KR20130108997A - 치환된 헤테로시클릴 벤질 피라졸 및 그의 용도 - Google Patents
치환된 헤테로시클릴 벤질 피라졸 및 그의 용도 Download PDFInfo
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- KR20130108997A KR20130108997A KR1020127032069A KR20127032069A KR20130108997A KR 20130108997 A KR20130108997 A KR 20130108997A KR 1020127032069 A KR1020127032069 A KR 1020127032069A KR 20127032069 A KR20127032069 A KR 20127032069A KR 20130108997 A KR20130108997 A KR 20130108997A
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10004855.2 | 2010-05-08 | ||
| EP10004855 | 2010-05-08 | ||
| PCT/EP2011/057021 WO2011141326A1 (de) | 2010-05-08 | 2011-05-03 | Substituierte heterocyclylbenzyl-pyrazole und ihre verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20130108997A true KR20130108997A (ko) | 2013-10-07 |
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ID=44063276
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020127032069A Withdrawn KR20130108997A (ko) | 2010-05-08 | 2011-05-03 | 치환된 헤테로시클릴 벤질 피라졸 및 그의 용도 |
Country Status (26)
| Country | Link |
|---|---|
| US (2) | US20130172311A1 (https=) |
| EP (1) | EP2569312B1 (https=) |
| JP (1) | JP5727002B2 (https=) |
| KR (1) | KR20130108997A (https=) |
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| AR (1) | AR081368A1 (https=) |
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Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2685875C (en) * | 2007-05-01 | 2015-10-06 | Hill's Pet Nutrition, Inc. | Methods and compositions for diagnosing osteoarthritis in a feline |
| CA2687306A1 (en) * | 2007-05-18 | 2008-11-27 | Bayer Schering Pharma Aktiengesellschaft | Heteroaryl substituted pyrazole derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis |
| PE20130228A1 (es) * | 2010-05-08 | 2013-03-15 | Bayer Ip Gmbh | Heterociclilbencilpirazoles sustituidos |
| EP2867230B1 (en) | 2012-07-02 | 2020-02-12 | Monsanto Technology LLC | Process for the preparation of 3,5-disubstituted-1,2,4-oxadiazoles |
| EP2888253A4 (en) * | 2012-08-24 | 2016-01-06 | Univ Texas | HETEROCYCLIC HIF ACTIVITY MODULATORS FOR THE TREATMENT OF DISEASES |
| US20140073634A1 (en) * | 2012-08-24 | 2014-03-13 | Institute For Applied Cancer Science/The University of Texas MD Anderson Cancer Center | Heterocyclic modulators of hif activity for treatment of disease |
| ES2691643T3 (es) | 2012-08-24 | 2018-11-28 | Board Of Regents, The University Of Texas System | Moduladores heterocíclicos de la actividad de HIF para el tratamiento de enfermedades |
| WO2015130790A2 (en) | 2014-02-25 | 2015-09-03 | Board Of Regents, University Of Texas System | Salts of heterocyclic modulators of hif activity for treatment of disease |
| US10191597B2 (en) | 2015-06-30 | 2019-01-29 | Synaptics Incorporated | Modulating a reference voltage to preform capacitive sensing |
| KR102544307B1 (ko) * | 2017-01-13 | 2023-06-15 | 닛산 가가쿠 가부시키가이샤 | 방향족 디아민 화합물 전구체의 제조 방법 |
| CN115944626B (zh) * | 2022-12-08 | 2024-04-19 | 桂林医学院附属医院 | 小分子化合物在制备抗缺氧或缺血再灌注损伤药物中的应用 |
| WO2025096662A1 (en) * | 2023-10-30 | 2025-05-08 | Pretzel Therapeutics, Inc. | Compositions and inhibitors of polrmt |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6610726B2 (en) * | 2001-06-29 | 2003-08-26 | North Shore-Long Island Jewish Research Institute | Compositions and agents for modulating cellular proliferation and angiogenesis |
| AU2004228057A1 (en) | 2003-04-03 | 2004-10-21 | Merck & Co., Inc. | Di-aryl substituted pyrazole modulators of metabotropic glutamate receptor-5 |
| AU2004275694B2 (en) | 2003-06-30 | 2008-03-06 | Bizbiotech Co., Ltd. | Compounds, compositions and methods |
| CN1842332A (zh) * | 2003-06-30 | 2006-10-04 | Hif生物公司 | 化合物、组合物及方法 |
| GB0508472D0 (en) * | 2005-04-26 | 2005-06-01 | Glaxo Group Ltd | Compounds |
| WO2007065010A2 (en) | 2005-12-02 | 2007-06-07 | Hif Bio, Inc. | Anti-angiogenesis compounds |
| CA2687306A1 (en) * | 2007-05-18 | 2008-11-27 | Bayer Schering Pharma Aktiengesellschaft | Heteroaryl substituted pyrazole derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis |
| AU2009316019A1 (en) * | 2008-11-14 | 2010-05-20 | Bayer Intellectual Property Gmbh | Heterocyclically substituted aryl compounds as HIF inhibitors |
| DE102008057344A1 (de) * | 2008-11-14 | 2010-05-20 | Bayer Schering Pharma Aktiengesellschaft | Aminoalkyl-substituierte Aryl-Verbindungen und ihre Verwendung |
| WO2010054764A1 (de) * | 2008-11-14 | 2010-05-20 | Bayer Schering Pharma Aktiengesellschaft | Heteroaromatische verbindungen zur verwendung als hif-inhibitoren |
| EP2202232A1 (en) | 2008-12-26 | 2010-06-30 | Laboratorios Almirall, S.A. | 1,2,4-oxadiazole derivatives and their therapeutic use |
| ES2405054T3 (es) | 2009-01-23 | 2013-05-30 | Bristol-Myers Squibb Company | Derivados de pirazol-1,2,4-oxadiazol como agonistas de esfingosina-1-fosfato |
| PE20130228A1 (es) * | 2010-05-08 | 2013-03-15 | Bayer Ip Gmbh | Heterociclilbencilpirazoles sustituidos |
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| US20120028950A1 (en) | 2012-02-02 |
| US8470811B2 (en) | 2013-06-25 |
| CU20120157A7 (es) | 2013-03-27 |
| CA2798375A1 (en) | 2011-11-17 |
| CN103003269B (zh) | 2015-11-25 |
| PE20130228A1 (es) | 2013-03-15 |
| JP2013526497A (ja) | 2013-06-24 |
| PH12012502202A1 (en) | 2013-02-04 |
| SG185459A1 (en) | 2012-12-28 |
| EP2569312B1 (de) | 2014-03-26 |
| MX2012012960A (es) | 2012-12-17 |
| EA201291167A1 (ru) | 2013-05-30 |
| US20130172311A1 (en) | 2013-07-04 |
| ECSP12012288A (es) | 2012-12-28 |
| IL222851A0 (en) | 2012-12-31 |
| CR20120570A (es) | 2013-04-22 |
| DOP2012000284A (es) | 2013-03-31 |
| AU2011252223A1 (en) | 2012-12-06 |
| MA34939B1 (fr) | 2014-03-01 |
| ES2462522T3 (es) | 2014-05-23 |
| TW201200510A (en) | 2012-01-01 |
| EP2569312A1 (de) | 2013-03-20 |
| TN2012000531A1 (en) | 2014-04-01 |
| WO2011141326A1 (de) | 2011-11-17 |
| CO6640218A2 (es) | 2013-03-22 |
| UY33369A (es) | 2011-12-01 |
| AR081368A1 (es) | 2012-08-29 |
| BR112012028651A2 (pt) | 2016-08-09 |
| JP5727002B2 (ja) | 2015-06-03 |
| CN103003269A (zh) | 2013-03-27 |
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