MX2013006694A - Procedimiento para producir oxindoles sustituidos con triazinilo. - Google Patents

Procedimiento para producir oxindoles sustituidos con triazinilo.

Info

Publication number
MX2013006694A
MX2013006694A MX2013006694A MX2013006694A MX2013006694A MX 2013006694 A MX2013006694 A MX 2013006694A MX 2013006694 A MX2013006694 A MX 2013006694A MX 2013006694 A MX2013006694 A MX 2013006694A MX 2013006694 A MX2013006694 A MX 2013006694A
Authority
MX
Mexico
Prior art keywords
producing
triazinyl
substituted oxindoles
salts
compounds
Prior art date
Application number
MX2013006694A
Other languages
English (en)
Inventor
Mark James Ford
Gunter Karig
Konrad Siegel
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of MX2013006694A publication Critical patent/MX2013006694A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/66—1,3,5-Triazines, not hydrogenated and not substituted at the ring nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • AIDS & HIV (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Procedimiento para la preparación de oxindoles sustituidos con triazinilo de fórmula (3) (Ver Formula) y sus sales haciendo reaccionar un oxindol (1) con una triazina (2) en presencia de un carbonato, un hidróxido, un fosfato o una mezcla de dos o más de los compuestos anteriormente mencionados, y también los compuestos de fórmula (3) y sus sales (3") y el uso de ambos para producir agentes para la protección de cultivos.
MX2013006694A 2010-12-21 2011-12-19 Procedimiento para producir oxindoles sustituidos con triazinilo. MX2013006694A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201061425349P 2010-12-21 2010-12-21
EP10196205 2010-12-21
PCT/EP2011/073283 WO2012084855A2 (de) 2010-12-21 2011-12-19 Verfahren zur herstellung von triazinylsubstituierten oxindolen

Publications (1)

Publication Number Publication Date
MX2013006694A true MX2013006694A (es) 2013-07-29

Family

ID=44148782

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013006694A MX2013006694A (es) 2010-12-21 2011-12-19 Procedimiento para producir oxindoles sustituidos con triazinilo.

Country Status (12)

Country Link
US (2) US8962828B2 (es)
EP (1) EP2655361B1 (es)
JP (1) JP5980808B2 (es)
KR (1) KR101902599B1 (es)
CN (1) CN103380125B (es)
BR (1) BR112013016028B1 (es)
DK (1) DK2655361T3 (es)
ES (1) ES2571553T3 (es)
IL (1) IL226866A (es)
MX (1) MX2013006694A (es)
TW (1) TWI546296B (es)
WO (1) WO2012084855A2 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2571553T3 (es) * 2010-12-21 2016-05-25 Bayer Ip Gmbh Procedimiento para la preparación de oxindoles sustituidos con triazinilo
US8969553B2 (en) * 2010-12-21 2015-03-03 Bayer Intellectual Property Gmbh Method for producing N-sulfonyl-substituted oxindoles
WO2018163216A1 (en) 2017-03-10 2018-09-13 Council Of Scientific & Industrial Research Spirooxindole compounds as gsk3β inhibitors and process for preparation thereof
EP3360417A1 (de) 2017-11-02 2018-08-15 Bayer CropScience Aktiengesellschaft Verwendung von sulfonylindol als herbizid
KR102214988B1 (ko) * 2019-06-20 2021-02-10 영남대학교 산학협력단 신규한 옥시인돌 유도체 및 이를 유효성분으로 함유하는 항균용 조성물

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9707800D0 (en) 1996-05-06 1997-06-04 Zeneca Ltd Chemical compounds
JP3632947B2 (ja) 1998-07-29 2005-03-30 クミアイ化学工業株式会社 ジフルオロメタンスルホニルアニリド誘導体、その製造方法及びそれを有効成分とする除草剤
ES2306671T3 (es) 1999-10-07 2008-11-16 Amgen Inc. Inhibidores de triazina quinasa.
US6864255B2 (en) 2001-04-11 2005-03-08 Amgen Inc. Substituted triazinyl amide derivatives and methods of use
SE0200979D0 (sv) 2002-03-28 2002-03-28 Astrazeneca Ab New compounds
SE0302546D0 (sv) 2003-09-24 2003-09-24 Astrazeneca Ab New compounds
US20050070718A1 (en) 2003-09-30 2005-03-31 Abbott Gmbh & Co. Kg Heteroaryl-substituted 1,3-dihydroindol-2-one derivatives and medicaments containing them
WO2005061519A1 (en) 2003-12-19 2005-07-07 Takeda San Diego, Inc. Kinase inhibitors
JP2006056871A (ja) 2004-07-23 2006-03-02 Bayer Cropscience Ag スルホンアニリド類の農園芸用殺菌剤としての利用
US7576082B2 (en) 2005-06-24 2009-08-18 Hoffman-La Roche Inc. Oxindole derivatives
JP2007106745A (ja) 2005-09-16 2007-04-26 Bayer Cropscience Ag スルホンアニリド類の除草剤としての利用
WO2007089193A1 (en) 2006-02-02 2007-08-09 Astrazeneca Ab A process for preparing 2-hydroxy-3- [5- (morpholin-4-ylmethyl)pyridin-2-yl] lh-indole-5-carbonitrile as a free base or salts thereof
US7851468B2 (en) 2006-05-15 2010-12-14 Cephalon, Inc. Substituted pyrazolo[3,4-d]pyrimidines
DE102006040915A1 (de) 2006-08-26 2008-03-20 Abbott Gmbh & Co. Kg Substituierte Oxindol-Derivate, diese enthaltende Arzneimittel und deren Verwendung
FR2909668B1 (fr) 2006-12-12 2009-01-23 Sanofi Aventis Sa Derives de 5-alkyloxy-indolin-2-one,leur preparation et leurs applications en therapeutique
US20090291982A1 (en) 2008-05-22 2009-11-26 Astrazeneca Ab New Substituted Oxindole Derivative 352
ES2571553T3 (es) * 2010-12-21 2016-05-25 Bayer Ip Gmbh Procedimiento para la preparación de oxindoles sustituidos con triazinilo
TWI531566B (zh) * 2010-12-21 2016-05-01 拜耳農業科學股份有限公司 製備２－（三羰基）磺醯替苯胺類的方法
US8969553B2 (en) * 2010-12-21 2015-03-03 Bayer Intellectual Property Gmbh Method for producing N-sulfonyl-substituted oxindoles

Also Published As

Publication number Publication date
DK2655361T3 (en) 2016-05-23
KR20140005921A (ko) 2014-01-15
US20130345422A1 (en) 2013-12-26
EP2655361B1 (de) 2016-02-24
IL226866A (en) 2016-12-29
WO2012084855A3 (de) 2012-09-07
KR101902599B1 (ko) 2018-09-28
JP2014501744A (ja) 2014-01-23
US9522904B2 (en) 2016-12-20
US20150126737A1 (en) 2015-05-07
CN103380125B (zh) 2015-11-25
US8962828B2 (en) 2015-02-24
BR112013016028A2 (pt) 2018-07-10
TWI546296B (zh) 2016-08-21
BR112013016028B1 (pt) 2019-05-07
CN103380125A (zh) 2013-10-30
TW201238960A (en) 2012-10-01
JP5980808B2 (ja) 2016-08-31
EP2655361A2 (de) 2013-10-30
WO2012084855A2 (de) 2012-06-28
ES2571553T3 (es) 2016-05-25

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