KR850001339B1 - 페니실란산 1,1-디옥사이드 및 그의 에스테르의 제조방법 - Google Patents

페니실란산 1,1-디옥사이드 및 그의 에스테르의 제조방법 Download PDF

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Publication number
KR850001339B1
KR850001339B1 KR1019800000885A KR800000885A KR850001339B1 KR 850001339 B1 KR850001339 B1 KR 850001339B1 KR 1019800000885 A KR1019800000885 A KR 1019800000885A KR 800000885 A KR800000885 A KR 800000885A KR 850001339 B1 KR850001339 B1 KR 850001339B1
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KR
South Korea
Prior art keywords
acid
dioxide
solution
added
beta
Prior art date
Application number
KR1019800000885A
Other languages
English (en)
Korean (ko)
Inventor
쉴즈 무어 버나드
디이 캐롤 로니
알프레드 폴크만 로버트
Original Assignee
화이자 인코포레이티드
테렌스 제이. 겔라거
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 화이자 인코포레이티드, 테렌스 제이. 겔라거 filed Critical 화이자 인코포레이티드
Application granted granted Critical
Publication of KR850001339B1 publication Critical patent/KR850001339B1/ko

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
KR1019800000885A 1979-03-05 1980-03-04 페니실란산 1,1-디옥사이드 및 그의 에스테르의 제조방법 KR850001339B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US1780879A 1979-03-05 1979-03-05
US1781079A 1979-03-05 1979-03-05
US17810 1979-03-05
US17808 1979-03-05

Publications (1)

Publication Number Publication Date
KR850001339B1 true KR850001339B1 (ko) 1985-09-19

Family

ID=26690337

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019800000885A KR850001339B1 (ko) 1979-03-05 1980-03-04 페니실란산 1,1-디옥사이드 및 그의 에스테르의 제조방법

Country Status (36)

Country Link
KR (1) KR850001339B1 (es)
AR (1) AR225031A1 (es)
AT (1) AT366693B (es)
AU (1) AU522572B2 (es)
BG (1) BG33292A3 (es)
CH (1) CH644608A5 (es)
CS (1) CS215130B2 (es)
DD (1) DD149367A5 (es)
DE (1) DE3008257C2 (es)
DK (2) DK159852C (es)
EG (1) EG14437A (es)
ES (1) ES8103094A1 (es)
FI (1) FI70024C (es)
FR (1) FR2450836B1 (es)
GB (1) GB2045755B (es)
GR (1) GR67234B (es)
HK (1) HK66587A (es)
HU (1) HU186304B (es)
IE (1) IE49535B1 (es)
IL (1) IL59515A (es)
IN (1) IN153685B (es)
IT (1) IT1130300B (es)
KE (1) KE3464A (es)
LU (1) LU82215A1 (es)
MX (1) MX6032E (es)
MY (1) MY8500319A (es)
NL (1) NL180317C (es)
NO (2) NO800618L (es)
PL (1) PL125197B1 (es)
PT (1) PT70897A (es)
RO (1) RO80112A (es)
SE (2) SE449103B (es)
SG (1) SG55884G (es)
SU (1) SU1192626A3 (es)
UA (1) UA6342A1 (es)
YU (1) YU42328B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN159362B (es) * 1981-03-23 1987-05-09 Pfizer
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
PT76527B (en) * 1982-04-19 1985-12-09 Gist Brocades Nv A process for the preparation of penicillanic acid 1,1-dioxide and derivatives thereof
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139047A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (es) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
EP0013617B1 (en) * 1979-01-10 1984-07-04 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives

Also Published As

Publication number Publication date
ES489185A0 (es) 1981-02-16
GB2045755A (en) 1980-11-05
DK159852B (da) 1990-12-17
NO800618L (no) 1980-09-08
AR225031A1 (es) 1982-02-15
DK166353B (da) 1993-04-13
HK66587A (en) 1987-09-25
AU522572B2 (en) 1982-06-17
GR67234B (es) 1981-06-25
ATA119080A (de) 1981-09-15
DE3008257A1 (de) 1980-09-11
IT1130300B (it) 1986-06-11
BG33292A3 (en) 1983-01-14
CS215130B2 (en) 1982-07-30
IL59515A (en) 1983-02-23
RO80112A (ro) 1982-10-26
DK166353C (da) 1993-09-06
FR2450836A1 (fr) 1980-10-03
FI800661A (fi) 1980-09-06
PL222448A1 (es) 1981-01-02
NO823127L (no) 1980-09-08
NL8001285A (nl) 1980-09-09
FI70024C (fi) 1986-09-12
SU1192626A3 (ru) 1985-11-15
IT8020367A0 (it) 1980-03-05
PT70897A (en) 1980-04-01
DE3008257C2 (de) 1984-03-01
KE3464A (en) 1984-10-12
DK92680A (da) 1980-09-06
DK159852C (da) 1991-05-06
IN153685B (es) 1984-08-04
AT366693B (de) 1982-04-26
GB2045755B (en) 1983-01-26
DD149367A5 (de) 1981-07-08
NL180317B (nl) 1986-09-01
SE8603309D0 (sv) 1986-08-04
SE449103B (sv) 1987-04-06
SG55884G (en) 1985-03-08
ES8103094A1 (es) 1981-02-16
SE8603309L (sv) 1986-08-04
SE8000512L (sv) 1980-09-06
YU58580A (en) 1983-02-28
HU186304B (en) 1985-07-29
YU42328B (en) 1988-08-31
MX6032E (es) 1984-10-04
PL125197B1 (en) 1983-04-30
UA6342A1 (uk) 1994-12-29
DK145690A (da) 1990-06-14
LU82215A1 (fr) 1980-09-24
FR2450836B1 (fr) 1986-03-21
FI70024B (fi) 1986-01-31
NL180317C (nl) 1987-02-02
MY8500319A (en) 1985-12-31
IL59515A0 (en) 1980-06-30
IE49535B1 (en) 1985-10-16
AU5610480A (en) 1980-09-11
EG14437A (en) 1984-09-30
CH644608A5 (de) 1984-08-15
DK145690D0 (da) 1990-06-14
IE800429L (en) 1980-09-05

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