KR860007237A - 이소프레노이드아민 유도체의 제조방법 - Google Patents

이소프레노이드아민 유도체의 제조방법 Download PDF

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KR860007237A
KR860007237A KR1019860001919A KR860001919A KR860007237A KR 860007237 A KR860007237 A KR 860007237A KR 1019860001919 A KR1019860001919 A KR 1019860001919A KR 860001919 A KR860001919 A KR 860001919A KR 860007237 A KR860007237 A KR 860007237A
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alkyl
phenyl
group
alkoxy
iii
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KR1019860001919A
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KR910002687B1 (ko
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사이찌 마쓰모또
마사미 도떼우찌
다꾸지 미즈이
겐따로 히라이
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시오노기 세이야꾸 가부시끼가이샤
요시또시 가즈오
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
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    • C07D209/26—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with an acyl radical attached to the ring nitrogen atom
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Abstract

내용 없음

Description

이소프레노이드아민 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (1)

  1. 하기 일반식(Ⅱ)의 화합물과 하기 일반식(Ⅲ)의 화합물 또는 그의 반응성 유도체를 반응시켜서 하기일반식(A)의 화합물을 제조함을 특징으로 하는 방법
    식중, n은 1∼6의 정수이고 ; R은 (ⅰ) 수소, (ⅱ) 할로겐, 시아노, 페닐, C1∼C5알킬-페닐, 페녹시, 벤즈아미도, 디(C1∼C5알킬)아미노, C1∼C5알콕시, 및 5- 또는 6-원자 헤테로고리기로 구성된 군 중에서 선택된 어느 한가지에 의해 임의로 치환된 C1∼C15알킬, (ⅲ) 페닐 및 5-또는 6-원자 헤테로 고리기로 구성된 군중에서 선택된 어느 한가지에 의해 임의로 치환된 C2∼C5알케닐, (ⅳ) C4∼C12알카디에닐, (ⅴ)할로겐, C1∼C5알킬, C1∼C5알콕시, C1∼C5알카노일옥시, 디(C1∼C5알킬) 아미노, C2∼C6알콕시카르보닐, C1∼C5알킬티오, C1∼C5알킬술피닐, C1∼C5) 알킬술포닐, 니트로 및 히드록시로 구성된 군중에서 선택된 어느 한가지에 의해 임의로 치환된 아릴, (ⅵ)디(C1∼C5알킬)아미노-(C1∼C5알킬), 페닐(C1∼C5알킬), 할로게노페닐(C1∼C5알킬), 3,4-메틸렌디옥시페닐(C1∼C5알킬), 모름폴리닐(C1∼C5알킬), 피리딜-(C1∼C5알킬), 페닐, 할로게노페닐, 트리플루오르메틸페닐, C1∼C5알콕시-페닐, 피리딜 및 C1∼C5알킬로 구성된 군중에서 선택된 어느 한가지에 의해 임의로 치환된 아미노, (ⅶ) C1∼C5알킬, 페닐아미노, 할로게노페닐아미노, 트리플루오로메틸페닐아미노, C1∼C5알콕시페닐아미노, C1∼C5알콕시, C2∼C6알콕시카르보닐, 페닐, 피리딜, 할로게노벤조일, 할로게노벤질 및 3,4-메틸렌디옥시페닐메틸이다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019860001919A 1985-03-15 1986-03-15 이소프레노이드아민 유도체의 제조방법 KR910002687B1 (ko)

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WO2003078448A1 (en) 2002-03-13 2003-09-25 Signum Biosciences, Inc. Modulation of protein methylation and phosphoprotein phosphate
US20050137262A1 (en) * 2003-12-22 2005-06-23 Hu Patrick C. Highly concentrated pourable aqueous solutions of potassium ibuprofen, their preparation and their uses
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GB2172286A (en) 1986-09-17
US4900749A (en) 1990-02-13
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