LT3507291T - Kondensuoti bicikliniai sgc stimuliatoriai - Google Patents

Kondensuoti bicikliniai sgc stimuliatoriai

Info

Publication number
LT3507291T
LT3507291T LTEP17768311.7T LT17768311T LT3507291T LT 3507291 T LT3507291 T LT 3507291T LT 17768311 T LT17768311 T LT 17768311T LT 3507291 T LT3507291 T LT 3507291T
Authority
LT
Lithuania
Prior art keywords
condensed bicyclic
sgc stimulators
sgc
stimulators
bicyclic
Prior art date
Application number
LTEP17768311.7T
Other languages
English (en)
Lithuanian (lt)
Inventor
Glen Rennie
Rajesh Iyengar
Thomas Lee
Takashi Nakai
Ara Mermerian
Lei Jia
G-Yoon IM
Paul Renhowe
Joon Jung
Peter Germano
Karthik Iyer
Timothy Barden
Kim TANG
Original Assignee
Cyclerion Therapeutics, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cyclerion Therapeutics, Inc. filed Critical Cyclerion Therapeutics, Inc.
Publication of LT3507291T publication Critical patent/LT3507291T/lt

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41881,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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LTEP17768311.7T 2016-09-02 2017-09-01 Kondensuoti bicikliniai sgc stimuliatoriai LT3507291T (lt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662382942P 2016-09-02 2016-09-02
US201662423445P 2016-11-17 2016-11-17
US201762468598P 2017-03-08 2017-03-08
US201762482486P 2017-04-06 2017-04-06
PCT/US2017/049834 WO2018045276A1 (en) 2016-09-02 2017-09-01 Fused bicyclic sgc stimulators

Publications (1)

Publication Number Publication Date
LT3507291T true LT3507291T (lt) 2021-09-10

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LTEP17768311.7T LT3507291T (lt) 2016-09-02 2017-09-01 Kondensuoti bicikliniai sgc stimuliatoriai

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US (5) US10472363B2 (https=)
EP (2) EP3872080B1 (https=)
JP (2) JP7050759B2 (https=)
KR (2) KR102854313B1 (https=)
CN (2) CN117105939B (https=)
AU (2) AU2017321810B2 (https=)
CA (1) CA3035210A1 (https=)
CL (1) CL2019000486A1 (https=)
CO (1) CO2019001760A2 (https=)
CR (2) CR20220309A (https=)
CY (1) CY1124612T1 (https=)
DK (1) DK3507291T3 (https=)
ES (2) ES2957159T3 (https=)
HR (1) HRP20211355T1 (https=)
HU (1) HUE056051T2 (https=)
IL (2) IL292968B2 (https=)
LT (1) LT3507291T (https=)
MA (1) MA53999A (https=)
MX (3) MX383782B (https=)
MY (1) MY199759A (https=)
PE (1) PE20190607A1 (https=)
PH (1) PH12019500461B1 (https=)
PL (1) PL3507291T3 (https=)
PT (1) PT3507291T (https=)
RS (1) RS62256B1 (https=)
SG (1) SG11201901729YA (https=)
SI (1) SI3507291T1 (https=)
TW (2) TWI813078B (https=)
WO (1) WO2018045276A1 (https=)

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EP0890989A4 (en) * 1997-01-24 2006-11-02 Rohm Co Ltd SEMICONDUCTOR DEVICE AND MANUFACTURING METHOD
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