KR850002472A - 5-피리딜-1,3-티아졸 유도체의 제조방법 - Google Patents

5-피리딜-1,3-티아졸 유도체의 제조방법 Download PDF

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Publication number
KR850002472A
KR850002472A KR1019840005499A KR840005499A KR850002472A KR 850002472 A KR850002472 A KR 850002472A KR 1019840005499 A KR1019840005499 A KR 1019840005499A KR 840005499 A KR840005499 A KR 840005499A KR 850002472 A KR850002472 A KR 850002472A
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KR
South Korea
Prior art keywords
group
optionally substituted
pyridyl
following general
general formula
Prior art date
Application number
KR1019840005499A
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English (en)
Other versions
KR910004430B1 (ko
Inventor
신지 데라오 (외 1)
Original Assignee
구라바야시 이꾸시로
다께다 야꾸힝 고오교 가부시끼가이샤
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Priority claimed from JP16704283A external-priority patent/JPS6058981A/ja
Priority claimed from JP7781984A external-priority patent/JPS6110580A/ja
Application filed by 구라바야시 이꾸시로, 다께다 야꾸힝 고오교 가부시끼가이샤 filed Critical 구라바야시 이꾸시로
Publication of KR850002472A publication Critical patent/KR850002472A/ko
Application granted granted Critical
Publication of KR910004430B1 publication Critical patent/KR910004430B1/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

내용 없음

Description

5-피리딜-1,3-티아졸 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (2)

  1. 다음 일반식(Ⅱ)로 표시되는 화합물과 다음 일반식(Ⅲ)으로 표시되는 화합물을 반응 시킴을 특징으로 하는 다음 일반식(Ⅰ)로 표시되는 1,3-티아졸 유도체 또는 그의 염의 제조방법.
    [식중, R1은 임의로 치환된 알킬기, 알케 닐기, 아릴기, 아랄킬기, 시클로알킬기, 결합손으로서 탄소를 갖는 헤테로고리기 또는 아미노기를 나타내고, R2는 알킬기로 치환될 수 있는 피리딜기를 나타 내고, R3는 임의로 치환된 아릴기를 나타낸다.
    [식중, R2및 R3는 상기에 정의한 것과 같고, X는 할로겐 원자를 나타낸다.]
    [식중, R1은 상기에 정의한 것과 같다.]
  2. 유효 성분으로서, 다음 식(Ⅰ)의 화합물 또는 그의 염의 효과적인 양과 제약에 수용할 수 있는 담체를 함유 함을 특징으로하는 진통, 해열, 소염 및 항궤양 제약 조성물.
    [식중, R1은 임의로 치환된 알킬기, 알케닐기, 아릴기, 아랄킬기, 시클로알킬기, 결합손으로서 탄소를 갖는 헤테로고리기 또는 아미노기를 나타내고, R2는 알킬기로 치환될 수 있는 피리딜기를 나타내고, R3는 임의로 치환된 페닐기를 나타낸다.]
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019840005499A 1983-04-17 1984-09-08 5-피리딜-1,3-티아졸 유도체의 제조방법 KR910004430B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP77819 1983-04-17
JP167042 1983-09-09
JP16704283A JPS6058981A (ja) 1983-09-09 1983-09-09 ５−ピリジル−１，３−チアゾ−ル誘導体，その製造法およびそれを含んでなる医薬組成物
JP7781984A JPS6110580A (ja) 1984-04-17 1984-04-17 ５−ピリジル−１，３−チアゾ−ル誘導体，その製造法およびそれを含んでなる医薬組成物

Publications (2)

Publication Number Publication Date
KR850002472A true KR850002472A (ko) 1985-05-13
KR910004430B1 KR910004430B1 (ko) 1991-06-27

Family

ID=26418876

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019840005499A KR910004430B1 (ko) 1983-04-17 1984-09-08 5-피리딜-1,3-티아졸 유도체의 제조방법

Country Status (7)

Country Link
US (1) US4612321A (ko)
EP (1) EP0149884B1 (ko)
KR (1) KR910004430B1 (ko)
AU (1) AU567754B2 (ko)
CA (1) CA1255663A (ko)
DE (1) DE3486009T2 (ko)
HU (1) HU201753B (ko)

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EP1027050B1 (en) * 1997-10-27 2004-01-14 Takeda Chemical Industries, Ltd. 1,3-thiazoles as adenosine a3 receptor antagonists for the treatment of allergy, asthma and diabetes
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Also Published As

Publication number Publication date
DE3486009D1 (de) 1993-01-28
HUT37424A (en) 1985-12-28
CA1255663A (en) 1989-06-13
AU3243384A (en) 1985-03-14
AU567754B2 (en) 1987-12-03
EP0149884B1 (en) 1992-12-16
US4612321A (en) 1986-09-16
EP0149884A2 (en) 1985-07-31
HU201753B (en) 1990-12-28
EP0149884A3 (en) 1986-07-30
KR910004430B1 (ko) 1991-06-27
DE3486009T2 (de) 1993-04-15

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