MA26703A1 - Macrolides antibiotiques nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant - Google Patents

Macrolides antibiotiques nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant

Info

Publication number
MA26703A1
MA26703A1 MA25832A MA25832A MA26703A1 MA 26703 A1 MA26703 A1 MA 26703A1 MA 25832 A MA25832 A MA 25832A MA 25832 A MA25832 A MA 25832A MA 26703 A1 MA26703 A1 MA 26703A1
Authority
MA
Morocco
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
novel antibiotic
macrolides
Prior art date
Application number
MA25832A
Other languages
English (en)
Inventor
Kaneko Takushi
Original Assignee
Pfizer Products Inc Etat De Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc Etat De Co filed Critical Pfizer Products Inc Etat De Co
Publication of MA26703A1 publication Critical patent/MA26703A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Urology & Nephrology (AREA)
  • Genetics & Genomics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

DEPOSANT Société dite : PFIZER PRODUCTS INC REVENDICATION DE PRIORITES US 03/11/1998 60/106,836 Voir en annexe le titre de l'invention et le texte de l'abrégé Macrolides antibiotiques nouveaux, procédé pour leur préparation et compositions pharmaceutiqueS les contenant La présente invention concerne des composés répondant à la formule : dans laquelle a est égal à 0 ou 1, et R1, R2, R3, R4, R5, R6 et X représentent divers radicaux. Elle concerne également un procédé pour leur préparation et des compositions pharmaceutiques les contenant. Application : utilisation de ces composés et compositions pour le traitement d'infections par des bactéries et des protozoaires.
MA25832A 1998-11-03 1999-11-02 Macrolides antibiotiques nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant MA26703A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10683698P 1998-11-03 1998-11-03

Publications (1)

Publication Number Publication Date
MA26703A1 true MA26703A1 (fr) 2004-12-20

Family

ID=22313524

Family Applications (1)

Application Number Title Priority Date Filing Date
MA25832A MA26703A1 (fr) 1998-11-03 1999-11-02 Macrolides antibiotiques nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant

Country Status (34)

Country Link
US (3) US20020040007A1 (fr)
EP (1) EP1124837A2 (fr)
JP (1) JP4043191B2 (fr)
KR (1) KR20010083944A (fr)
CN (1) CN1376160A (fr)
AP (1) AP2001002131A0 (fr)
AU (1) AU5995299A (fr)
BG (1) BG105543A (fr)
BR (1) BR9914998A (fr)
CA (1) CA2349338C (fr)
CO (1) CO5140110A1 (fr)
CZ (1) CZ20011512A3 (fr)
EA (1) EA200100396A1 (fr)
EE (1) EE200100245A (fr)
GT (1) GT199900192A (fr)
HK (1) HK1049010A1 (fr)
HR (1) HRP20010306A2 (fr)
HU (1) HUP0104192A3 (fr)
ID (1) ID28286A (fr)
IL (1) IL142628A0 (fr)
IS (1) IS5919A (fr)
MA (1) MA26703A1 (fr)
NO (1) NO20012155L (fr)
OA (1) OA11670A (fr)
PA (1) PA8485101A1 (fr)
PE (1) PE20001289A1 (fr)
PL (1) PL348114A1 (fr)
SK (1) SK5812001A3 (fr)
SV (1) SV1999000188A (fr)
TN (1) TNSN99205A1 (fr)
TR (4) TR200200435T2 (fr)
UY (1) UY25780A1 (fr)
WO (1) WO2000026224A2 (fr)
ZA (1) ZA200103289B (fr)

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AP9801420A0 (en) * 1998-01-02 1998-12-31 Pfizer Prod Inc Novel macrolides.
BR9914998A (pt) 1998-11-03 2001-07-10 Pfizer Prod Inc Antibióticos macrólidos
ATE256694T1 (de) 1999-01-27 2004-01-15 Pfizer Prod Inc Ketolid-antibiotika
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
JP2003523938A (ja) 1999-04-16 2003-08-12 コーサン バイオサイエンシーズ, インコーポレイテッド マクロライド系抗感染剤
US6939861B2 (en) 1999-04-16 2005-09-06 Kosan Biosciences, Inc. Amido macrolides
US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
US6458771B1 (en) 1999-04-16 2002-10-01 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
US6514944B2 (en) 1999-04-16 2003-02-04 Kosan Biosciences, Inc. Macrolide antiinfective agents
EA200100983A1 (ru) 1999-05-24 2002-10-31 Пфайзер Продактс Инк. Производные 13-метилэритромицина
EP1114826A3 (fr) * 1999-12-29 2001-10-31 Pfizer Products Inc. Macrolides antibactériennes et prokinétiques
EP1146051A3 (fr) * 2000-04-10 2001-10-31 Pfizer Products Inc. Dérivées de l' érythromycine A
DK1167376T3 (da) * 2000-06-30 2004-10-25 Pfizer Prod Inc Makrolidantibiotika
JP2008508322A (ja) * 2004-07-28 2008-03-21 ランバクシー ラボラトリーズ リミテッド 抗菌剤としてのケトライド誘導体
EP1807439A2 (fr) * 2004-10-25 2007-07-18 Ranbaxy Laboratories Limited Derives de cetolides utiles comme agents antibacteriens
ES2339871T3 (es) 2004-12-21 2010-05-26 Pfizer Products Inc. Macrolidos.
US20090130225A1 (en) * 2005-11-23 2009-05-21 Anjan Chakrabarti Macrolides derivatives as antibacterial agents
US20090005325A1 (en) * 2005-11-23 2009-01-01 Biswajit Bas Ketolide Derivatives as Antibacterial Agents
US7801502B2 (en) * 2006-12-18 2010-09-21 Aai Corporation Method for implementing continuous radio frequency (RF) alignment in advanced electronic warfare (EW) signal stimulation systems
US8409628B2 (en) 2010-02-04 2013-04-02 Penguin IP Holdings, Inc. Methods and compositions for oxygenation of skin to treat skin disorders
WO2011123619A2 (fr) 2010-03-31 2011-10-06 Penguin Ip Holdings Inc. Mélanges perméables, procédés et compositions pour la peau
CN105358141A (zh) * 2013-05-01 2016-02-24 尼奥酷里私人有限公司 治疗细菌感染的方法
RU2537143C1 (ru) * 2013-11-08 2014-12-27 Государственное научное учреждение Ставропольский научно-исследовательский институт животноводства и кормопроизводства РАСХН Препарат для лечения и профилактики мастита у коров
WO2018080072A2 (fr) * 2016-10-27 2018-05-03 한국생명공학연구원 Nouveau composé à base de macrolide, son procédé de production, et composition pharmaceutique destinée à prévenir ou à traiter le paludisme et le contenant à titre de principe actif

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IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of the history of erythromycin
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FR2697524B1 (fr) 1992-11-05 1994-12-23 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
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PL191087B1 (pl) 1997-10-16 2006-03-31 Pliva Farmaceutska Ind 3,6-hemiketale oraz sposób ich wytwarzania
PT941998E (pt) * 1998-03-03 2004-12-31 Pfizer Prod Inc Antibioticos macrolidos do tipo 3,6-cetal
BR9914998A (pt) 1998-11-03 2001-07-10 Pfizer Prod Inc Antibióticos macrólidos
EA200100983A1 (ru) 1999-05-24 2002-10-31 Пфайзер Продактс Инк. Производные 13-метилэритромицина
EP1114826A3 (fr) 1999-12-29 2001-10-31 Pfizer Products Inc. Macrolides antibactériennes et prokinétiques
EP1122261A3 (fr) 2000-01-31 2001-09-26 Pfizer Products Inc. Macrolides antibactériennes à 13 ou 14 chainons
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AU2002316550A1 (en) 2001-07-03 2003-01-21 Chiron Corporation C12 modified erythromycin macrolides and ketolides having antibacterial activity

Also Published As

Publication number Publication date
US7071170B2 (en) 2006-07-04
HUP0104192A2 (hu) 2002-02-28
WO2000026224A2 (fr) 2000-05-11
SV1999000188A (es) 2000-10-16
ID28286A (id) 2001-05-10
TR200200436T2 (tr) 2002-06-21
EP1124837A2 (fr) 2001-08-22
BR9914998A (pt) 2001-07-10
WO2000026224A3 (fr) 2000-11-16
AU5995299A (en) 2000-05-22
PE20001289A1 (es) 2000-11-22
NO20012155D0 (no) 2001-05-02
CZ20011512A3 (cs) 2001-09-12
JP2002528553A (ja) 2002-09-03
NO20012155L (no) 2001-07-02
TR200200435T2 (tr) 2002-07-22
ZA200103289B (en) 2002-08-28
PA8485101A1 (es) 2002-08-26
AP2001002131A0 (en) 2001-06-30
PL348114A1 (en) 2002-05-06
US20030013665A1 (en) 2003-01-16
SK5812001A3 (en) 2001-12-03
EA200100396A1 (ru) 2001-10-22
UY25780A1 (es) 2001-08-27
KR20010083944A (ko) 2001-09-03
US20050004047A1 (en) 2005-01-06
HK1049010A1 (zh) 2003-04-25
HUP0104192A3 (en) 2003-12-29
TR200200434T2 (tr) 2002-09-23
IS5919A (is) 2001-04-17
OA11670A (en) 2005-01-12
CN1376160A (zh) 2002-10-23
TNSN99205A1 (fr) 2005-11-10
US6835716B2 (en) 2004-12-28
JP4043191B2 (ja) 2008-02-06
HRP20010306A2 (en) 2002-06-30
IL142628A0 (en) 2002-03-10
CO5140110A1 (es) 2002-03-22
CA2349338C (fr) 2005-12-06
EE200100245A (et) 2002-10-15
US20020040007A1 (en) 2002-04-04
TR200101241T2 (tr) 2001-09-21
BG105543A (en) 2001-12-29
GT199900192A (es) 2001-04-26
CA2349338A1 (fr) 2000-05-11

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