KR920003902B1 - 페니실린 유도체의 수화물 및 그 제조방법 - Google Patents

페니실린 유도체의 수화물 및 그 제조방법 Download PDF

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Publication number
KR920003902B1
KR920003902B1 KR1019870010566A KR870010566A KR920003902B1 KR 920003902 B1 KR920003902 B1 KR 920003902B1 KR 1019870010566 A KR1019870010566 A KR 1019870010566A KR 870010566 A KR870010566 A KR 870010566A KR 920003902 B1 KR920003902 B1 KR 920003902B1
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KR
South Korea
Prior art keywords
methyl
solution
asparazinylamoxicillin
trihydrate
water
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Expired
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KR1019870010566A
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English (en)
Korean (ko)
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KR880003955A (ko
Inventor
스스무 오오시로
마사루 세누마
미쓰요시 와가쓰마
Original Assignee
다나베 세이야꾸 가부시기가이샤
아다찌 게이지로오
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Publication of KR880003955A publication Critical patent/KR880003955A/ko
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Publication of KR920003902B1 publication Critical patent/KR920003902B1/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04—Preparation
    • C07D499/18—Separation; Purification
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
    • C07D499/68—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
KR1019870010566A 1986-09-24 1987-09-24 페니실린 유도체의 수화물 및 그 제조방법 Expired KR920003902B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP226423 1986-09-24
JP61226423A JPS6379888A (ja) 1986-09-24 1986-09-24 ペニシリン誘導体の安定型水和物

Publications (2)

Publication Number Publication Date
KR880003955A KR880003955A (ko) 1988-05-31
KR920003902B1 true KR920003902B1 (ko) 1992-05-18

Family

ID=16844890

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019870010566A Expired KR920003902B1 (ko) 1986-09-24 1987-09-24 페니실린 유도체의 수화물 및 그 제조방법

Country Status (24)

Country Link
US (1) US4866170A (enExample)
EP (1) EP0261823B1 (enExample)
JP (1) JPS6379888A (enExample)
KR (1) KR920003902B1 (enExample)
CN (1) CN1021225C (enExample)
AT (2) ATE59655T1 (enExample)
AU (1) AU592467B2 (enExample)
CA (1) CA1286285C (enExample)
DE (1) DE3766921D1 (enExample)
DK (1) DK167319B1 (enExample)
ES (1) ES2026545T3 (enExample)
FI (1) FI86853C (enExample)
GR (1) GR3001274T3 (enExample)
HK (1) HK42093A (enExample)
HU (1) HU196810B (enExample)
IE (1) IE60042B1 (enExample)
IL (1) IL83786A (enExample)
MY (1) MY102553A (enExample)
NO (1) NO169717C (enExample)
PH (1) PH23644A (enExample)
PT (1) PT85773B (enExample)
SG (1) SG15393G (enExample)
SU (1) SU1517764A3 (enExample)
ZA (1) ZA876739B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5375123A (en) * 1993-02-05 1994-12-20 Telefonakitebolaget L. M. Ericsson Allocation of channels using interference estimation
US6473602B1 (en) 1996-10-28 2002-10-29 Ericsson Inc. Mobile assisted handoff in radiocommunication systems
PE20000879A1 (es) * 1998-04-29 2000-09-23 Dsm Nv METODO PARA CRISTALIZAR UN ANTIBIOTICO ß-LACTAMICO
KR101879756B1 (ko) * 2016-11-30 2018-08-17 주식회사 지앤지비 욕실용 난방기

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL6705789A (enExample) * 1967-03-08 1968-09-09
GB1241844A (en) * 1968-08-23 1971-08-04 Beecham Group Ltd Penicillins
US4053609A (en) * 1975-09-12 1977-10-11 Tanabe Seiyaku Co., Ltd. Penicillins and processes for preparing the same
JPS5640686A (en) * 1979-09-11 1981-04-16 Tanabe Seiyaku Co Ltd Purification of penicillin derivative

Also Published As

Publication number Publication date
IL83786A0 (en) 1988-02-29
SU1517764A3 (ru) 1989-10-23
MY102553A (en) 1992-07-31
JPS6379888A (ja) 1988-04-09
DE3766921D1 (de) 1991-02-07
AT389311B (de) 1989-11-27
HUT45263A (en) 1988-06-28
HK42093A (en) 1993-05-07
FI874152A0 (fi) 1987-09-23
AU592467B2 (en) 1990-01-11
PT85773B (pt) 1990-07-31
US4866170A (en) 1989-09-12
GR3001274T3 (en) 1992-08-25
IL83786A (en) 1991-11-21
IE872346L (en) 1988-03-14
HU196810B (en) 1989-01-30
ATA273187A (de) 1989-04-15
EP0261823A1 (en) 1988-03-30
JPH0448795B2 (enExample) 1992-08-07
FI86853C (fi) 1992-10-26
ATE59655T1 (de) 1991-01-15
IE60042B1 (en) 1994-05-18
EP0261823B1 (en) 1991-01-02
NO873969L (no) 1988-03-25
FI874152L (fi) 1988-03-25
DK500887D0 (da) 1987-09-23
CA1286285C (en) 1991-07-16
ES2026545T3 (es) 1992-05-01
DK500887A (da) 1988-03-25
KR880003955A (ko) 1988-05-31
AU7882787A (en) 1988-03-31
NO873969D0 (no) 1987-09-23
SG15393G (en) 1993-04-16
DK167319B1 (da) 1993-10-11
ZA876739B (en) 1988-03-14
NO169717B (no) 1992-04-21
CN1021225C (zh) 1993-06-16
PT85773A (en) 1987-10-01
PH23644A (en) 1989-09-27
FI86853B (fi) 1992-07-15
NO169717C (no) 1992-07-29
CN87106308A (zh) 1988-04-13

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