MX2007009574A - Sal de monoclorhidrato de 1-[3-[3-(4-clorofenil)propoxi]-propil]- piperidina. - Google Patents
Sal de monoclorhidrato de 1-[3-[3-(4-clorofenil)propoxi]-propil]- piperidina.Info
- Publication number
- MX2007009574A MX2007009574A MX2007009574A MX2007009574A MX2007009574A MX 2007009574 A MX2007009574 A MX 2007009574A MX 2007009574 A MX2007009574 A MX 2007009574A MX 2007009574 A MX2007009574 A MX 2007009574A MX 2007009574 A MX2007009574 A MX 2007009574A
- Authority
- MX
- Mexico
- Prior art keywords
- chlorophenyl
- propyl
- propoxy
- piperidine
- monohydrochloride
- Prior art date
Links
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Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP05100942A EP1690858B1 (en) | 2005-02-10 | 2005-02-10 | Monohydrochloride salt of 1-[3-[3-(4-chlorophenyl)propoxy]propyl]-piperidine |
| PCT/EP2006/050703 WO2006084833A1 (en) | 2005-02-10 | 2006-02-06 | Monohydrochloride salt of 1- [3- [3- (4-chlorophenyl) propoxy] propyl] -piperidine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007009574A true MX2007009574A (es) | 2007-09-25 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007009574A MX2007009574A (es) | 2005-02-10 | 2006-02-06 | Sal de monoclorhidrato de 1-[3-[3-(4-clorofenil)propoxi]-propil]- piperidina. |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US8207197B2 (enExample) |
| EP (2) | EP1690858B1 (enExample) |
| JP (1) | JP5072604B2 (enExample) |
| KR (1) | KR101344271B1 (enExample) |
| CN (1) | CN101155793B (enExample) |
| AR (1) | AR054734A1 (enExample) |
| AT (2) | ATE391716T1 (enExample) |
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| CY (1) | CY1108428T1 (enExample) |
| DE (2) | DE602005005941D1 (enExample) |
| DK (1) | DK1846384T3 (enExample) |
| ES (1) | ES2309948T3 (enExample) |
| HR (1) | HRP20080446T3 (enExample) |
| ME (1) | ME01103B (enExample) |
| MX (1) | MX2007009574A (enExample) |
| PL (1) | PL1846384T3 (enExample) |
| PT (1) | PT1846384E (enExample) |
| RS (1) | RS50624B (enExample) |
| SI (1) | SI1846384T1 (enExample) |
| TW (1) | TWI393711B (enExample) |
| UY (1) | UY29369A1 (enExample) |
| WO (1) | WO2006084833A1 (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2167096A4 (en) * | 2007-06-13 | 2010-07-14 | Cypress Bioscience Inc | IMPROVING TOLERANCE TO MIRTAZAPINE AND A SECOND ACTIVE INGREDIENT BY THE COMBINED USE OF THEM |
| SG173639A1 (en) | 2009-02-11 | 2011-09-29 | Sunovion Pharmaceuticals Inc | Histamine h3 inverse agonists and antagonists and methods of use thereof |
| RU2011153723A (ru) | 2009-06-10 | 2013-07-20 | Суновион Фармасьютикалз Инк. | Обратные агонисты и антагонисты н3 рецепторов гистамина и способы их применения |
| US20110065694A1 (en) | 2009-09-11 | 2011-03-17 | Milan Chytil | Histamine H3 Inverse Agonists and Antagonists and Methods of Use Thereof |
| WO2014199935A1 (ja) * | 2013-06-10 | 2014-12-18 | 株式会社エム・エス・エス | 小胞体ストレスシグナルを抑制することによる，薬剤の副作用としての体重増加や肥満を防止するために用いられる肥満防止剤 |
| CN103435575A (zh) * | 2013-08-06 | 2013-12-11 | 中国人民解放军军事医学科学院毒物药物研究所 | 1-（ 3-（ 3-（ 4-氯苯基）丙氧基）丙基）哌啶盐酸盐的制备方法 |
| CN104447620B (zh) * | 2014-11-28 | 2016-05-04 | 瑞阳制药有限公司 | 1-[3-[3-(4-氯苯基)丙氧基]丙基]-哌啶盐酸盐的制备方法 |
| EP3239138A1 (en) | 2016-04-25 | 2017-11-01 | Sandoz Ag | Hydrogen fumarate salt of 1-[3-[3-(4-chlorophenyl)propoxy]propyl]piperidine |
| WO2020092604A1 (en) * | 2018-10-30 | 2020-05-07 | Concert Pharmaceuticals, Inc. | Deuterated pitolisant |
| IT201900013941A1 (it) | 2019-08-05 | 2021-02-05 | Procos Spa | PROCESSO PER LA SINTESI DI PITOLISANT HCl |
| CN110804026B (zh) * | 2019-11-18 | 2022-04-01 | 苏州永健生物医药有限公司 | 1- (3- (3-（4-氯苯基）丙氧基)丙基)哌啶盐酸盐的合成方法 |
| US11945788B2 (en) | 2021-06-07 | 2024-04-02 | Nuray Chemicals Private Limited | Process for preparing pitolisant hydrochloride and solid-state forms thereof |
| US11623920B2 (en) | 2021-06-07 | 2023-04-11 | Nuray Chemicals Private Limited | Process for preparing pitolisant hydrochloride and solid-state forms thereof |
| EP4457219A4 (en) * | 2021-12-29 | 2025-12-10 | Biophore India Pharmaceuticals Pvt Ltd | SOLID FORMS OF 1-3-[3-(4-CHLOROPHENYL)PROPOXY]PROPYL PIPERIDINE HYDROCHLORIDE AND THEIR PREPARATION PROCESS |
| US20250281475A1 (en) * | 2022-05-04 | 2025-09-11 | Msn Laboratories Private Limited, R & D Center | A pharmaceutical composition of pitolisant hydrochloride and their process for the preparation |
| WO2024084379A1 (en) * | 2022-10-17 | 2024-04-25 | Biophore India Pharmaceuticals Pvt. Ltd | A NOVEL PROCESS FOR THE PREPARATION OF AMORPHOUS SOLID DISPERSION OF 1-{3-[3-(4-CHLOROPHENYL) PROPOXY] PROPYL} PIPERIDINE, HYDROCHLORIDE WITH HYDROXYPROPYL BETA-CYCLODEXTRIN (HPβCD) |
| EP4374854A1 (en) | 2022-11-28 | 2024-05-29 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Pharmaceutical mixture comprising amorphous pitolisant |
| KR20250165426A (ko) | 2023-03-31 | 2025-11-25 | 바이오프로제 파르마 | 피톨리산트 염산염의 다형(多形) 형태 |
| WO2025082972A1 (en) | 2023-10-16 | 2025-04-24 | Bioprojet Pharma | Enteric coated pitolisant formulations and methods of use |
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| EP0982300A3 (en) * | 1998-07-29 | 2000-03-08 | Societe Civile Bioprojet | Non-imidazole alkylamines as histamine H3 - receptor ligands and their therapeutic applications |
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2006
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- 2006-02-06 PL PL06708050T patent/PL1846384T3/pl unknown
- 2006-02-06 EP EP06708050A patent/EP1846384B1/en active Active
- 2006-02-06 SI SI200630073T patent/SI1846384T1/sl unknown
- 2006-02-06 WO PCT/EP2006/050703 patent/WO2006084833A1/en not_active Ceased
- 2006-02-06 AT AT06708050T patent/ATE402154T1/de active
- 2006-02-06 ME MEP-2008-394A patent/ME01103B/me unknown
- 2006-02-06 CN CN200680008857.1A patent/CN101155793B/zh active Active
- 2006-02-06 ES ES06708050T patent/ES2309948T3/es active Active
- 2006-02-06 HR HR20080446T patent/HRP20080446T3/xx unknown
- 2006-02-06 DE DE602006001938T patent/DE602006001938D1/de active Active
- 2006-02-06 CA CA2597016A patent/CA2597016C/en active Active
- 2006-02-06 JP JP2007554541A patent/JP5072604B2/ja active Active
- 2006-02-06 PT PT06708050T patent/PT1846384E/pt unknown
- 2006-02-06 US US11/815,736 patent/US8207197B2/en active Active
- 2006-02-08 TW TW095104184A patent/TWI393711B/zh active
- 2006-02-08 AR ARP060100448A patent/AR054734A1/es not_active Application Discontinuation
- 2006-02-09 UY UY29369A patent/UY29369A1/es not_active Application Discontinuation
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2007
- 2007-09-06 KR KR1020077020422A patent/KR101344271B1/ko active Active
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2008
- 2008-10-21 CY CY20081101174T patent/CY1108428T1/el unknown
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2012
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