MD59B1 - Procedeu de capatare 5 pipe-ridino-7-n-(n-pentil)-n-(beta-oxietil)-amino)-s-triazolo (1,5-a) pirimidinei - Google Patents

Procedeu de capatare 5 pipe-ridino-7-n-(n-pentil)-n-(beta-oxietil)-amino)-s-triazolo (1,5-a) pirimidinei

Info

Publication number
MD59B1
MD59B1 MD940068A MD940068A MD59B1 MD 59 B1 MD59 B1 MD 59B1 MD 940068 A MD940068 A MD 940068A MD 940068 A MD940068 A MD 940068A MD 59 B1 MD59 B1 MD 59B1
Authority
MD
Moldova
Prior art keywords
pyridino
triazolo
oxyethyl
pyrimidine
pentyl
Prior art date
Application number
MD940068A
Other languages
English (en)
Other versions
MD59C2 (ro
Inventor
Martina Ballnus
Ernst Tenor
Eckehard Thomas
Rudi Pasche
Hans-Juergen Mest
Hans-Ulrich Block
Peter Mentz
Ingrid Heinroth-Hoffman
Original Assignee
Rodleben Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rodleben Pharma Gmbh filed Critical Rodleben Pharma Gmbh
Publication of MD59B1 publication Critical patent/MD59B1/ro
Publication of MD59C2 publication Critical patent/MD59C2/ro

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Cardiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MD94-0068A 1984-04-17 1994-02-15 Procedeu de obţinere a 5-piperidino-7-I N-(n-pentil)-N-(-oxietil)-aminoI-S-triazolo(1,5-a) pirimidinei MD59C2 (ro)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DD84262043A DD228811A1 (de) 1984-04-17 1984-04-17 Verfahren zur herstellung von neuen triazolopyrimidinen

Publications (2)

Publication Number Publication Date
MD59B1 true MD59B1 (ro) 1994-08-31
MD59C2 MD59C2 (ro) 1995-01-31

Family

ID=5556238

Family Applications (1)

Application Number Title Priority Date Filing Date
MD94-0068A MD59C2 (ro) 1984-04-17 1994-02-15 Procedeu de obţinere a 5-piperidino-7-I N-(n-pentil)-N-(-oxietil)-aminoI-S-triazolo(1,5-a) pirimidinei

Country Status (15)

Country Link
JP (1) JPS60224692A (ro)
AT (1) AT391866B (ro)
BE (2) BE902218A (ro)
CH (1) CH669196A5 (ro)
DD (1) DD228811A1 (ro)
DE (1) DE3512629C2 (ro)
ES (1) ES8706682A1 (ro)
FR (1) FR2562895B1 (ro)
GB (1) GB2157684B (ro)
LT (1) LT2594B (ro)
MD (1) MD59C2 (ro)
NL (1) NL8501111A (ro)
SE (1) SE466104B (ro)
SU (1) SU1468423A3 (ro)
YU (1) YU47167B (ro)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT76810A (en) * 1994-09-16 1997-11-28 Novo Nordisk As [1,2,4]triazolo[4,3-a]quinoxalinone derivatives, process for their preparation and pharmaceutical compositions containing them
US5869486A (en) * 1995-02-24 1999-02-09 Ono Pharmaceutical Co., Ltd. Fused pyrimidines and pyriazines as pharmaceutical compounds
EP0757984B1 (en) * 1995-08-08 2002-10-30 Ono Pharmaceutical Co., Ltd. Hydroxamic acid derivatives useful for inhibiting gelatinase
JP2001322933A (ja) 2000-05-15 2001-11-20 Ucb Sa Cd40シグナル遮断剤
RU2401268C2 (ru) * 2005-08-24 2010-10-10 Пфайзер Инк. КРИСТАЛЛИЧЕСКАЯ ФОРМА (R)-6-ЦИКЛОПЕНТИЛ-6-(2-(2,6-ДИЭТИЛПИРИДИН-4-ИЛ)ЭТИЛ)-3-((5,7-ДИМЕТИЛ-[1,2,4]ТРИАЗОЛО[1,5-a]ПИРИМИДИН-2-ИЛ)МЕТИЛ)-4-ГИДРОКСИ-5,6-ДИГИДРОПИРАН-2-ОНА, ЕЕ ПРИМЕНЕНИЕ И ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ, СОДЕРЖАЩАЯ ЕЕ
US8186931B2 (en) 2006-08-17 2012-05-29 Steven Borntrager Powered hand truck
MD4246C1 (ro) * 2012-03-12 2014-03-31 Иван ПРИДА Butoi pentru maturarea produselor alcoolice
WO2018175906A1 (en) 2017-03-24 2018-09-27 Nanosyn, Inc. Fused triazolo-pyrimidine compounds having useful pharmaceutical application

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE61269C (de) * 1891-04-01 1892-03-23 J. NEWBURG in Berlin O., Am Schlesischen Bahnhof Nr. 5 Waschmaschine
CH569734A5 (en) * 1967-07-01 1975-11-28 Hydrierwerk Rodleben Veb 5-and 7-basically subst s-triazolo 1 5-a pyrimidines
DE1720004A1 (de) * 1968-03-08 1971-05-19 Hydrierwerk Rodleben Veb Verfahren zur Herstellung von s-Triazolo(1.5-a)pyrimidinen,die in 5- und 7-Stellung durch basische Gruppen substituiert sind

Also Published As

Publication number Publication date
JPS60224692A (ja) 1985-11-09
SE8501835D0 (sv) 1985-04-15
NL8501111A (nl) 1985-11-18
LT2594B (lt) 1994-03-25
BE902218A (fr) 1985-08-16
CH669196A5 (de) 1989-02-28
DE3512629A1 (de) 1986-10-09
DE3512629C2 (de) 1995-07-06
ATA105085A (de) 1990-06-15
YU47167B (sh) 1995-01-31
GB8509561D0 (en) 1985-05-22
ES542269A0 (es) 1987-07-01
BE903828R (fr) 1986-04-01
FR2562895A1 (fr) 1985-10-18
YU64185A (sh) 1992-09-07
AT391866B (de) 1990-12-10
DD228811A1 (de) 1985-10-23
GB2157684B (en) 1987-11-11
FR2562895B1 (fr) 1988-10-07
SE466104B (sv) 1991-12-16
JPH0455193B2 (ro) 1992-09-02
SE8501835L (sv) 1985-10-18
ES8706682A1 (es) 1987-07-01
GB2157684A (en) 1985-10-30
SU1468423A3 (ru) 1989-03-23
MD59C2 (ro) 1995-01-31

Similar Documents

Publication Publication Date Title
DE3576367D1 (de) Elektroformungsverfahren.
DK159585D0 (da) Benzoylureaderivater
ES549920A0 (es) Procedimiento para preparar (2-oxo-1,2,3,5-tetrahidroimidazo(2,1-b) quinazolinil)-oxialquilamidas
IT8423280A0 (it) Processo per la sintesi di 2-metossi-6-bromo-naftalene.
MD59B1 (ro) Procedeu de capatare 5 pipe-ridino-7-n-(n-pentil)-n-(beta-oxietil)-amino)-s-triazolo (1,5-a) pirimidinei
AR242388A1 (es) Procedimiento para preparar 1,6-naftiridin-2(1h)-onas,compuestos intermediarios y procedimiento.
DK292684D0 (da) Befaestelse for beklaedningsgenstand
IT1211125B (it) Composti azotati. processo per la preparazione di
IT1177104B (it) Processo per la preparazione di (2,2)-paraciclofano
IT1139269B (it) Processo per la preparazione di 1,1-dialo-1,2,2,2-tetrafluoroetani
YU95186A (en) Process for obtaining substituted 1,2,3,5-tetrahydroimidazo(2,1-b)hynazolin-2-(1h)-ones
IT1199413B (it) Processo per la preparazione di pirido-imidazo-rifamicine
FI922267L (fi) Menetelmä uusien terapeuttisesti käyttökelpoisten 3-isoksatsolyyli-4-okso-imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi
ES540594A0 (es) Procedimiento de preparar 7,8 dihidroimidazo (1,5-a) piraci-na-8-onas.
BR8502920A (pt) Processo para a preparacao de 2-benzil-7,7-dimetil-6,8-dioxa-2-aza-espiro(3,5)nonano
LV5512A3 (lv) 5-Piperidino-7-ÚN-(n-pentil)-N-(beta-oksietil)-amino¾-S-triazol(1,5-a)pirimidina iegusanas panemeis
IT8445726A0 (it) Procedimento per la fabbricazione di asciugabiancheria.
ES538991A0 (es) Procedimiento para la obtencion de quinazolin-2.4(1h.3h)-dionas substituidas
ES546556A0 (es) Procedimiento para la obtencion de sulfoniliso (tio)ureas
FI922269L (fi) Menetelmä uusien terapeuttisesti käyttökelpoisten 4-okso-imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi
IT1209606B (it) Processo per la preparazione di isossazoli 3,5-disostituiti.
RO93222A2 (ro) Procedeu pentru obtinerea acidului 1,4-dihidroxi-2-naftoic
BR8506809A (pt) Encaixe"zif"para porta-chips
IT1210009B (it) Processo per la preparazione di tiocarbammati.
ES506367A0 (es) Procedimiento para la obtencion de 2(1h)-piridinonas

Legal Events

Date Code Title Description
1M4A Expiration of terms