KR20140003376A - 프레가발린의 경구투여용 제제 - Google Patents
프레가발린의 경구투여용 제제 Download PDFInfo
- Publication number
- KR20140003376A KR20140003376A KR1020137003217A KR20137003217A KR20140003376A KR 20140003376 A KR20140003376 A KR 20140003376A KR 1020137003217 A KR1020137003217 A KR 1020137003217A KR 20137003217 A KR20137003217 A KR 20137003217A KR 20140003376 A KR20140003376 A KR 20140003376A
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- Prior art keywords
- oral
- formulation
- pregabalin
- oral administration
- matrix
- Prior art date
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- Ceased
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Images
Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
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- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A—HUMAN NECESSITIES
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
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- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
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- Hematology (AREA)
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- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10008104.1 | 2010-08-03 | ||
| EP10008104A EP2415460A1 (de) | 2010-08-03 | 2010-08-03 | Orale Darreichungsform von Pregabalin |
| PCT/EP2011/003873 WO2012016683A2 (en) | 2010-08-03 | 2011-08-02 | Oral dosage form of pregabalin |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20140003376A true KR20140003376A (ko) | 2014-01-09 |
Family
ID=43216378
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020137003217A Ceased KR20140003376A (ko) | 2010-08-03 | 2011-08-02 | 프레가발린의 경구투여용 제제 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20130149253A1 (https=) |
| EP (2) | EP2415460A1 (https=) |
| JP (1) | JP5937593B2 (https=) |
| KR (1) | KR20140003376A (https=) |
| CA (1) | CA2806752A1 (https=) |
| WO (1) | WO2012016683A2 (https=) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104561442A (zh) * | 2014-10-23 | 2015-04-29 | 江浦不锈钢制造有限公司 | 一种核电用奥氏体不锈钢的制备方法 |
| WO2018143511A1 (ko) * | 2017-02-01 | 2018-08-09 | 지엘팜텍 주식회사 | 프레가발린 함유 경구용 서방성 삼중정제 |
| WO2018143512A1 (ko) * | 2017-02-01 | 2018-08-09 | 지엘팜텍 주식회사 | 프레가발린 함유 고팽윤성 서방성 삼중정제 |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2849733B1 (en) * | 2011-12-19 | 2020-04-08 | Mahmut Bilgic | Effervescent pharmaceutical formulations comprising pregabalin and vitamin b12 |
| WO2013100873A1 (en) * | 2011-12-19 | 2013-07-04 | Mahmut Bilgic | Pharmaceutical formulation of pregabalin (particle size 300-2500 micrometer) |
| WO2013100874A1 (en) * | 2011-12-19 | 2013-07-04 | Mahmut Bilgic | Effervescent pregablin formulation |
| MX2013001278A (es) * | 2013-01-31 | 2014-07-30 | Miguel Ángel García Pérez | Composicion farmaceutica con un sistema bifasico de liberacion inmediata para el control de eventos convulsivos y del dolor. |
| US9913803B2 (en) * | 2013-08-26 | 2018-03-13 | Amorsa Therapeutics, Inc. | Single-layer oral dose of neuro-attenuating ketamine |
| IN2014MU00198A (https=) * | 2014-01-21 | 2015-08-28 | Intas Pharmaceuticals Ltd | |
| PL235144B1 (pl) * | 2014-06-03 | 2020-06-01 | Univ Medyczny Im Piastow Slaskich We Wroclawiu | Sposób wytwarzania tabletki flotacyjnej o przedłużonym oddziaływaniu substancji leczniczych z błoną śluzową żołądka oraz kompozycja farmaceutyczna |
| WO2016062182A1 (zh) * | 2014-10-24 | 2016-04-28 | 江苏恒瑞医药股份有限公司 | 一种普瑞巴林缓释制剂 |
| JP6919119B2 (ja) * | 2017-01-23 | 2021-08-18 | 日新製薬株式会社 | ３位が置換されたγ−アミノ酪酸誘導体を含有する圧縮固形医薬組成物。 |
| CN121015618A (zh) * | 2020-07-20 | 2025-11-28 | 四川海思科制药有限公司 | 一种稠合三环γ-氨基酸衍生物的缓释药物制剂及其制备方法 |
| CN112245404A (zh) * | 2020-11-02 | 2021-01-22 | 成都晶富医药科技有限公司 | 一种普瑞巴林胶囊及其制备方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3856816B2 (ja) | 1992-05-20 | 2006-12-13 | ノースウェスターン ユニヴァーシティ | 抗発作治療用のｇａｂａ及びｌ−グルタミン酸類縁体 |
| ATE245414T1 (de) * | 1998-09-14 | 2003-08-15 | Ranbaxy Lab Ltd | Oral verabreichtes system zur zeitlich und räumlich gesteuerten arzneistoffabgabe |
| CA2356829A1 (en) * | 2000-09-22 | 2002-03-22 | Warner-Lambert Company | Method for treating asthma using pregabalin |
| US20070184104A1 (en) * | 2001-10-25 | 2007-08-09 | Depomed, Inc. | Gastric retentive gabapentin dosage forms and methods for using same |
| CA2491665A1 (fr) * | 2004-12-24 | 2006-06-24 | Louis Cartilier | Formulation de comprime pour liberation soutenue de principe actif |
| WO2007048223A2 (en) * | 2005-10-25 | 2007-05-03 | Pharmascience Inc. | A gastric retention drug delivery system |
| US20070092565A1 (en) * | 2005-10-25 | 2007-04-26 | Pharmascience Inc. | Gastric retention drug delivery system |
| NL2000281C2 (nl) * | 2005-11-02 | 2007-08-07 | Pfizer Prod Inc | Vaste farmaceutische samenstellingen die pregabaline bevatten. |
| JP2009522294A (ja) * | 2005-12-29 | 2009-06-11 | デポメッド， インコーポレイテッド | 胃保持型ガバペンチン投薬形態およびその使用方法 |
| CA2661172A1 (en) * | 2006-09-04 | 2008-05-29 | Panacea Biotec Limited | Programmable buoyant delivery technology |
| CA2673336A1 (en) * | 2006-12-21 | 2008-06-26 | Xenoport, Inc. | Levodopa dimethyl-substituted diester prodrugs, compositions, and methods of use |
| US20110268666A1 (en) * | 2008-09-29 | 2011-11-03 | Yissum Research Development Company of the Research University of Jerusalem, Ltd. | Novel gastroretentive delivery system |
| EP2448406B1 (en) * | 2009-02-26 | 2016-04-20 | Relmada Therapeutics, Inc. | Extended release oral pharmaceutical compositions of 3-hydroxy-n-methylmorphinan and method of use |
| JP6170918B2 (ja) * | 2011-07-26 | 2017-07-26 | ユーハン・コーポレイションＹＵＨＡＮ Ｃｏｒｐｏｒａｔｉｏｎ | 二相の放出制御システムによるプレガバリンを含む徐放錠 |
-
2010
- 2010-08-03 EP EP10008104A patent/EP2415460A1/de not_active Withdrawn
-
2011
- 2011-08-02 US US13/812,506 patent/US20130149253A1/en not_active Abandoned
- 2011-08-02 CA CA2806752A patent/CA2806752A1/en not_active Abandoned
- 2011-08-02 EP EP11741406.0A patent/EP2600831A2/en not_active Withdrawn
- 2011-08-02 KR KR1020137003217A patent/KR20140003376A/ko not_active Ceased
- 2011-08-02 WO PCT/EP2011/003873 patent/WO2012016683A2/en not_active Ceased
- 2011-08-02 JP JP2013522132A patent/JP5937593B2/ja active Active
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104561442A (zh) * | 2014-10-23 | 2015-04-29 | 江浦不锈钢制造有限公司 | 一种核电用奥氏体不锈钢的制备方法 |
| WO2018143511A1 (ko) * | 2017-02-01 | 2018-08-09 | 지엘팜텍 주식회사 | 프레가발린 함유 경구용 서방성 삼중정제 |
| WO2018143512A1 (ko) * | 2017-02-01 | 2018-08-09 | 지엘팜텍 주식회사 | 프레가발린 함유 고팽윤성 서방성 삼중정제 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20130149253A1 (en) | 2013-06-13 |
| EP2415460A1 (de) | 2012-02-08 |
| CA2806752A1 (en) | 2012-02-09 |
| WO2012016683A3 (en) | 2012-05-31 |
| EP2600831A2 (en) | 2013-06-12 |
| JP2013535477A (ja) | 2013-09-12 |
| JP5937593B2 (ja) | 2016-06-22 |
| WO2012016683A2 (en) | 2012-02-09 |
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