KR830001202A - 2-클로로설피닐 아제티딘온의 제조방법 - Google Patents

2-클로로설피닐 아제티딘온의 제조방법 Download PDF

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Publication number
KR830001202A
KR830001202A KR1019790003525A KR790003525A KR830001202A KR 830001202 A KR830001202 A KR 830001202A KR 1019790003525 A KR1019790003525 A KR 1019790003525A KR 790003525 A KR790003525 A KR 790003525A KR 830001202 A KR830001202 A KR 830001202A
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KR
South Korea
Prior art keywords
chlorosulfinyl
structural formula
azetidine
producing
linked
Prior art date
Application number
KR1019790003525A
Other languages
English (en)
Other versions
KR830001346B1 (ko
Inventor
타센추
Original Assignee
아더 알. 웨일
일라이 릴리 앤드 캄파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 아더 알. 웨일, 일라이 릴리 앤드 캄파니 filed Critical 아더 알. 웨일
Publication of KR830001202A publication Critical patent/KR830001202A/ko
Application granted granted Critical
Publication of KR830001346B1 publication Critical patent/KR830001346B1/ko

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C07D205/095Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4 and with a nitrogen atom directly attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

내용 없음

Description

2-클로로설피닐 아제티딘온의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (1)

  1. 다음 구조식 1의 페니실린 설폭사이드 에스테르를 N-클로로 할로겐화제와 무수상태의 불활성 유기용매중에서 교차 결합된 폴리비닐피리딘 폴리머(폴리머는 약 1% 내지 10% 교차 결합되어 있음) 존재하에서 반응시킴을 특징으로 해서 다음 구조식 2의 2-클로로설피닐 아제티딘-4-온을 제조하는 방법.
    상기 구조식에서
    R은 카복실산의 잔기이며 R1은 카복실산보호기이다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019790003525A 1978-11-13 1979-10-13 2-클로로 설피닐 아제티딘온의 제조방법 KR830001346B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US96034778A 1978-11-13 1978-11-13
US960347 1978-11-13

Publications (2)

Publication Number Publication Date
KR830001202A true KR830001202A (ko) 1983-04-29
KR830001346B1 KR830001346B1 (ko) 1983-07-14

Family

ID=25503072

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019790003525A KR830001346B1 (ko) 1978-11-13 1979-10-13 2-클로로 설피닐 아제티딘온의 제조방법

Country Status (8)

Country Link
JP (1) JPS5566558A (ko)
KR (1) KR830001346B1 (ko)
BE (1) BE879211A (ko)
CS (1) CS209825B2 (ko)
MA (1) MA18604A1 (ko)
MW (1) MW3079A1 (ko)
ZA (1) ZA795243B (ko)
ZM (1) ZM8279A1 (ko)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1069126A (en) * 1974-12-24 1980-01-01 Eli Lilly And Company Sulfinyl halides and their preparation from penicillin sulfoxides

Also Published As

Publication number Publication date
JPS5566558A (en) 1980-05-20
CS209825B2 (en) 1981-12-31
ZM8279A1 (en) 1980-05-21
MA18604A1 (fr) 1980-07-01
KR830001346B1 (ko) 1983-07-14
ZA795243B (en) 1981-05-27
MW3079A1 (en) 1981-04-08
BE879211A (fr) 1980-04-08
JPS641469B2 (ko) 1989-01-11

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