KR20120063515A - Ｐｉ３ 키나제 억제제 및 이들의 용도 - Google Patents

Ｐｉ３ 키나제 억제제 및 이들의 용도 Download PDF

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KR20120063515A
KR20120063515A KR1020127009074A KR20127009074A KR20120063515A KR 20120063515 A KR20120063515 A KR 20120063515A KR 1020127009074 A KR1020127009074 A KR 1020127009074A KR 20127009074 A KR20127009074 A KR 20127009074A KR 20120063515 A KR20120063515 A KR 20120063515A
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South Korea
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ring
nitrogen
oxygen
sulfur
membered
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Korean (ko)
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더창 뉴
러셀 씨. 피터
저스윈더 싱
아서 에프. 클루지
호르모츠 마즈디야스니
정둥 주
리신 차오
케빈 쿤츠
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아빌라 테라퓨틱스, 인크.
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • C12N9/00—Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/10—Transferases (2.)
    • C12N9/12—Transferases (2.) transferring phosphorus containing groups, e.g. kinases (2.7)
    • C12N9/1205—Phosphotransferases with an alcohol group as acceptor (2.7.1), e.g. protein kinases

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KR1020127009074A 2009-09-09 2010-09-09 Ｐｉ３ 키나제 억제제 및 이들의 용도 Ceased KR20120063515A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US24094709P 2009-09-09 2009-09-09
US61/240,947 2009-09-09
US37139610P 2010-08-06 2010-08-06
US61/371,396 2010-08-06

Publications (1)

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KR20120063515A true KR20120063515A (ko) 2012-06-15

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KR1020127009074A Ceased KR20120063515A (ko) 2009-09-09 2010-09-09 Ｐｉ３ 키나제 억제제 및 이들의 용도

Country Status (16)

Country Link
US (1) US20110230476A1 (https=)
EP (1) EP2475375A4 (https=)
JP (1) JP2013504325A (https=)
KR (1) KR20120063515A (https=)
CN (1) CN102625708A (https=)
AU (1) AU2010292198A1 (https=)
BR (1) BR112012008385A2 (https=)
CA (1) CA2773848A1 (https=)
IL (1) IL218555A0 (https=)
MX (1) MX339584B (https=)
NZ (2) NZ598808A (https=)
PH (1) PH12012500491A1 (https=)
RU (1) RU2595718C2 (https=)
SG (2) SG10201405598QA (https=)
TW (2) TW201609747A (https=)
WO (1) WO2011031896A2 (https=)

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