A/es unknown
- 2016-07-28 WO PCT/EP2016/001309 patent/WO2017016668A1/en active Application Filing
-
2018
- 2018-11-09 HK HK18114384.5A patent/HK1255248A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
ES2760625T3 (es) | 2020-05-14 |
EP3328847B1 (en) | 2019-09-11 |
US10351549B2 (en) | 2019-07-16 |
CA2992054A1 (en) | 2017-02-02 |
HK1255248A1 (zh) | 2019-08-09 |
JP2018521090A (ja) | 2018-08-02 |
CN107922384A (zh) | 2018-04-17 |
US20180237415A1 (en) | 2018-08-23 |
WO2017016668A1 (en) | 2017-02-02 |
EP3328847A1 (en) | 2018-06-06 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PH12018500586A1 (en) | Farnesoid x receptor agonists and uses thereof | |
MX2018014154A (es) | Polinucleotidos moduladores. | |
MX2018000419A (es) | Derivados de amida sustituida que tienen actividad multimodal contra el dolor. | |
TW201613901A (en) | New compounds | |
MX2016006623A (es) | Compuestos de inhibidor de autotaxina. | |
PH12016500978A1 (en) | Piperazine derivatives having multimodal activity against pain | |
MX2017006437A (es) | Compuestos espiroisoquinolin-1,4'-piperidinicos con actividad multimodal contra el dolor. | |
MX2016006604A (es) | Derivados de piperidina con actividad multimodal contra el dolor. | |
PH12016502307B1 (en) | Alkyl derivatives of 1-oxa-4,9-diazaspiro undecane compounds having multimodal activity against pain | |
MY199091A (en) | Therapeutic compounds | |
PH12016501527A1 (en) | Pharmaceutical composition comprising diamino heterocyclic carboxamide compound as active ingredient | |
MX2021010041A (es) | Composiciones farmaceuticas que comprenden inhibidores de la proteina quinasa akt. | |
MX2017014456A (es) | Usos terapeuticos de l-4-cloroquinurenina. | |
MX2020009966A (es) | Formas de dosificacion y usos terapeuticos de la l-4-cloro quinurenina. | |
MX2016006603A (es) | Compuestos piperidinicos con actividad multimodal contra el dolor. | |
MX2017006513A (es) | Compuestos de tipo 1,9-diazaespiroundecano con actividad multimodal contra el dolor. | |
PH12018500814A1 (en) | Oxadiazaspiro compounds for the treatment of drug abuse and addiction | |
PH12018500682A1 (en) | Oxa-diazaspiro compounds having activity against pain | |
PH12018502280A1 (en) | Tetrahydropyran and thiopyran derivatives having multimodal activity against pain | |
IN2013MU03118A (es) | ||
PH12017501979A1 (en) | Pharmaceutical compound | |
MX2018004774A (es) | Derivados de morfolina sustituidos que tienen actividad contra el dolor. | |
MX2018000418A (es) | Derivados de amida que tienen actividad multimodal contra el dolor. | |
MX2018003564A (es) | 1,4-benzodiazepinas biheteroarilo sustituidas y usos de las mismas para el tratamiento del cancer. | |
MX2018004776A (es) | Compuestos oxaazaespiricos con actividad contral el dolor. |