KR20160145833A - 티에노트리아졸로디아제핀 화합물을 사용한 급성 골수성 백혈병 및/또는 급성 림프아구성 백혈병의 치료 방법 - Google Patents

티에노트리아졸로디아제핀 화합물을 사용한 급성 골수성 백혈병 및/또는 급성 림프아구성 백혈병의 치료 방법 Download PDF

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KR20160145833A
KR20160145833A KR1020167033946A KR20167033946A KR20160145833A KR 20160145833 A KR20160145833 A KR 20160145833A KR 1020167033946 A KR1020167033946 A KR 1020167033946A KR 20167033946 A KR20167033946 A KR 20167033946A KR 20160145833 A KR20160145833 A KR 20160145833A
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compound
leukemia
formula
solid dispersion
acute
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케이 노엘
마리아 이 리베이로
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온코에틱스 게엠베하
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
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    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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KR1020167033946A 2014-05-02 2015-05-01 티에노트리아졸로디아제핀 화합물을 사용한 급성 골수성 백혈병 및/또는 급성 림프아구성 백혈병의 치료 방법 Withdrawn KR20160145833A (ko)

Applications Claiming Priority (15)

Application Number Priority Date Filing Date Title
US201461987822P 2014-05-02 2014-05-02
US61/987,822 2014-05-02
US201461990465P 2014-05-08 2014-05-08
US61/990,465 2014-05-08
US201462012128P 2014-06-13 2014-06-13
US201462012135P 2014-06-13 2014-06-13
US62/012,135 2014-06-13
US62/012,128 2014-06-13
US201462080804P 2014-11-17 2014-11-17
US201462080771P 2014-11-17 2014-11-17
US62/080,771 2014-11-17
US62/080,804 2014-11-17
US201462086456P 2014-12-02 2014-12-02
US62/086,456 2014-12-02
PCT/US2015/028891 WO2015168621A1 (en) 2014-05-02 2015-05-01 Method of treating acute myeloid leukemia and/or acute lymphoblastic leukemia using thienotriazolodiazepine compounds

Publications (1)

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KR20160145833A true KR20160145833A (ko) 2016-12-20

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KR1020167033946A Withdrawn KR20160145833A (ko) 2014-05-02 2015-05-01 티에노트리아졸로디아제핀 화합물을 사용한 급성 골수성 백혈병 및/또는 급성 림프아구성 백혈병의 치료 방법

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Country Link
US (1) US9956228B2 (enExample)
EP (1) EP3137085A4 (enExample)
JP (1) JP2017514909A (enExample)
KR (1) KR20160145833A (enExample)
CN (1) CN107073014A (enExample)
AU (1) AU2015252844A1 (enExample)
CA (1) CA2947601A1 (enExample)
MX (1) MX2016014301A (enExample)
RU (1) RU2016146099A (enExample)
WO (1) WO2015168621A1 (enExample)

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WO2018200041A1 (en) 2017-04-26 2018-11-01 University Of Cincinnati Methods, agents, and compositions for the treatment of acute myeloid leukemia
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KR20160036591A (ko) * 2013-08-01 2016-04-04 온코에틱스 게엠베하 티에노트리아졸로디아제핀 화합물을 함유하는 약학적 제제
EP3074018A1 (en) * 2013-11-27 2016-10-05 Oncoethix GmbH Method of treating leukemia using pharmaceutical formulation containing thienotriazolodiazepine compounds
WO2016030509A1 (en) * 2014-08-28 2016-03-03 Oncoethix Gmbh Methods of treating acute myeloid leukemia or acute lymphoid leukemia using pharmaceutical compositions containing thienotriazolodiazepine compounds

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US20170049784A1 (en) 2017-02-23
RU2016146099A3 (enExample) 2018-12-25
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US9956228B2 (en) 2018-05-01
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