MA26690A1 - COMPOSITIONS PHARMACEUTIQUES CONTENANT DES DERIVES DE PYRIDO [1,2-a ] PYRAZINE ET PROCEDE POUR LEUR PREPARATION - Google Patents

COMPOSITIONS PHARMACEUTIQUES CONTENANT DES DERIVES DE PYRIDO [1,2-a ] PYRAZINE ET PROCEDE POUR LEUR PREPARATION

Info

Publication number
MA26690A1
MA26690A1 MA25774A MA25774A MA26690A1 MA 26690 A1 MA26690 A1 MA 26690A1 MA 25774 A MA25774 A MA 25774A MA 25774 A MA25774 A MA 25774A MA 26690 A1 MA26690 A1 MA 26690A1
Authority
MA
Morocco
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
pyrazine
derivatives
Prior art date
Application number
MA25774A
Other languages
English (en)
Inventor
Howard Zorn Stevin
Mclean Stafford
Rose Jackson Elisa
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of MA26690A1 publication Critical patent/MA26690A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Abstract

DEPOSANT Société dite : PFIZER PRODUCTS INC. REVENDICATION DE PRIORITES US 21/09/1998 60/101,191 US 12/10/1998 60/103,868 Voir en annexe le titre de l'invention et le texte de l'abrégé "Compositions pharmaceutiques contenant des dérivés de pyrido [1,2-a]pyrazine et procédé pour leur préparation' L'invention concerne des compositions pharmaceutiques contenant des composés de formule (I) dans laquelle X et Y représentent divers radicaux. Elle concerne également un procédé pour leur préparation. Application : Utilisation de ces compositions dans le traitement de la maladie de Parkinson, du trouble d'hyperactivite par défaut d'attention et de microadénomes chez des mammifères.
MA25774A 1998-09-21 1999-09-20 COMPOSITIONS PHARMACEUTIQUES CONTENANT DES DERIVES DE PYRIDO [1,2-a ] PYRAZINE ET PROCEDE POUR LEUR PREPARATION MA26690A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10119198P 1998-09-21 1998-09-21
US10386898P 1998-10-12 1998-10-12

Publications (1)

Publication Number Publication Date
MA26690A1 true MA26690A1 (fr) 2004-12-20

Family

ID=26798000

Family Applications (1)

Application Number Title Priority Date Filing Date
MA25774A MA26690A1 (fr) 1998-09-21 1999-09-20 COMPOSITIONS PHARMACEUTIQUES CONTENANT DES DERIVES DE PYRIDO [1,2-a ] PYRAZINE ET PROCEDE POUR LEUR PREPARATION

Country Status (38)

Country Link
US (2) US6300329B1 (fr)
EP (1) EP1115402A1 (fr)
JP (1) JP2002526448A (fr)
KR (3) KR20040054752A (fr)
CN (1) CN1319013A (fr)
AP (1) AP1456A (fr)
AR (1) AR029739A1 (fr)
AU (1) AU760230B2 (fr)
BG (1) BG105445A (fr)
BR (1) BR9913975A (fr)
CA (1) CA2344670A1 (fr)
CO (1) CO5140075A1 (fr)
CZ (1) CZ20011006A3 (fr)
DZ (1) DZ2894A1 (fr)
EA (2) EA200100204A1 (fr)
EE (1) EE200100179A (fr)
GE (1) GEP20033081B (fr)
GT (1) GT199900154A (fr)
HN (1) HN1999000146A (fr)
HR (1) HRP20010209A2 (fr)
HU (1) HUP0103691A3 (fr)
ID (1) ID28028A (fr)
IL (2) IL164839A0 (fr)
IS (1) IS5852A (fr)
MA (1) MA26690A1 (fr)
MY (1) MY127939A (fr)
NO (1) NO20011409L (fr)
NZ (1) NZ509855A (fr)
OA (1) OA11653A (fr)
PA (1) PA8482001A1 (fr)
PE (1) PE20001084A1 (fr)
PL (1) PL346904A1 (fr)
SK (1) SK3592001A3 (fr)
TN (1) TNSN99177A1 (fr)
TR (2) TR200402083T2 (fr)
TW (1) TW518225B (fr)
WO (1) WO2000016777A1 (fr)
YU (1) YU21701A (fr)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1999000146A (es) * 1998-09-21 2000-11-11 Pfizer Prod Inc Agentes farmaceuticos para el tratamiento de la enfermedad de parkinson, adhd y microadenomas.
US8030294B2 (en) * 2000-03-16 2011-10-04 The Mclean Hospital Corporation Compounds for the treatment of psychiatric or substance abuse disorders
GB0027020D0 (en) * 2000-11-03 2000-12-20 Univ Manchester Treatment of movement disorders
US7053092B2 (en) 2001-01-29 2006-05-30 Otsuka Pharmaceutical Co., Ltd. 5-HT1a receptor subtype agonist
US7132287B2 (en) 2001-06-18 2006-11-07 Psychiatric Genomics, Inc. Method for neural stem cell differentiation using 5HT-1A agonists
US20030036555A1 (en) * 2001-08-03 2003-02-20 Boehringer Ingelheim Pharma Kg Pramipexole for the treatment of ADHD
AR033485A1 (es) 2001-09-25 2003-12-26 Otsuka Pharma Co Ltd Sustancia medicinal de aripiprazol de baja higroscopicidad y proceso para la preparacion de la misma
US7737128B2 (en) * 2004-06-10 2010-06-15 The Mclean Hospital Corporation Pyrimidines, such as uridine, in treatments for patients with bipolar disorder
WO2006020703A1 (fr) * 2004-08-11 2006-02-23 The Mclean Hospital Corporation Compose pour le traitement de la dependance, de la suppression et de l'usage de la marijuana
MY148644A (en) 2005-07-18 2013-05-15 Orion Corp New pharmaceutical compounds
GT200600414A (es) 2005-09-12 2007-09-20 Sal de glucuranato de compuesto de piperazine
TW200800306A (en) 2005-09-12 2008-01-01 Wyeth Corp Sustained-release formulation and uses thereof
GT200600416A (es) 2005-09-12 2007-09-20 Sales salicilato y gentisato de un compuesto de piperazina
US9066903B2 (en) * 2006-02-28 2015-06-30 The United States Of America As Represented By The Department Of Veterans Affairs Pharmacological treatment of Parkinson's disease
US20080131492A1 (en) * 2006-06-23 2008-06-05 Spherics, Inc. Dosage forms for movement disorder treatment
WO2008083442A1 (fr) * 2007-01-10 2008-07-17 Brc Operations Pty Limited Procédé pour la formulation de médicaments mixtes contre tdah
CN101318020B (zh) * 2007-06-06 2011-09-28 四川科瑞德制药有限公司 抗焦虑或/和抗抑郁的药物组合物及用途
US20100041621A1 (en) * 2008-08-15 2010-02-18 Perry Renshaw Methods and compositions for improving cognitive performance
GB201112987D0 (en) 2011-07-28 2011-09-14 Ge Healthcare Ltd Novel compound
WO2014078568A1 (fr) 2012-11-14 2014-05-22 The Johns Hopkins University Méthodes et compositions pour le traitement de la schizophrénie
WO2014172372A1 (fr) 2013-04-15 2014-10-23 Northwestern University Traitement de troubles dopaminergiques
CN104892589A (zh) 2014-03-07 2015-09-09 中国科学院上海药物研究所 一类杂环化合物、其制备方法和用途
US11426366B2 (en) 2015-05-15 2022-08-30 Arizona Board Of Regents On Behalf Of The Universsity Of Arizona Compositions and methods for treating motor disorders

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX19222A (es) * 1989-01-23 1993-12-01 Pfizer Agentes ansioliticos bis-aza-biciclicos
WO1992000075A1 (fr) * 1990-06-29 1992-01-09 Pfizer Inc. Derives de pyridopyrazine utilises dans le traitement de l'abus et de la dependance de substances
US5281607B1 (en) * 1992-10-08 1998-05-19 Univ New York Method of using alpha 2-antagonists for the treatment of neurodegenerative diseases
GB9408084D0 (en) * 1994-04-23 1994-06-15 Boots Co Plc Medical treatment
ES2163506T3 (es) * 1994-06-14 2002-02-01 Pfizer Derivados de bencimidazolona con actividad dopaminergica central.
US5877183A (en) * 1996-06-06 1999-03-02 Ergo Research Corporation Treatment of lipid and glucose metabolism disorders with dopamine and serotonin agonists
HN1999000146A (es) * 1998-09-21 2000-11-11 Pfizer Prod Inc Agentes farmaceuticos para el tratamiento de la enfermedad de parkinson, adhd y microadenomas.

Also Published As

Publication number Publication date
KR100468340B1 (ko) 2005-01-27
KR20030088512A (ko) 2003-11-19
GT199900154A (es) 2001-03-06
SK3592001A3 (en) 2001-12-03
PA8482001A1 (es) 2000-05-24
AU5383199A (en) 2000-04-10
EE200100179A (et) 2002-10-15
DZ2894A1 (fr) 2003-12-15
TR200402083T2 (tr) 2004-10-21
PL346904A1 (en) 2002-03-11
KR20010075222A (ko) 2001-08-09
IL164839A0 (en) 2005-12-18
YU21701A (sh) 2004-07-15
CO5140075A1 (es) 2002-03-22
KR20040054752A (ko) 2004-06-25
US20010034347A1 (en) 2001-10-25
HUP0103691A3 (en) 2003-01-28
GEP20033081B (en) 2003-10-27
ID28028A (id) 2001-05-03
NO20011409D0 (no) 2001-03-20
NZ509855A (en) 2003-04-29
CN1319013A (zh) 2001-10-24
EA200301063A1 (ru) 2004-12-30
HUP0103691A2 (hu) 2002-02-28
TR200101357T2 (tr) 2001-08-21
BG105445A (en) 2001-12-29
BR9913975A (pt) 2001-06-19
AP2001002102A0 (en) 2001-03-31
IS5852A (is) 2001-02-20
HRP20010209A2 (en) 2002-04-30
EP1115402A1 (fr) 2001-07-18
OA11653A (en) 2004-12-08
CA2344670A1 (fr) 2000-03-30
AR029739A1 (es) 2003-07-16
CZ20011006A3 (cs) 2001-09-12
JP2002526448A (ja) 2002-08-20
TNSN99177A1 (fr) 2005-11-10
TW518225B (en) 2003-01-21
HN1999000146A (es) 2000-11-11
US6300329B1 (en) 2001-10-09
WO2000016777A1 (fr) 2000-03-30
EA200100204A1 (ru) 2001-08-27
PE20001084A1 (es) 2000-10-18
AP1456A (en) 2005-09-30
NO20011409L (no) 2001-03-28
US6608064B2 (en) 2003-08-19
IL141507A0 (en) 2002-03-10
AU760230B2 (en) 2003-05-08
MY127939A (en) 2007-01-31

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