MA33022B1 - Composition à libération contrôlée pour produire une préparation à libération prolongée contenant de l'udénafil - Google Patents
Composition à libération contrôlée pour produire une préparation à libération prolongée contenant de l'udénafilInfo
- Publication number
- MA33022B1 MA33022B1 MA33942A MA33942A MA33022B1 MA 33022 B1 MA33022 B1 MA 33022B1 MA 33942 A MA33942 A MA 33942A MA 33942 A MA33942 A MA 33942A MA 33022 B1 MA33022 B1 MA 33022B1
- Authority
- MA
- Morocco
- Prior art keywords
- produce
- odiphenyl
- mixture
- order
- textured
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
LA PRÉSENTE INVENTION CONCERNE UNE COMPOSITION À LIBÉRATION CONTRÔLÉE POUR PRODUIRE UNE PRÉPARATION À LIBÉRATION PROLONGÉE CONTENANT DE L'UDÉNAFIL. PLUS PARTICULIÈREMENT, LA PRÉSENTE INVENTION CONCERNE UNE COMPOSITION À LIBÉRATION CONTRÔLÉE POUR PRODUIRE UNE PRÉPARATION À LIBÉRATION PROLONGÉE CONTENANT DE L'UDÉNAFIL, LADITE COMPOSITION CONTENANT (A) DE L'UDÉNAFIL ET UN SEL PHARMACEUTIQUEMENT ACCEPTABLE, (B) UN MODULATEUR DE SOLUBILITÉ, (C) UN ADSORBANT, ET (D) UN POLYMÈRE HYDROPHILE. LA COMPOSITION À LIBÉRATION CONTRÔLÉE POUR PRODUIRE UNE PRÉPARATION À LIBÉRATION PROLONGÉE CONTENANT DE L'UDÉNAFIL SELON LA PRÉSENTE INVENTION LIBÈRE DES MÉDICAMENTS CONSTAMMENT QUEL QUE SOIT LE NIVEAU DE PH DANS LE TRACTUS GASTRO-INTESTINAL, ET AINSI RÉGULE LIBREMENT LA DURÉE DE LIBÉRATION DE MÉDICAMENT DANS LA PLAGE DE 3 À 24 HEURES, ET RÉDUIT LA VARIABILITÉ DE L'EFFET DE MÉDICAMENTS ENTRE INDIVIDUS. DE PLUS, LA COMPOSITION DE LA PRÉSENTE INVENTION PEUT ÊTRE PRODUITE DANS UNE PRÉPARATION À LIBÉRATION PROLONGÉE QUI A UNE CONDITION OPTIMALE POUR EXPRIMER L'EFFET DE MÉDICAMENTS DANS LE TRAITEMENT DE MALADIES TELLES QUE L'HYPERTENSION ARTÉRIELLE PULMONAIRE, L'HYPERTENSION PORTALE HÉPATIQUE, UNE HYPERPLASIE PROSTATIQUE BÉNIGNE, ET SIMILAIRE, QUI PEUVENT ÊTRE TRAITÉES PAR L'UDÉNAFIL ET QUI REQUIÈRENT L'ADMINISTRATION DE MÉDICAMENTS SUR UNE LONGUE DURÉE. LA COMPOSITION DE LA PRÉSENTE INVENTION PEUT RÉGULER LA LIBÉRATION DE MÉDICAMENTS EN FONCTION DU TEMPS NÉCESSAIRE POUR L'ABSORPTION DE CEUX-CI LORSQUE LESDITS MÉDICAMENTS SONT ADMINISTRÉS À UN CORPS VIVANT, ET AINSI PEUVENT ÊTRE UTILISÉS DE MANIÈRE BÉNÉFIQUE DANS LA PRÉVENTION ET LE TRAITEMENT D'UN TROUBLE DE L'ÉRECTION.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR1020080128499A KR101004205B1 (ko) | 2008-12-17 | 2008-12-17 | 유데나필 함유 서방성 제제를 제조하기 위한 제어방출 조성물 |
PCT/KR2009/007382 WO2010071320A2 (fr) | 2008-12-17 | 2009-12-10 | Composition à libération contrôlée pour produire une préparation à libération prolongée contenant de l'udénafil |
Publications (1)
Publication Number | Publication Date |
---|---|
MA33022B1 true MA33022B1 (fr) | 2012-02-01 |
Family
ID=42269213
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA33942A MA33022B1 (fr) | 2008-12-17 | 2009-12-10 | Composition à libération contrôlée pour produire une préparation à libération prolongée contenant de l'udénafil |
Country Status (14)
Country | Link |
---|---|
US (1) | US20110250279A1 (fr) |
EP (1) | EP2374479A4 (fr) |
JP (1) | JP2012512242A (fr) |
KR (1) | KR101004205B1 (fr) |
CN (1) | CN102307597A (fr) |
AU (1) | AU2009327758A1 (fr) |
BR (1) | BRPI0923003A2 (fr) |
CA (1) | CA2746190A1 (fr) |
MA (1) | MA33022B1 (fr) |
MX (1) | MX2011006450A (fr) |
RU (1) | RU2480240C2 (fr) |
SG (1) | SG172084A1 (fr) |
WO (1) | WO2010071320A2 (fr) |
ZA (1) | ZA201104445B (fr) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102871997B (zh) * | 2011-07-12 | 2013-11-13 | 山东绿叶制药有限公司 | 含有去甲基文拉法辛苯甲酸酯类化合物的缓释药物组合物 |
EP2919903B1 (fr) | 2012-11-14 | 2020-07-22 | W.R. Grace & CO. - CONN. | Compositions contenant un matériau biologiquement actif et un oxyde inorganique non ordonné |
EP3082428A4 (fr) | 2013-12-09 | 2017-08-02 | Respira Therapeutics, Inc. | Formulations en poudre d'inhibiteur pde5 et procédés y associés |
TN2017000029A1 (en) | 2014-08-12 | 2018-07-04 | Mezzion Pharma Co Ltd | Methods of improving myocardial performance in fontan patients using udenafil compositions |
WO2016168077A1 (fr) * | 2015-04-16 | 2016-10-20 | Bpsi Holdings, Llc | Compositions d'oxyde de polyéthylène stabilisé |
KR102249155B1 (ko) * | 2019-07-26 | 2021-05-07 | 주식회사 코아팜바이오 | 유데나필을 함유하는 약제학적 조성물 |
Family Cites Families (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR0136527Y1 (ko) | 1993-11-30 | 1999-03-20 | 이대원 | 와이어 본딩 헤드 |
GB9523752D0 (en) | 1995-11-21 | 1996-01-24 | Pfizer Ltd | Pharmaceutical formulations |
US6200604B1 (en) * | 1998-03-27 | 2001-03-13 | Cima Labs Inc. | Sublingual buccal effervescent |
EP2127642A3 (fr) * | 1998-08-13 | 2010-02-24 | Cima Labs, Inc. | Microémulsions en tant que formes galéniques solides pour administration orale |
EA002720B1 (ru) | 1998-08-27 | 2002-08-29 | Фармациа Энд Апджон Аб | Терапевтическая композиция для введения толтеродина с контролируемым высвобождением и способ лечения мочевого пузыря с её использованием |
UA67802C2 (uk) * | 1998-10-23 | 2004-07-15 | Пфайзер Рісьоч Енд Дівелепмент Компані, Н.В./С.А. | Фармацевтична композиція з контрольованим вивільненням інгібітора цгмф фде-5 (варіанти), спосіб її одержання та спосіб лікування еректильної дисфункції |
WO2000054777A1 (fr) * | 1999-03-16 | 2000-09-21 | Pentech Pharmaceuticals, Inc. | Liberation controlee de sildenafil administre par voie sublinguale ou orale |
TWI224966B (en) | 1999-11-02 | 2004-12-11 | Pfizer | Pharmaceutical composition (I) useful for treating or preventing pulmonary hypertension in a patient |
DE60038698T2 (de) | 1999-12-23 | 2009-05-07 | Pfizer Products Inc., Groton | Hydrogel-gesteuerte dosierungsform |
ATE444060T1 (de) * | 2001-06-22 | 2009-10-15 | Pfizer Prod Inc | Pharmazeutische zusammensetzungen enthaltend dispersionen aus arzneistoffen und neutralen polymeren |
JP4547148B2 (ja) | 2001-06-22 | 2010-09-22 | ベンド・リサーチ・インコーポレーテッド | 非晶質薬剤の吸着物の医薬組成物 |
KR200270330Y1 (ko) | 2001-10-09 | 2002-04-03 | 이대범 | 퍼머용 아이롱 |
US20050042177A1 (en) | 2003-07-23 | 2005-02-24 | Elan Pharma International Ltd. | Novel compositions of sildenafil free base |
DE102004027743A1 (de) | 2004-06-07 | 2006-01-05 | Fresenius Medical Care Deutschland Gmbh | Kappe, insbesondere Desinfektionskappe, Detektionsvorrichtung für die Peritonealdialyse, Beutelset für die Peritonealdialyse und dessen Verwendung |
WO2006102964A2 (fr) | 2005-03-29 | 2006-10-05 | Evonik Röhm Gmbh | Forme pharmaceutique multiparticulaire constituee de pellets renfermant une substance ayant un effet modulaire sur la liberation de l'ingredient actif |
US20070031349A1 (en) * | 2005-06-23 | 2007-02-08 | David Monteith | Rapidly absorbing oral formulations of PDE 5 inhibitors |
KR100912680B1 (ko) * | 2006-03-16 | 2009-08-19 | (주) 벡스코아 | 제어 방출 제형 |
KR100792126B1 (ko) | 2006-04-04 | 2008-01-04 | 동아제약주식회사 | 피라졸로피리미디논 화합물을 유효성분으로 함유하는전립선 비대증 예방 및 치료제 |
KR101304343B1 (ko) * | 2006-04-06 | 2013-09-11 | 한미사이언스 주식회사 | Pde-5 억제제의 경구용 속용제형 |
KR100780479B1 (ko) * | 2006-05-08 | 2007-11-28 | 윈셋파마 주식회사 | 이부딜라스트 함유 경구용 제제 및 이의 제조방법 |
KR100791844B1 (ko) * | 2006-06-30 | 2008-01-07 | 주식회사유한양행 | 메트포르민 또는 그의 염을 함유하는 서방성 제제 및 그의제조방법 |
US20080014257A1 (en) * | 2006-07-14 | 2008-01-17 | Par Pharmaceutical, Inc. | Oral dosage forms |
KR200483492Y1 (ko) | 2015-03-31 | 2017-05-22 | 산제트 인터내셔널 컴퍼니, 리미티드 | 공작기계의 지능형 제어 시스템 |
-
2008
- 2008-12-17 KR KR1020080128499A patent/KR101004205B1/ko active IP Right Grant
-
2009
- 2009-12-10 CA CA2746190A patent/CA2746190A1/fr not_active Abandoned
- 2009-12-10 RU RU2011129643/15A patent/RU2480240C2/ru not_active IP Right Cessation
- 2009-12-10 MA MA33942A patent/MA33022B1/fr unknown
- 2009-12-10 WO PCT/KR2009/007382 patent/WO2010071320A2/fr active Application Filing
- 2009-12-10 SG SG2011042561A patent/SG172084A1/en unknown
- 2009-12-10 MX MX2011006450A patent/MX2011006450A/es not_active Application Discontinuation
- 2009-12-10 AU AU2009327758A patent/AU2009327758A1/en not_active Abandoned
- 2009-12-10 US US13/140,241 patent/US20110250279A1/en not_active Abandoned
- 2009-12-10 JP JP2011542002A patent/JP2012512242A/ja not_active Abandoned
- 2009-12-10 CN CN2009801562658A patent/CN102307597A/zh active Pending
- 2009-12-10 BR BRPI0923003A patent/BRPI0923003A2/pt not_active IP Right Cessation
- 2009-12-10 EP EP09833598A patent/EP2374479A4/fr not_active Withdrawn
-
2011
- 2011-06-15 ZA ZA2011/04445A patent/ZA201104445B/en unknown
Also Published As
Publication number | Publication date |
---|---|
WO2010071320A2 (fr) | 2010-06-24 |
SG172084A1 (en) | 2011-07-28 |
MX2011006450A (es) | 2011-07-28 |
EP2374479A4 (fr) | 2012-09-12 |
AU2009327758A1 (en) | 2011-07-07 |
KR101004205B1 (ko) | 2010-12-24 |
KR20100069939A (ko) | 2010-06-25 |
EP2374479A2 (fr) | 2011-10-12 |
CN102307597A (zh) | 2012-01-04 |
US20110250279A1 (en) | 2011-10-13 |
ZA201104445B (en) | 2012-03-28 |
BRPI0923003A2 (pt) | 2015-12-15 |
WO2010071320A3 (fr) | 2010-09-30 |
JP2012512242A (ja) | 2012-05-31 |
RU2011129643A (ru) | 2013-01-27 |
CA2746190A1 (fr) | 2010-06-24 |
RU2480240C2 (ru) | 2013-04-27 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MY153921A (en) | Aminopyrazole derivatives | |
HK1128471A1 (en) | Heterocyclic non-nucleoside compounds, their preparation, pharmaceutical composition and their use as antiviral agents | |
MX2010004576A (es) | Derivados de pirimidina novedosos. | |
MX2010005889A (es) | Derivados de tiofeno como agonistas de s1p1/edg1. | |
DK2321321T3 (da) | Triazolo [4,5-d]pyramidinderivater og anvendelse deraf som purinreceptorantagonister | |
MX2009009597A (es) | Derivados de amino-piridina como agonistas del receptor s1p1/edg1. | |
MX2009007254A (es) | Composiciones de tableta en tableta. | |
MY154909A (en) | Novel thiophene derivatives | |
MY153975A (en) | Pyridine derivatives as s1p1/edg1 receptor modulators | |
WO2007098128A3 (fr) | Formules liquides de phényléphrine | |
MY149869A (en) | Thiophene derivatives as s1p1/edg1 receptor agonists | |
MY153985A (en) | Aminotriazole derivatives as alx agonists | |
IL192948A0 (en) | Novel pyridine derivatives | |
DOP2011000354A (es) | Composiciones sublinguales de dexmedetomidina y metodos de uso de ellas | |
WO2009063222A3 (fr) | Compositions solides | |
MA33022B1 (fr) | Composition à libération contrôlée pour produire une préparation à libération prolongée contenant de l'udénafil | |
TW200942524A (en) | Novel aminomethyl benzene derivatives | |
MX2010001574A (es) | Ligandos del receptor cannabinoide. | |
JO2831B1 (en) | Quinclidine carbonate derivatives and pharmaceutical compounds | |
TW200942530A (en) | Pyridine compounds | |
UA103025C2 (ru) | Твердая композиция лекарственного средства замедленного высвобождения | |
EA200601759A1 (ru) | Композиции рамиприла | |
MX2010000266A (es) | Un método para disminuir los síntomas del consumo de alcohol. | |
MX2009010689A (es) | Formulaciones novedosas para el suministro de agentes terapeuticos de peptidos antivirales. | |
IL191758A0 (en) | Composition with sustained release of the active ingredient, process for the preparation thereof and use thereof |