LU82082A1 - Carbamates de mercaptoacyl hydroxy prolines,a action antihypertensive - Google Patents

Carbamates de mercaptoacyl hydroxy prolines,a action antihypertensive Download PDF

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Publication number
LU82082A1
LU82082A1 LU82082A LU82082A LU82082A1 LU 82082 A1 LU82082 A1 LU 82082A1 LU 82082 A LU82082 A LU 82082A LU 82082 A LU82082 A LU 82082A LU 82082 A1 LU82082 A1 LU 82082A1
Authority
LU
Luxembourg
Prior art keywords
methyl
proline
oxy
radical
carbonyl
Prior art date
Application number
LU82082A
Other languages
English (en)
French (fr)
Inventor
J Krapcho
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of LU82082A1 publication Critical patent/LU82082A1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
LU82082A 1979-01-15 1980-01-14 Carbamates de mercaptoacyl hydroxy prolines,a action antihypertensive LU82082A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US317879A 1979-01-15 1979-01-15
US317879 1979-01-15

Publications (1)

Publication Number Publication Date
LU82082A1 true LU82082A1 (fr) 1980-04-23

Family

ID=21704564

Family Applications (1)

Application Number Title Priority Date Filing Date
LU82082A LU82082A1 (fr) 1979-01-15 1980-01-14 Carbamates de mercaptoacyl hydroxy prolines,a action antihypertensive

Country Status (21)

Country Link
JP (2) JPS5598161A (de)
AT (1) AT364377B (de)
AU (1) AU526767B2 (de)
BE (1) BE881153A (de)
CA (1) CA1138452A (de)
CH (2) CH646950A5 (de)
DE (1) DE3001113A1 (de)
DK (1) DK14980A (de)
FR (1) FR2446281A1 (de)
GB (2) GB2040937B (de)
GR (1) GR73002B (de)
HU (2) HU182778B (de)
IE (1) IE49357B1 (de)
IT (1) IT1140505B (de)
LU (1) LU82082A1 (de)
NL (1) NL8000206A (de)
NO (1) NO800077L (de)
NZ (1) NZ192522A (de)
PH (2) PH14946A (de)
SE (1) SE8000298L (de)
ZA (1) ZA8035B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4316905A (en) * 1980-07-01 1982-02-23 E. R. Squibb & Sons, Inc. Mercaptoacyl derivatives of various 4-substituted prolines
ZA832762B (en) * 1982-04-30 1983-12-28 Squibb & Sons Inc Substituted 4-phenoxy prolines

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4052511A (en) * 1976-02-13 1977-10-04 E. R. Squibb & Sons, Inc. Carboxyacylproline derivatives
US4046889A (en) * 1976-02-13 1977-09-06 E. R. Squibb & Sons, Inc. Azetidine-2-carboxylic acid derivatives
AU509899B2 (en) * 1976-02-13 1980-05-29 E.R. Squibb & Sons, Inc. Proline derivatives and related compounds

Also Published As

Publication number Publication date
FR2446281B1 (de) 1984-01-20
ATA19080A (de) 1981-03-15
CA1138452A (en) 1982-12-28
JPH0125744B2 (de) 1989-05-19
AU526767B2 (en) 1983-01-27
NL8000206A (nl) 1980-07-17
IE49357B1 (en) 1985-09-18
AT364377B (de) 1981-10-12
JPH0378378B2 (de) 1991-12-13
IT8019209A0 (it) 1980-01-14
ZA8035B (en) 1980-12-31
GB2040937A (en) 1980-09-03
FR2446281A1 (fr) 1980-08-08
BE881153A (fr) 1980-07-15
GR73002B (de) 1984-01-24
SE8000298L (sv) 1980-07-16
HU182778B (en) 1984-03-28
DK14980A (da) 1980-07-16
DE3001113A1 (de) 1980-07-24
GB2040937B (en) 1982-11-24
IE800048L (en) 1980-07-15
AU5432780A (en) 1980-07-24
JPH01301656A (ja) 1989-12-05
CH646690A5 (de) 1984-12-14
NO800077L (no) 1980-07-16
NZ192522A (en) 1982-06-29
JPS5598161A (en) 1980-07-25
IT1140505B (it) 1986-10-01
PH15318A (en) 1982-11-18
HU179621B (en) 1982-11-29
GB2088875B (en) 1983-06-08
GB2088875A (en) 1982-06-16
CH646950A5 (de) 1984-12-28
PH14946A (en) 1982-02-02

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