KR20080036585A - 근육 이완 및 항―염증 활성이 있는 티오콜히코시드 유사체 - Google Patents
근육 이완 및 항―염증 활성이 있는 티오콜히코시드 유사체 Download PDFInfo
- Publication number
- KR20080036585A KR20080036585A KR1020087001654A KR20087001654A KR20080036585A KR 20080036585 A KR20080036585 A KR 20080036585A KR 1020087001654 A KR1020087001654 A KR 1020087001654A KR 20087001654 A KR20087001654 A KR 20087001654A KR 20080036585 A KR20080036585 A KR 20080036585A
- Authority
- KR
- South Korea
- Prior art keywords
- demethoxy
- myorelaxant
- meoh
- inflammatory activity
- aminothiocolhitchin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/24—Condensed ring systems having three or more rings
- C07H15/248—Colchicine radicals, e.g. colchicosides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C323/39—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
- C07C323/40—Y being a hydrogen or a carbon atom
- C07C323/41—Y being a hydrogen or an acyclic carbon atom
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biochemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Molecular Biology (AREA)
- Pain & Pain Management (AREA)
- General Chemical & Material Sciences (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Epidemiology (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI2005A001418 | 2005-07-22 | ||
| IT001418A ITMI20051418A1 (it) | 2005-07-22 | 2005-07-22 | Analoghi del tiocolchicoside ad attivita'miorilassante e antiinfiammatoria |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20080036585A true KR20080036585A (ko) | 2008-04-28 |
Family
ID=37420844
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020087001654A KR20080036585A (ko) | 2005-07-22 | 2006-07-20 | 근육 이완 및 항―염증 활성이 있는 티오콜히코시드 유사체 |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP1907405A1 (es) |
| JP (1) | JP2009502755A (es) |
| KR (1) | KR20080036585A (es) |
| CN (1) | CN101228175A (es) |
| AU (1) | AU2006271923A1 (es) |
| BR (1) | BRPI0613680A2 (es) |
| CA (1) | CA2615860A1 (es) |
| IL (1) | IL188900A0 (es) |
| IT (1) | ITMI20051418A1 (es) |
| MX (1) | MX2008000968A (es) |
| NO (1) | NO20080377L (es) |
| NZ (1) | NZ565265A (es) |
| RU (1) | RU2008102251A (es) |
| WO (1) | WO2007009772A1 (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8421747B2 (en) * | 2008-09-24 | 2013-04-16 | Microsoft Corporation | Object detection and user settings |
| WO2010138670A2 (en) * | 2009-05-27 | 2010-12-02 | Mutual Pharmaceutical Company, Inc. | Thiocolchicine derivatives, method of making and methods of use thereof |
| CN102741223A (zh) * | 2010-01-22 | 2012-10-17 | 共有药物有限公司 | 硫代秋水仙碱和秋水仙碱类似物、其制备方法和使用方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1291550B1 (it) * | 1997-04-11 | 1999-01-11 | Indena Spa | Derivati della colchicina e della tiocolchicina ad attivita' antinfiammatoria e miorilassante |
| ITMI20031144A1 (it) * | 2003-06-06 | 2004-12-07 | Indena Spa | Analoghi del colchicoside. |
-
2005
- 2005-07-22 IT IT001418A patent/ITMI20051418A1/it unknown
-
2006
- 2006-07-20 NZ NZ565265A patent/NZ565265A/en unknown
- 2006-07-20 MX MX2008000968A patent/MX2008000968A/es unknown
- 2006-07-20 EP EP06762703A patent/EP1907405A1/en not_active Withdrawn
- 2006-07-20 AU AU2006271923A patent/AU2006271923A1/en not_active Abandoned
- 2006-07-20 CN CNA2006800267270A patent/CN101228175A/zh active Pending
- 2006-07-20 CA CA002615860A patent/CA2615860A1/en not_active Abandoned
- 2006-07-20 BR BRPI0613680-0A patent/BRPI0613680A2/pt not_active IP Right Cessation
- 2006-07-20 RU RU2008102251/04A patent/RU2008102251A/ru not_active Application Discontinuation
- 2006-07-20 WO PCT/EP2006/007108 patent/WO2007009772A1/en not_active Application Discontinuation
- 2006-07-20 KR KR1020087001654A patent/KR20080036585A/ko not_active Application Discontinuation
- 2006-07-20 JP JP2008521882A patent/JP2009502755A/ja not_active Ceased
-
2008
- 2008-01-21 IL IL188900A patent/IL188900A0/en unknown
- 2008-01-21 NO NO20080377A patent/NO20080377L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| RU2008102251A (ru) | 2009-07-27 |
| JP2009502755A (ja) | 2009-01-29 |
| BRPI0613680A2 (pt) | 2011-01-25 |
| ITMI20051418A1 (it) | 2007-01-23 |
| MX2008000968A (es) | 2008-03-26 |
| EP1907405A1 (en) | 2008-04-09 |
| AU2006271923A1 (en) | 2007-01-25 |
| CN101228175A (zh) | 2008-07-23 |
| WO2007009772A1 (en) | 2007-01-25 |
| NO20080377L (no) | 2008-02-01 |
| CA2615860A1 (en) | 2007-01-25 |
| NZ565265A (en) | 2010-01-29 |
| IL188900A0 (en) | 2008-04-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |