KR20170021904A - 스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물 - Google Patents

스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물 Download PDF

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Publication number
KR20170021904A
KR20170021904A KR1020177004540A KR20177004540A KR20170021904A KR 20170021904 A KR20170021904 A KR 20170021904A KR 1020177004540 A KR1020177004540 A KR 1020177004540A KR 20177004540 A KR20177004540 A KR 20177004540A KR 20170021904 A KR20170021904 A KR 20170021904A
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South Korea
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alkyl
formula
group
substituted
compound
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Korean (ko)
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콜렌 뢰거
미하엘 앰부엘
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노파르티스 아게
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Application filed by 노파르티스 아게 filed Critical 노파르티스 아게
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/133—Amines having hydroxy groups, e.g. sphingosine
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
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    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
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    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Inorganic Chemistry (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Zoology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Medical Informatics (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Biotechnology (AREA)
  • Botany (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Hospice & Palliative Care (AREA)
  • Oncology (AREA)
KR1020177004540A 2007-10-12 2008-10-09 스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물 Withdrawn KR20170021904A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US97948207P 2007-10-12 2007-10-12
US60/979,482 2007-10-12
PCT/US2008/079264 WO2009048993A2 (en) 2007-10-12 2008-10-09 Compositions comprising sphingosine 1 phosphate (s1p) receptor modulators

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020167004264A Division KR101710845B1 (ko) 2007-10-12 2008-10-09 스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물

Publications (1)

Publication Number Publication Date
KR20170021904A true KR20170021904A (ko) 2017-02-28

Family

ID=40032615

Family Applications (3)

Application Number Title Priority Date Filing Date
KR1020177004540A Withdrawn KR20170021904A (ko) 2007-10-12 2008-10-09 스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물
KR1020167004264A Active KR101710845B1 (ko) 2007-10-12 2008-10-09 스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물
KR1020107010336A Active KR101600098B1 (ko) 2007-10-12 2008-10-09 스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물

Family Applications After (2)

Application Number Title Priority Date Filing Date
KR1020167004264A Active KR101710845B1 (ko) 2007-10-12 2008-10-09 스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물
KR1020107010336A Active KR101600098B1 (ko) 2007-10-12 2008-10-09 스핑고신 1 포스페이트 (ｓ1ｐ) 수용체 조절제를 포함하는 조성물

Country Status (32)

Country Link
US (6) US8673918B2 (https=)
EP (7) EP3733161A1 (https=)
JP (2) JP6034000B2 (https=)
KR (3) KR20170021904A (https=)
CN (1) CN101820916A (https=)
AR (1) AR068986A1 (https=)
AU (1) AU2008310846C1 (https=)
BR (1) BRPI0818161B8 (https=)
CA (2) CA2699788C (https=)
CL (1) CL2008003003A1 (https=)
CO (1) CO6270342A2 (https=)
DK (1) DK2952177T3 (https=)
EC (1) ECSP10010169A (https=)
ES (2) ES2545361T3 (https=)
HR (1) HRP20150838T1 (https=)
HU (2) HUE027696T2 (https=)
IL (3) IL204514B (https=)
JO (2) JOP20080436B1 (https=)
MA (1) MA31799B1 (https=)
MX (1) MX337152B (https=)
MY (1) MY159358A (https=)
NZ (1) NZ600355A (https=)
PE (2) PE20130309A1 (https=)
PL (2) PL2465492T3 (https=)
PT (2) PT2465492E (https=)
RU (1) RU2010118457A (https=)
SG (2) SG187458A1 (https=)
SI (2) SI2952177T1 (https=)
TN (1) TN2010000136A1 (https=)
TW (1) TW200927142A (https=)
WO (1) WO2009048993A2 (https=)
ZA (1) ZA201001819B (https=)

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