KR20150064232A - 치료제의 경구 투여를 위한 제제 및 관련 방법 - Google Patents
치료제의 경구 투여를 위한 제제 및 관련 방법 Download PDFInfo
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- KR20150064232A KR20150064232A KR1020157013456A KR20157013456A KR20150064232A KR 20150064232 A KR20150064232 A KR 20150064232A KR 1020157013456 A KR1020157013456 A KR 1020157013456A KR 20157013456 A KR20157013456 A KR 20157013456A KR 20150064232 A KR20150064232 A KR 20150064232A
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- South Korea
- Prior art keywords
- fatty acid
- ampb
- formulation
- amphotericin
- polyethylene oxide
- Prior art date
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- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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Applications Claiming Priority (7)
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| US94030707P | 2007-05-25 | 2007-05-25 | |
| US60/940,307 | 2007-05-25 | ||
| US97670807P | 2007-10-01 | 2007-10-01 | |
| US60/976,708 | 2007-10-01 | ||
| US4147808P | 2008-04-01 | 2008-04-01 | |
| US61/041,478 | 2008-04-01 | ||
| PCT/CA2008/000975 WO2008144888A1 (en) | 2007-05-25 | 2008-05-23 | Formulations for the oral administration of therapeutic agents and related methods |
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| KR1020167005288A Ceased KR20160029866A (ko) | 2007-05-25 | 2008-05-23 | 치료제의 경구 투여를 위한 제제 및 관련 방법 |
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| KR1020097027108A Ceased KR20100017928A (ko) | 2007-05-25 | 2008-05-23 | 치료제의 경구 투여를 위한 제제 및 관련 방법 |
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| JP (1) | JP5501224B2 (https=) |
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| CN (1) | CN101687044B (https=) |
| CA (1) | CA2688036C (https=) |
| IL (1) | IL202111A (https=) |
| MX (1) | MX2009012782A (https=) |
| NZ (1) | NZ582332A (https=) |
| RU (1) | RU2485975C2 (https=) |
| WO (1) | WO2008144888A1 (https=) |
| ZA (1) | ZA200908928B (https=) |
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| NO2252275T3 (https=) * | 2008-02-13 | 2018-04-28 | ||
| CN102389401B (zh) * | 2011-11-22 | 2013-05-22 | 陆荣政 | 一种右旋布洛芬颗粒及其制备方法 |
| WO2014152207A1 (en) | 2013-03-15 | 2014-09-25 | Mylan Laboratories, Inc. | Hot melt granulation formulations of poorly water-soluble active agents |
| US20170217976A1 (en) * | 2014-03-21 | 2017-08-03 | Chironwells Gmbh | 6-(amino acid)-morphinan derivatives in combination with permeation enhancers for use as an orally, rectally, transdermally or nasally administered medicament |
| KR101542364B1 (ko) * | 2014-10-31 | 2015-08-07 | 대화제약 주식회사 | 탁산을 포함하는 경구 투여용 약학 조성물 |
| WO2016112339A1 (en) * | 2015-01-09 | 2016-07-14 | Ico Therapeutics Inc. | Stable formulations for the oral administration of amphotericin b and related methods |
| CN105018542B (zh) * | 2015-07-10 | 2018-01-02 | 北京师范大学 | 烟曲霉teqa在制备奥沙西泮中的应用 |
| CN106063779A (zh) * | 2016-06-12 | 2016-11-02 | 上海上药第生化药业有限公司 | 一种维生素k1药物的新剂型及制备方法 |
| EP3585397A4 (en) * | 2017-02-21 | 2020-11-25 | iCo Therapeutics Inc. | ORAL AMPHOTERICIN B SOLID FORMULATIONS |
| US20230310465A1 (en) * | 2020-08-18 | 2023-10-05 | Leiutis Pharmaceuticals Llp | Nano lipid carrier system for improving permeation of active ingredients |
| BR102020022824A8 (pt) * | 2020-11-09 | 2024-01-02 | Fundacao Oswaldo Cruz | Composição, composição farmacêutica, e, uso de uma composição tópica estável compreendendo uma nanoemulsão, e de pelo menos um composto antileishmanial |
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| AU598958B2 (en) * | 1987-11-12 | 1990-07-05 | Vestar, Inc. | Improved amphotericin b liposome preparation |
| WO1993011777A1 (en) * | 1991-12-11 | 1993-06-24 | Temple University - Of The Commonwealth System Of Higher Education | Amphotericin b composition with enhanced antifungal activity |
| FR2710535B1 (fr) * | 1993-09-30 | 1995-11-24 | Gattefosse Ets Sa | Composition à usage pharmaceutique ou cosmétique apte à former une microémulsion. |
| US6217886B1 (en) * | 1997-07-14 | 2001-04-17 | The Board Of Trustees Of The University Of Illinois | Materials and methods for making improved micelle compositions |
| US6248363B1 (en) * | 1999-11-23 | 2001-06-19 | Lipocine, Inc. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
| US6294192B1 (en) * | 1999-02-26 | 2001-09-25 | Lipocine, Inc. | Triglyceride-free compositions and methods for improved delivery of hydrophobic therapeutic agents |
| US6852334B1 (en) * | 1999-04-20 | 2005-02-08 | The University Of British Columbia | Cationic peg-lipids and methods of use |
| US20030236236A1 (en) | 1999-06-30 | 2003-12-25 | Feng-Jing Chen | Pharmaceutical compositions and dosage forms for administration of hydrophobic drugs |
| US6596306B1 (en) * | 2000-07-07 | 2003-07-22 | David Ho Sue San Ho | Drug delivery system:formulation for fat-soluble drugs |
| IN188843B (https=) * | 2000-06-22 | 2002-11-09 | Vinod Daftary Gautam Dr | |
| DE10036871A1 (de) * | 2000-07-28 | 2002-02-14 | Pharmasol Gmbh | Dispersionen zur Formulierung wenig oder schwer löslicher Wirkstoffe |
| AU2002214854A1 (en) * | 2000-10-25 | 2002-05-06 | Inex Pharmaceuticals Corporation | Lipid formulations for target delivery |
| US8067032B2 (en) * | 2000-12-22 | 2011-11-29 | Baxter International Inc. | Method for preparing submicron particles of antineoplastic agents |
| FR2827770B1 (fr) * | 2001-07-27 | 2005-08-19 | Gattefosse Ets Sa | Composition pharmaceutique a usage oral comprenant un principe actif susceptible de subir un important effet de premier passage intestinal |
| US6660761B2 (en) * | 2002-02-06 | 2003-12-09 | Council Of Scientific And Industrial Research | Method of treatment for fungal infections with a synergistic formulation of antifungal agents |
| JP2003252750A (ja) | 2002-02-26 | 2003-09-10 | ▲寛▼治 ▲高▼田 | 水溶性の難・低吸収性薬物のバイオアベイラビリティ改善技術 |
| CN1290893C (zh) * | 2002-05-03 | 2006-12-20 | 詹森药业有限公司 | 聚合物微乳状液 |
| US20040116360A1 (en) * | 2002-10-15 | 2004-06-17 | Kwon Glen S. | Encapsulation and deaggregation of polyene antibiotics using poly(ethylene glycol)-phospholipid micelles |
| AU2002350719A1 (en) * | 2002-11-29 | 2004-06-23 | Janssen Pharmaceutica N.V. | Pharmaceutical compositions comprising a basic respectively acidic drug compound, a surfactant and a physiologically tolerable water-soluble acid respectively base |
| US7731947B2 (en) * | 2003-11-17 | 2010-06-08 | Intarcia Therapeutics, Inc. | Composition and dosage form comprising an interferon particle formulation and suspending vehicle |
| CN1897918A (zh) * | 2003-11-17 | 2007-01-17 | 阿尔萨公司 | 包含两亲性分子作为混悬载体的组合物和剂型 |
| EP1706098A4 (en) * | 2003-11-26 | 2012-08-15 | Supernus Pharmaceuticals Inc | MICRO-LAYER SYSTEMS FOR THE TRANSPORT OF LIPOPHILES AND BZW. HYDROPHOBIC COMPOUNDS |
| MXPA06015220A (es) * | 2004-06-21 | 2007-12-13 | Nektar Therapeutics | Composiciones comprendiendo anfotericina b, metodos y sistemas. |
| CN100418536C (zh) * | 2005-04-06 | 2008-09-17 | 河南省眼科研究所 | 一种用于眼科的抗真菌药物组合物 |
| CA2604943C (en) | 2005-04-15 | 2013-09-17 | Clarus Therapeutics, Inc. | Pharmaceutical delivery systems for hydrophobic drugs and compositions comprising same |
| CN100418537C (zh) * | 2005-07-15 | 2008-09-17 | 同济大学 | 两性霉素b缓释微球及其制备方法 |
| WO2008058234A2 (en) | 2006-11-08 | 2008-05-15 | Memory Pharmaceuticals Corporation | Pharmaceutical formulations for 1,4-dihyrdropyridine compounds having improved solubility |
| KR20100017109A (ko) * | 2007-05-18 | 2010-02-16 | 싸이도우스 엘엘씨. | 지프라시돈 제제 |
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| RU2009148315A (ru) | 2011-06-27 |
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| CA2688036C (en) | 2016-08-16 |
| CN101687044B (zh) | 2014-10-29 |
| JP5501224B2 (ja) | 2014-05-21 |
| MX2009012782A (es) | 2010-03-04 |
| EP2164518A1 (en) | 2010-03-24 |
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| ZA200908928B (en) | 2014-05-28 |
| US20140228308A1 (en) | 2014-08-14 |
| WO2008144888A1 (en) | 2008-12-04 |
| AU2008255525A1 (en) | 2008-12-04 |
| CA2688036A1 (en) | 2008-12-04 |
| RU2485975C2 (ru) | 2013-06-27 |
| EP2164518B1 (en) | 2019-04-24 |
| KR20100017928A (ko) | 2010-02-16 |
| IL202111A (en) | 2015-06-30 |
| KR20160029866A (ko) | 2016-03-15 |
| US20100273728A1 (en) | 2010-10-28 |
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