KR830006277A - 티오포름아미이드 유도체의 제조방법 - Google Patents

티오포름아미이드 유도체의 제조방법 Download PDF

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KR830006277A
KR830006277A KR1019810001943A KR810001943A KR830006277A KR 830006277 A KR830006277 A KR 830006277A KR 1019810001943 A KR1019810001943 A KR 1019810001943A KR 810001943 A KR810001943 A KR 810001943A KR 830006277 A KR830006277 A KR 830006277A
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South Korea
Prior art keywords
radical
pyrid
sulfur
iii
following formula
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KR1019810001943A
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KR850001043B1 (ko
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아루프 쟈안-크로오드
부우쇼오돈 쟈안
화하제 다니엘
제임스 크로오드
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쟈안허어슨
로오느-푸우랜크 인더스트리이즈
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/12—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
    • C07D213/32—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/08—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Abstract

내용 없음

Description

티오포름 아미이드 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (1)

  1. 암모니아 또는 하기 구조식 Ⅱ의 암모니아를 하기구조식 Ⅲ의 디티오에스테르와 반응시킨다음 얻어진 생성물을 분리시켜 하기 구조식 Ⅰ의 티 어포름아미이드 유도체를 제조하는 방법.
    상기 구조식 들중에서, R은 수소원자 되는 탄소수 1-4를 갖는 직쇄 또는 촉쇄 알킬 라디칼이며,
    (ⅰ) Het가, 피리드-3-일, 피리드-4-일, 피리다지닐, 피라지닐, 피리미디닐, 퀴놀일, 이미다졸일, 나프티리디닐, 퀴녹사리닐과 퀴나졸리닐로부터 선정되고 하나 또는 두개의 질소원자를 갖는 방향족형질의 복소환식 라디칼을 나타내며, X는 황 또는 산소원자를 나타내며 Y는 황 또는 산소원자, 원자가 결합 또는 메틸렌 라디칼을 나타내거나
    (ⅱ) Het가 피리드-2-일 라디칼을 나타내고, X는 황 또는 산소원자를 나타내며 Y는 황 또는 산소원자 또는 메틸렌 라디칼을 나타내거나, 또는
    (ⅲ) Het가 피리드-2-일 라디칼을 나타내고, X는 산소원자를 나타내며 Y는 원자가 결합을 나타내며,
    R'는 탄소수 1-4를 갖는 직쇄 또는 측쇄 알킬 라디칼 또는 벤질 또는 카르복시에틸 라디칼이다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019810001943A 1980-08-18 1981-05-30 티오포름 아마이드 유도체의 제조방법 KR850001043B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR18,035 1980-08-18
FR8018035A FR2488609A1 (fr) 1980-08-18 1980-08-18 Nouveaux derives de la thioformamide, leur preparation et les medicaments qui les contiennent

Publications (2)

Publication Number Publication Date
KR830006277A true KR830006277A (ko) 1983-09-20
KR850001043B1 KR850001043B1 (ko) 1985-07-19

Family

ID=9245232

Family Applications (1)

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KR1019810001943A KR850001043B1 (ko) 1980-08-18 1981-05-30 티오포름 아마이드 유도체의 제조방법

Country Status (24)

Country Link
US (1) US4379154A (ko)
EP (2) EP0077083B1 (ko)
JP (1) JPS5742687A (ko)
KR (1) KR850001043B1 (ko)
AT (1) ATE14730T1 (ko)
CA (1) CA1161039A (ko)
DE (1) DE3161861D1 (ko)
DK (1) DK158735C (ko)
ES (2) ES501060A0 (ko)
FI (1) FI810835L (ko)
FR (1) FR2488609A1 (ko)
GR (1) GR72767B (ko)
HU (1) HU187325B (ko)
IE (1) IE51263B1 (ko)
IL (1) IL62380A (ko)
MA (1) MA19106A1 (ko)
NO (1) NO810962L (ko)
NZ (1) NZ197071A (ko)
OA (1) OA06767A (ko)
PH (1) PH16520A (ko)
PL (2) PL130679B1 (ko)
PT (1) PT72718B (ko)
SU (2) SU1093248A3 (ko)
ZA (1) ZA813159B (ko)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2511371A1 (fr) * 1981-08-11 1983-02-18 Rhone Poulenc Sante Nouveaux nitriles heterocycliques, leur preparation et leur utilisation pour la preparation de medicaments
FR2528849B1 (fr) * 1982-06-17 1985-06-21 Rhone Poulenc Sante Nouveaux derives de la thioformamide, leur preparation et les medicaments qui les contiennent
FR2573428B1 (fr) * 1984-11-20 1987-01-30 Rhone Poulenc Sante Nouveaux derives de la thioformamide, leur preparation et les medicaments qui les contiennent
GB8907306D0 (en) * 1989-03-31 1989-05-17 May & Baker Ltd New compositions of matter
FR2653770B1 (fr) * 1989-10-31 1992-01-03 Rhone Poulenc Sante Procede de preparation de (pyridyl-3)-2 tetrahydrothiopyrannecarbothioamide-2-oxydes-1-(1r,2r), les (pyridyl-3)-2 tetrhydrothiopyrannecarbothioamide-2-oxydes-1-(1r,2r) ainsi obtenus et les compositions pharmaceutiques qui les contiennent.
JPH04211048A (ja) * 1990-03-05 1992-08-03 Mitsubishi Kasei Corp チオカルバモイルアセトニトリル誘導体
CA2119876A1 (en) * 1991-10-14 1993-04-29 Yasuhiro Kabasawa Thioformamide derivative
US5625068A (en) * 1995-06-05 1997-04-29 American Cyanamid Company Substituted quinoline herbicide intermediates and process

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1056205B (it) * 1970-07-30 1982-01-30 Fujisawa Pharmaceutical Co Composto a paste di derivati tioa cetammidici e loro sali procedimento per il suo ottenimento e composizioni che lo contengono
DK627174A (ko) * 1974-01-17 1975-09-08 Ciba Geigy Ag
FR2452488A1 (fr) * 1979-03-30 1980-10-24 Rhone Poulenc Ind Nouveaux derives du (pyridyl-2)-2 tetrahydrothiophene, leur preparation et les medicaments qui les contiennent
IE49570B1 (en) * 1979-03-30 1985-10-30 Rhone Poulenc Ind 2-(pyrid-2-yl)tetrahydrothiophene derivatives
JPS6134433A (ja) * 1984-08-31 1986-02-18 Nippon Telegr & Teleph Corp <Ntt> ｘｙ平面位置決め用アクチユエ−タ装置

Also Published As

Publication number Publication date
FR2488609A1 (fr) 1982-02-19
PL230552A1 (ko) 1982-03-01
PT72718A (fr) 1981-04-01
US4379154A (en) 1983-04-05
ES503727A0 (es) 1982-12-01
MA19106A1 (fr) 1981-10-01
PT72718B (fr) 1982-03-24
DK158735B (da) 1990-07-09
EP0046417A1 (fr) 1982-02-24
HU187325B (en) 1985-12-28
GR72767B (ko) 1983-12-02
SU1209029A3 (ru) 1986-01-30
FR2488609B1 (ko) 1984-05-04
DK130781A (da) 1982-02-19
NO810962L (no) 1982-02-19
PL130679B1 (en) 1984-08-31
JPS5742687A (en) 1982-03-10
IE51263B1 (en) 1986-11-26
IE811036L (en) 1982-02-18
EP0046417B1 (fr) 1984-01-11
SU1093248A3 (ru) 1984-05-15
DE3161861D1 (en) 1984-02-16
ZA813159B (en) 1983-07-27
ES8301475A1 (es) 1982-12-01
ATE14730T1 (de) 1985-08-15
ES8202819A1 (es) 1982-02-01
OA06767A (fr) 1982-12-31
FI810835L (fi) 1982-02-19
JPH0259150B2 (ko) 1990-12-11
CA1161039A (fr) 1984-01-24
KR850001043B1 (ko) 1985-07-19
EP0077083B1 (fr) 1985-08-07
EP0077083A1 (fr) 1983-04-20
DK158735C (da) 1990-12-03
IL62380A (en) 1984-11-30
ES501060A0 (es) 1982-02-01
PH16520A (en) 1983-11-10
NZ197071A (en) 1983-07-15
PL130530B1 (en) 1984-08-31
IL62380A0 (en) 1981-05-20

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