MX2007000906A - Procedimiento para la preparacion de 3-(4-piperidinil) -2, 3, 4, 5-tetrahidro-1, 3-benzodiazepin -2(1h)-ona. - Google Patents
Procedimiento para la preparacion de 3-(4-piperidinil) -2, 3, 4, 5-tetrahidro-1, 3-benzodiazepin -2(1h)-ona.Info
- Publication number
- MX2007000906A MX2007000906A MX2007000906A MX2007000906A MX2007000906A MX 2007000906 A MX2007000906 A MX 2007000906A MX 2007000906 A MX2007000906 A MX 2007000906A MX 2007000906 A MX2007000906 A MX 2007000906A MX 2007000906 A MX2007000906 A MX 2007000906A
- Authority
- MX
- Mexico
- Prior art keywords
- benzodiazepin
- piperidinyl
- tetrahydro
- producing
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pain & Pain Management (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Es objeto de la presente invencion un procedimiento para la preparacion del compuesto 3-(4-piperidinil)- 2, 3, 4, 5- tetrahidro??l, 3??benzodiazepjn-2 (1H)-ona de la formula que se ha de encontrar como elemento en antagonistas de CGRP que son apropiados sobre todo para la terapia oral de la migrana.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP04017424A EP1619187A1 (de) | 2004-07-23 | 2004-07-23 | Verfahren zur Herstellung von 3-(4-Piperidinyl)- 2,3,4,5-tetrahydro-1,3-benzodiazepin-2(1H)-on |
PCT/EP2005/007778 WO2006010511A1 (de) | 2004-07-23 | 2005-07-16 | Verfahren zur herstellung 3-(4-piperidinyl)-2,3,4,5-tetrahydro-1,3-benzodiazepin-2(1h)-on |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2007000906A true MX2007000906A (es) | 2007-04-13 |
Family
ID=34925890
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2007000906A MX2007000906A (es) | 2004-07-23 | 2005-07-16 | Procedimiento para la preparacion de 3-(4-piperidinil) -2, 3, 4, 5-tetrahidro-1, 3-benzodiazepin -2(1h)-ona. |
Country Status (19)
Country | Link |
---|---|
US (1) | US7141667B2 (es) |
EP (2) | EP1619187A1 (es) |
JP (1) | JP4516118B2 (es) |
KR (1) | KR20070046881A (es) |
CN (2) | CN102040590A (es) |
AR (1) | AR050352A1 (es) |
AU (1) | AU2005266579A1 (es) |
BR (1) | BRPI0513468A (es) |
CA (1) | CA2572811C (es) |
EA (1) | EA011260B1 (es) |
EC (1) | ECSP077190A (es) |
IL (1) | IL180848A0 (es) |
MX (1) | MX2007000906A (es) |
NO (1) | NO20070366L (es) |
NZ (1) | NZ553294A (es) |
TW (1) | TW200613283A (es) |
UA (1) | UA87507C2 (es) |
WO (1) | WO2006010511A1 (es) |
ZA (1) | ZA200609919B (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN101146799A (zh) | 2005-03-23 | 2008-03-19 | 贝林格尔·英格海姆国际有限公司 | Cgrp拮抗剂、其制备方法以及其作为药物的用途 |
US7473778B2 (en) * | 2005-12-24 | 2009-01-06 | Boehringer Ingelheim International Gmbh | 3-(4-piperidinyl)-2,3,4,5-tetrahydro-1,3-benzodiazepin-2(1H)-one |
DE102007038251A1 (de) | 2007-08-13 | 2009-02-19 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neues Herstellverfahren |
US8829006B2 (en) | 2007-11-22 | 2014-09-09 | Boehringer Ingelheim International Gmbh | Compounds |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3474090A (en) * | 1966-12-22 | 1969-10-21 | American Cyanamid Co | 3-aminoalkyl-1,3-benzodiazepin-2-ones |
FR2518544A1 (fr) * | 1981-12-22 | 1983-06-24 | Lipha | Benzodiazepines-1,3 thione-2, procede de preparation et medicament les contenant |
DE19911039A1 (de) | 1999-03-12 | 2000-09-14 | Boehringer Ingelheim Pharma | Abgewandelte Aminosäureamide, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung |
FR2791021B1 (fr) * | 1999-03-16 | 2001-05-11 | France Design | Arceau de protection pour vehicule decouvrable a toit repliable |
-
2004
- 2004-07-23 EP EP04017424A patent/EP1619187A1/de not_active Withdrawn
-
2005
- 2005-07-16 WO PCT/EP2005/007778 patent/WO2006010511A1/de active Application Filing
- 2005-07-16 BR BRPI0513468-4A patent/BRPI0513468A/pt not_active IP Right Cessation
- 2005-07-16 CN CN2010106088785A patent/CN102040590A/zh active Pending
- 2005-07-16 JP JP2007521872A patent/JP4516118B2/ja not_active Expired - Fee Related
- 2005-07-16 AU AU2005266579A patent/AU2005266579A1/en not_active Abandoned
- 2005-07-16 CN CNA2005800242298A patent/CN1989114A/zh active Pending
- 2005-07-16 UA UAA200701639A patent/UA87507C2/ru unknown
- 2005-07-16 EA EA200700041A patent/EA011260B1/ru not_active IP Right Cessation
- 2005-07-16 MX MX2007000906A patent/MX2007000906A/es active IP Right Grant
- 2005-07-16 EP EP05775923A patent/EP1773789A1/de not_active Withdrawn
- 2005-07-16 NZ NZ553294A patent/NZ553294A/en not_active IP Right Cessation
- 2005-07-16 CA CA2572811A patent/CA2572811C/en not_active Expired - Fee Related
- 2005-07-16 KR KR1020077004190A patent/KR20070046881A/ko not_active Application Discontinuation
- 2005-07-19 US US11/185,593 patent/US7141667B2/en active Active
- 2005-07-22 AR ARP050103035A patent/AR050352A1/es not_active Application Discontinuation
- 2005-07-22 TW TW094125013A patent/TW200613283A/zh unknown
-
2006
- 2006-11-28 ZA ZA200609919A patent/ZA200609919B/en unknown
-
2007
- 2007-01-19 NO NO20070366A patent/NO20070366L/no not_active Application Discontinuation
- 2007-01-22 IL IL180848A patent/IL180848A0/en unknown
- 2007-01-22 EC EC2007007190A patent/ECSP077190A/es unknown
Also Published As
Publication number | Publication date |
---|---|
US20060019946A1 (en) | 2006-01-26 |
BRPI0513468A (pt) | 2008-05-06 |
EP1773789A1 (de) | 2007-04-18 |
UA87507C2 (en) | 2009-07-27 |
AU2005266579A1 (en) | 2006-02-02 |
WO2006010511A8 (de) | 2006-05-18 |
IL180848A0 (en) | 2007-07-04 |
NO20070366L (no) | 2007-02-06 |
KR20070046881A (ko) | 2007-05-03 |
AR050352A1 (es) | 2006-10-18 |
CA2572811A1 (en) | 2006-02-02 |
EA200700041A1 (ru) | 2007-08-31 |
US7141667B2 (en) | 2006-11-28 |
JP4516118B2 (ja) | 2010-08-04 |
CA2572811C (en) | 2012-09-11 |
JP2008507484A (ja) | 2008-03-13 |
NZ553294A (en) | 2009-07-31 |
ZA200609919B (en) | 2008-07-30 |
TW200613283A (en) | 2006-05-01 |
WO2006010511A1 (de) | 2006-02-02 |
CN1989114A (zh) | 2007-06-27 |
EP1619187A1 (de) | 2006-01-25 |
EA011260B1 (ru) | 2009-02-27 |
ECSP077190A (es) | 2007-03-29 |
CN102040590A (zh) | 2011-05-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant or registration |