MD59B1 - Process for obtaining 5-pyridino-7-n- (n-pentyl) -n- (beta-oxyethyl) -amino) -s-triazolo (1,5-a) pyrimidine - Google Patents

Process for obtaining 5-pyridino-7-n- (n-pentyl) -n- (beta-oxyethyl) -amino) -s-triazolo (1,5-a) pyrimidine

Info

Publication number
MD59B1
MD59B1 MD940068A MD940068A MD59B1 MD 59 B1 MD59 B1 MD 59B1 MD 940068 A MD940068 A MD 940068A MD 940068 A MD940068 A MD 940068A MD 59 B1 MD59 B1 MD 59B1
Authority
MD
Moldova
Prior art keywords
pyridino
triazolo
oxyethyl
pyrimidine
pentyl
Prior art date
Application number
MD940068A
Other languages
Romanian (ro)
Other versions
MD59C2 (en
Inventor
Martina Ballnus
Ernst Tenor
Eckehard Thomas
Rudi Pasche
Hans-Juergen Mest
Hans-Ulrich Block
Peter Mentz
Ingrid Heinroth-Hoffman
Original Assignee
Rodleben Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rodleben Pharma Gmbh filed Critical Rodleben Pharma Gmbh
Publication of MD59B1 publication Critical patent/MD59B1/en
Publication of MD59C2 publication Critical patent/MD59C2/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Cardiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MD94-0068A 1984-04-17 1994-02-15 Process for obtaining the 5-piperidino-7-N-(N-pentyl)-N-(b-oxyethyl)-amino)-S-triazolo (1,5-a) pyrimidine MD59C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DD84262043A DD228811A1 (en) 1984-04-17 1984-04-17 PROCESS FOR THE PREPARATION OF NEW TRIAZOLOPYRIMIDINES

Publications (2)

Publication Number Publication Date
MD59B1 true MD59B1 (en) 1994-08-31
MD59C2 MD59C2 (en) 1995-01-31

Family

ID=5556238

Family Applications (1)

Application Number Title Priority Date Filing Date
MD94-0068A MD59C2 (en) 1984-04-17 1994-02-15 Process for obtaining the 5-piperidino-7-N-(N-pentyl)-N-(b-oxyethyl)-amino)-S-triazolo (1,5-a) pyrimidine

Country Status (15)

Country Link
JP (1) JPS60224692A (en)
AT (1) AT391866B (en)
BE (2) BE902218A (en)
CH (1) CH669196A5 (en)
DD (1) DD228811A1 (en)
DE (1) DE3512629C2 (en)
ES (1) ES8706682A1 (en)
FR (1) FR2562895B1 (en)
GB (1) GB2157684B (en)
LT (1) LT2594B (en)
MD (1) MD59C2 (en)
NL (1) NL8501111A (en)
SE (1) SE466104B (en)
SU (1) SU1468423A3 (en)
YU (1) YU47167B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2200055A1 (en) * 1994-09-16 1996-03-21 Novo Nordisk A/S [1,2,4]triazolo[4,3-a]quinoxalinone derivatives, their preparation and use
US5869486A (en) * 1995-02-24 1999-02-09 Ono Pharmaceutical Co., Ltd. Fused pyrimidines and pyriazines as pharmaceutical compounds
EP0757984B1 (en) * 1995-08-08 2002-10-30 Ono Pharmaceutical Co., Ltd. Hydroxamic acid derivatives useful for inhibiting gelatinase
JP2001322933A (en) 2000-05-15 2001-11-20 Ucb Sa CD40 signal blocker
RU2401268C2 (en) * 2005-08-24 2010-10-10 Пфайзер Инк. CRYSTALLINE FORM OF (R)-6-CYCLOPENTYL-6-(2-(2,6-DIETHYLPYRIDIN-4-YL)ETHYL)-3-((5,7-DIMETHYL-[1,2,4]TRIAZOLO[1,5-a]PYRIMIDIN-2-YL)METHYL)-4-HYDROXY-5,6-DIHYDROPYRAN-2-ONE, USE THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING SAID COMPOUND
US8186931B2 (en) 2006-08-17 2012-05-29 Steven Borntrager Powered hand truck
MD4246C1 (en) * 2012-03-12 2014-03-31 Иван ПРИДА Barrel for aging alcoholic products
KR102642378B1 (en) 2017-03-24 2024-02-28 픽사이 인코포레이티드 Fused triazolo-pyrimidine compounds with useful pharmaceutical applications

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE61269C (en) * 1891-04-01 1892-03-23 J. NEWBURG in Berlin O., Am Schlesischen Bahnhof Nr. 5 Washing machine
CH569734A5 (en) * 1967-07-01 1975-11-28 Hydrierwerk Rodleben Veb 5-and 7-basically subst s-triazolo 1 5-a pyrimidines
DE1720004A1 (en) * 1968-03-08 1971-05-19 Hydrierwerk Rodleben Veb Process for the preparation of s-triazolo (1.5-a) pyrimidines which are substituted in the 5- and 7-positions by basic groups

Also Published As

Publication number Publication date
ES542269A0 (en) 1987-07-01
BE902218A (en) 1985-08-16
MD59C2 (en) 1995-01-31
AT391866B (en) 1990-12-10
GB2157684B (en) 1987-11-11
FR2562895B1 (en) 1988-10-07
ATA105085A (en) 1990-06-15
DE3512629C2 (en) 1995-07-06
SE466104B (en) 1991-12-16
JPH0455193B2 (en) 1992-09-02
YU64185A (en) 1992-09-07
DD228811A1 (en) 1985-10-23
SE8501835D0 (en) 1985-04-15
YU47167B (en) 1995-01-31
GB8509561D0 (en) 1985-05-22
SU1468423A3 (en) 1989-03-23
LT2594B (en) 1994-03-25
ES8706682A1 (en) 1987-07-01
GB2157684A (en) 1985-10-30
DE3512629A1 (en) 1986-10-09
CH669196A5 (en) 1989-02-28
FR2562895A1 (en) 1985-10-18
NL8501111A (en) 1985-11-18
BE903828R (en) 1986-04-01
SE8501835L (en) 1985-10-18
JPS60224692A (en) 1985-11-09

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Legal Events

Date Code Title Description
1M4A Expiration of terms