KR830001906B1 - β-락탐 화합물의 할로겐화 반응물 제조방법 - Google Patents

β-락탐 화합물의 할로겐화 반응물 제조방법 Download PDF

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Publication number
KR830001906B1
KR830001906B1 KR1019800000400A KR800000400A KR830001906B1 KR 830001906 B1 KR830001906 B1 KR 830001906B1 KR 1019800000400 A KR1019800000400 A KR 1019800000400A KR 800000400 A KR800000400 A KR 800000400A KR 830001906 B1 KR830001906 B1 KR 830001906B1
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KR
South Korea
Prior art keywords
carboxylate
hydroxy
phosphite
amino
cepem
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019800000400A
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English (en)
Korean (ko)
Other versions
KR830001955A (ko
Inventor
델로스. 하트필드 로우웰.
크리스 브라스즈크작 라리
웨인퓌셔 잭.
Original Assignee
일라이 릴리 앤드 캄파니
아서 알. 훼일
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21732838&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR830001906(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 일라이 릴리 앤드 캄파니, 아서 알. 훼일 filed Critical 일라이 릴리 앤드 캄파니
Publication of KR830001955A publication Critical patent/KR830001955A/ko
Application granted granted Critical
Publication of KR830001906B1 publication Critical patent/KR830001906B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
    • H—ELECTRICITY
    • H01—ELECTRIC ELEMENTS
    • H01L—SEMICONDUCTOR DEVICES NOT COVERED BY CLASS H10
    • H01L2224/00—Indexing scheme for arrangements for connecting or disconnecting semiconductor or solid-state bodies and methods related thereto as covered by H01L24/00
    • H01L2224/74—Apparatus for manufacturing arrangements for connecting or disconnecting semiconductor or solid-state bodies and for methods related thereto
    • H01L2224/78—Apparatus for connecting with wire connectors
    • H—ELECTRICITY
    • H01—ELECTRIC ELEMENTS
    • H01L—SEMICONDUCTOR DEVICES NOT COVERED BY CLASS H10
    • H01L2924/00—Indexing scheme for arrangements or methods for connecting or disconnecting semiconductor or solid-state bodies as covered by H01L24/00
    • H01L2924/0001—Technical content checked by a classifier
    • H01L2924/00014—Technical content checked by a classifier the subject-matter covered by the group, the symbol of which is combined with the symbol of this group, being disclosed without further technical details
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
KR1019800000400A 1979-02-01 1980-02-01 β-락탐 화합물의 할로겐화 반응물 제조방법 Expired KR830001906B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8647 1979-02-01
US06/008,647 US4226986A (en) 1979-02-01 1979-02-01 Process for halogenation of β-lactam compounds
US008647 1979-02-01

Publications (2)

Publication Number Publication Date
KR830001955A KR830001955A (ko) 1983-05-21
KR830001906B1 true KR830001906B1 (ko) 1983-09-19

Family

ID=21732838

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1019800000400A Expired KR830001906B1 (ko) 1979-02-01 1980-02-01 β-락탐 화합물의 할로겐화 반응물 제조방법
KR1019800000398A Expired KR830001892B1 (ko) 1979-02-01 1980-02-01 베타 락탐 화합물의 할로겐화 제조 방법

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1019800000398A Expired KR830001892B1 (ko) 1979-02-01 1980-02-01 베타 락탐 화합물의 할로겐화 제조 방법

Country Status (22)

Country Link
US (1) US4226986A (enExample)
EP (1) EP0014566B1 (enExample)
JP (1) JPS55104289A (enExample)
KR (2) KR830001906B1 (enExample)
BE (1) BE881426A (enExample)
BG (1) BG35896A3 (enExample)
CA (1) CA1150725A (enExample)
CH (1) CH642971A5 (enExample)
CS (1) CS275604B6 (enExample)
DE (1) DE3063395D1 (enExample)
ES (2) ES488234A0 (enExample)
FR (1) FR2447926A1 (enExample)
GB (1) GB2041374B (enExample)
HU (1) HU182065B (enExample)
IE (1) IE49503B1 (enExample)
IL (1) IL59266A (enExample)
IT (1) IT1130240B (enExample)
LU (1) LU82121A1 (enExample)
MX (1) MX6576E (enExample)
PH (2) PH14774A (enExample)
RO (1) RO84256B (enExample)
ZM (1) ZM1280A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1148938A (en) * 1979-05-08 1983-06-28 John R. Corfield Preparation of cephalosporins and intermediates employed therein
US4281117A (en) * 1980-09-04 1981-07-28 Eli Lilly And Company Process for 3-chloro cephalosporin nucleus
IN181695B (enExample) * 1992-08-10 1998-09-05 Ranbaxy Lab Ltd
US5604222A (en) * 1993-12-27 1997-02-18 Lupin Laboratories, Ltd. Method for the preparation of 2-chloro sulfinyl azetidinones
US5578721A (en) * 1994-07-11 1996-11-26 Lupin Laboratories Limited Process for preparation of 3-exomethylene cepham sulfoxide esters
JP6669831B2 (ja) * 2018-10-02 2020-03-18 株式会社ユニバーサルエンターテインメント 遊技機

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3925372A (en) * 1973-02-23 1975-12-09 Lilly Co Eli Alpha-aminoacyl-3-halo cephalosporins
US3962227A (en) * 1973-02-23 1976-06-08 Eli Lilly And Company 3-halo cephalosporins
GB1472869A (en) * 1975-08-11 1977-05-11 Farmaceutici Italia Intermediates for cephalosporin synthesis
IE45158B1 (en) * 1976-08-16 1982-06-30 Lilly Co Eli 3-chloro-cephem synthesis
GB1576219A (en) * 1976-12-31 1980-10-01 Connlab Holdings Ltd Thiazoleneazetidinone derivatives

Also Published As

Publication number Publication date
FR2447926B1 (enExample) 1982-12-31
IL59266A0 (en) 1980-05-30
RO84256A (ro) 1984-05-23
KR830001892B1 (ko) 1983-09-17
EP0014566B1 (en) 1983-05-25
IL59266A (en) 1983-05-15
PH17758A (en) 1984-11-27
GB2041374B (en) 1983-04-13
CS275604B6 (en) 1992-03-18
ES8106530A1 (es) 1981-08-16
EP0014566A1 (en) 1980-08-20
IT8019610A0 (it) 1980-01-31
ES8104302A1 (es) 1981-04-16
PH14774A (en) 1981-12-09
KR830001955A (ko) 1983-05-21
JPH0115515B2 (enExample) 1989-03-17
IT1130240B (it) 1986-06-11
LU82121A1 (fr) 1980-04-23
FR2447926A1 (fr) 1980-08-29
CH642971A5 (fr) 1984-05-15
MX6576E (es) 1985-07-24
HU182065B (en) 1983-12-28
JPS55104289A (en) 1980-08-09
ES488234A0 (es) 1981-04-16
IE49503B1 (en) 1985-10-16
ZM1280A1 (en) 1980-09-22
US4226986A (en) 1980-10-07
CS8000660A2 (en) 1991-03-12
IE800187L (en) 1980-08-01
GB2041374A (en) 1980-09-10
DE3063395D1 (en) 1983-07-07
RO84256B (ro) 1984-07-30
KR830001957A (ko) 1983-05-19
CA1150725A (en) 1983-07-26
BG35896A3 (en) 1984-07-16
BE881426A (fr) 1980-07-30
ES495102A0 (es) 1981-08-16

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US4223133A (en) Cephalosporin reduction process
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Patent event code: PA01091R01D

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Patent event date: 19800201

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Patent event code: PG16051S01I

Patent event date: 19830819

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