KR850001339B1 - 페니실란산 1,1-디옥사이드 및 그의 에스테르의 제조방법 - Google Patents
페니실란산 1,1-디옥사이드 및 그의 에스테르의 제조방법 Download PDFInfo
- Publication number
- KR850001339B1 KR850001339B1 KR1019800000885A KR800000885A KR850001339B1 KR 850001339 B1 KR850001339 B1 KR 850001339B1 KR 1019800000885 A KR1019800000885 A KR 1019800000885A KR 800000885 A KR800000885 A KR 800000885A KR 850001339 B1 KR850001339 B1 KR 850001339B1
- Authority
- KR
- South Korea
- Prior art keywords
- acid
- dioxide
- solution
- added
- ethyl acetate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Cosmetics (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1781079A | 1979-03-05 | 1979-03-05 | |
| US1780879A | 1979-03-05 | 1979-03-05 | |
| US17810 | 1979-03-05 | ||
| US17808 | 1979-03-05 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR850001339B1 true KR850001339B1 (ko) | 1985-09-19 |
Family
ID=26690337
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019800000885A Expired KR850001339B1 (ko) | 1979-03-05 | 1980-03-04 | 페니실란산 1,1-디옥사이드 및 그의 에스테르의 제조방법 |
Country Status (36)
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4419284A (en) * | 1981-03-23 | 1983-12-06 | Pfizer Inc. | Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide |
| IN159362B (enExample) * | 1981-03-23 | 1987-05-09 | Pfizer | |
| US4360463A (en) | 1981-09-02 | 1982-11-23 | Pfizer Inc. | Pure 6,6-diiodopenicillanic acid and process for its preparation |
| PT76526B (en) * | 1982-04-19 | 1986-01-21 | Gist Brocades Nv | Preparation of 6-alpha-bromo- and/or 6,6-dibromopenicillanic acid 1,1-dioxides |
| IT1190897B (it) * | 1982-06-29 | 1988-02-24 | Opos Biochimica Srl | Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico |
| US4606865A (en) * | 1982-09-20 | 1986-08-19 | Astra Lakemedel Aktiebolag | Methods for the preparation of α-bromodiethylcarbonate |
| EP0139047A1 (en) * | 1983-10-18 | 1985-05-02 | Gist-Brocades N.V. | Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide |
| EP0139048A1 (en) * | 1983-10-18 | 1985-05-02 | Gist-Brocades N.V. | Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide |
| US4596677A (en) * | 1984-04-06 | 1986-06-24 | Bristol-Myers Company | Anhydropenicillin intermediates |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IN149747B (enExample) * | 1977-06-07 | 1982-04-03 | Pfizer | |
| CA1158639A (en) * | 1978-12-11 | 1983-12-13 | Eric M. Gordon | 6-bromopenicillanic acid sulfone |
| DE3068390D1 (en) * | 1979-01-10 | 1984-08-09 | Beecham Group Plc | Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds |
| IE49881B1 (en) * | 1979-02-13 | 1986-01-08 | Leo Pharm Prod Ltd | B-lactam intermediates |
-
1980
- 1980-01-22 SE SE8000512A patent/SE449103B/sv not_active IP Right Cessation
- 1980-02-11 IN IN98/DEL/80A patent/IN153685B/en unknown
- 1980-02-27 UA UA2889601A patent/UA6342A1/uk unknown
- 1980-02-27 SU SU802889601A patent/SU1192626A3/ru active
- 1980-02-29 HU HU80479A patent/HU186304B/hu unknown
- 1980-03-03 YU YU585/80A patent/YU42328B/xx unknown
- 1980-03-03 GB GB8007122A patent/GB2045755B/en not_active Expired
- 1980-03-03 IL IL59515A patent/IL59515A/xx unknown
- 1980-03-03 LU LU82215A patent/LU82215A1/fr unknown
- 1980-03-03 AR AR280148A patent/AR225031A1/es active
- 1980-03-04 IE IE429/80A patent/IE49535B1/en not_active IP Right Cessation
- 1980-03-04 DE DE3008257A patent/DE3008257C2/de not_active Expired
- 1980-03-04 NL NLAANVRAGE8001285,A patent/NL180317C/xx not_active IP Right Cessation
- 1980-03-04 DK DK092680A patent/DK159852C/da not_active IP Right Cessation
- 1980-03-04 FI FI800661A patent/FI70024C/fi not_active IP Right Cessation
- 1980-03-04 PT PT70897A patent/PT70897A/pt unknown
- 1980-03-04 AU AU56104/80A patent/AU522572B2/en not_active Expired
- 1980-03-04 ES ES489185A patent/ES489185A0/es active Granted
- 1980-03-04 KR KR1019800000885A patent/KR850001339B1/ko not_active Expired
- 1980-03-04 GR GR61347A patent/GR67234B/el unknown
- 1980-03-04 CS CS801496A patent/CS215130B2/cs unknown
- 1980-03-04 PL PL1980222448A patent/PL125197B1/pl unknown
- 1980-03-04 AT AT0119080A patent/AT366693B/de not_active IP Right Cessation
- 1980-03-04 NO NO800618A patent/NO800618L/no unknown
- 1980-03-04 DD DD80219432A patent/DD149367A5/de unknown
- 1980-03-04 EG EG123/80A patent/EG14437A/xx active
- 1980-03-04 FR FR8004764A patent/FR2450836B1/fr not_active Expired
- 1980-03-04 CH CH171080A patent/CH644608A5/de not_active IP Right Cessation
- 1980-03-04 RO RO80100366A patent/RO80112A/ro unknown
- 1980-03-05 MX MX808687U patent/MX6032E/es unknown
- 1980-03-05 IT IT20367/80A patent/IT1130300B/it active
- 1980-03-05 BG BG046874A patent/BG33292A3/xx unknown
-
1982
- 1982-09-15 NO NO823127A patent/NO823127L/no unknown
-
1984
- 1984-08-13 SG SG558/84A patent/SG55884G/en unknown
- 1984-09-24 KE KE3464A patent/KE3464A/xx unknown
-
1985
- 1985-12-30 MY MY319/85A patent/MY8500319A/xx unknown
-
1986
- 1986-08-04 SE SE8603309A patent/SE8603309D0/xx not_active Application Discontinuation
-
1987
- 1987-09-17 HK HK665/87A patent/HK66587A/xx not_active IP Right Cessation
-
1990
- 1990-06-14 DK DK145690A patent/DK166353C/da not_active IP Right Cessation
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| KR840000797B1 (ko) | 6β-하이드록시알킬페니실란산 유도체의 제조방법 | |
| US4234579A (en) | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors | |
| US4276285A (en) | Combinations of penicillanic acid 1,1-dioxide with 7-(D-2-[4-ethylpiperazin-2,3-dione-1-carboxamido]-2-[4-hydroxyphenyl]acetamido)-3-([1-methyl-5-tetrazolyl]thiomethyl)-3-desacetoxymethylcephalosporanic acid | |
| KR850001339B1 (ko) | 페니실란산 1,1-디옥사이드 및 그의 에스테르의 제조방법 | |
| US4256733A (en) | Acetoxymethyl penam compounds as β-lactamase inhibitors | |
| US4420426A (en) | 6-Alpha-halopenicillanic acid 1,1-dioxides | |
| CA1109859A (en) | Thiooxime cephalosporin and penicillin derivatives | |
| KR840000589B1 (ko) | 6-β-치환된 페니실란산의 제조방법 | |
| US4260598A (en) | Method for increasing antibacterial effectiveness of a β-lactam antibiotic | |
| EP0181702B1 (en) | 6-substituted penicillanic acid 1,1-dioxide compounds | |
| JPS6033397B2 (ja) | ペナム−１，１−ジオキシド | |
| US4452796A (en) | 6-Aminoalkylpenicillanic acid 1,1-dioxides as beta-lactamase inhibitors | |
| EP0287734A1 (en) | 2-Beta-substituted methyl-penam derivatives | |
| US4714761A (en) | 6,6-dihalopenicillanic acid 1,1-dioxides and process | |
| US4762920A (en) | 6,6-Dihalopenicillanic acid 1,1-dioxides | |
| US4656263A (en) | 6-β-substituted penicillanic acid compound free of the 6-α-epimer | |
| JPS6145993B2 (enExample) | ||
| EP0002927B1 (en) | Penicillanic acid derivatives, processes for their preparation and pharmaceutical compositions containing them | |
| US4613462A (en) | 6-substituted penicillanic acid 1,1-dioxide compounds | |
| US4518530A (en) | 6-β-Substituted penicillanic acids as β-lactamase inhibitors | |
| US4517126A (en) | Penicillanic acid derivative | |
| KR810002025B1 (ko) | 페니실란산 1, 1-디옥사이드의 제조방법 | |
| KR820000740B1 (ko) | 페니실란산 1, 1-디옥사이드의 제조방법 | |
| CA1152982A (en) | Process and intermediates for penicillanic acid, 1,1-dioxide and esters thereof | |
| KR830001902B1 (ko) | 폐니실란산유도체의 제조방법 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0109 | Patent application |
St.27 status event code: A-0-1-A10-A12-nap-PA0109 |
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| P11-X000 | Amendment of application requested |
St.27 status event code: A-2-2-P10-P11-nap-X000 |
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| P13-X000 | Application amended |
St.27 status event code: A-2-2-P10-P13-nap-X000 |
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| PG1501 | Laying open of application |
St.27 status event code: A-1-1-Q10-Q12-nap-PG1501 |
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| PE0902 | Notice of grounds for rejection |
St.27 status event code: A-1-2-D10-D21-exm-PE0902 |
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| T11-X000 | Administrative time limit extension requested |
St.27 status event code: U-3-3-T10-T11-oth-X000 |
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| P11-X000 | Amendment of application requested |
St.27 status event code: A-2-2-P10-P11-nap-X000 |
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| P13-X000 | Application amended |
St.27 status event code: A-2-2-P10-P13-nap-X000 |
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| PE0601 | Decision on rejection of patent |
St.27 status event code: N-2-6-B10-B15-exm-PE0601 |
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| PG1605 | Publication of application before grant of patent |
St.27 status event code: A-2-2-Q10-Q13-nap-PG1605 |
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St.27 status event code: A-1-2-D10-D22-exm-PE0701 |
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