NO20080377L - Tiokochikosidanaloger med myorelakserende og antiinflammatorisk aktivitet - Google Patents

Tiokochikosidanaloger med myorelakserende og antiinflammatorisk aktivitet

Info

Publication number
NO20080377L
NO20080377L NO20080377A NO20080377A NO20080377L NO 20080377 L NO20080377 L NO 20080377L NO 20080377 A NO20080377 A NO 20080377A NO 20080377 A NO20080377 A NO 20080377A NO 20080377 L NO20080377 L NO 20080377L
Authority
NO
Norway
Prior art keywords
inflammatory activity
thiocochicoside
myorelaxative
analogues
formula
Prior art date
Application number
NO20080377A
Other languages
English (en)
Norwegian (no)
Inventor
Paolo Morazzoni
Gabriele Fontana
Antonella Riva
Ezio Bombardelli
Donato Pocar
Maria Luisa Gelmi
Guido Pontremoli
Original Assignee
Indena Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Indena Spa filed Critical Indena Spa
Publication of NO20080377L publication Critical patent/NO20080377L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/24Condensed ring systems having three or more rings
    • C07H15/248Colchicine radicals, e.g. colchicosides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/23Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/39Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
    • C07C323/40Y being a hydrogen or a carbon atom
    • C07C323/41Y being a hydrogen or an acyclic carbon atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
NO20080377A 2005-07-22 2008-01-21 Tiokochikosidanaloger med myorelakserende og antiinflammatorisk aktivitet NO20080377L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT001418A ITMI20051418A1 (it) 2005-07-22 2005-07-22 Analoghi del tiocolchicoside ad attivita'miorilassante e antiinfiammatoria
PCT/EP2006/007108 WO2007009772A1 (en) 2005-07-22 2006-07-20 Thiocolchicoside analogues with myorelaxant and anti-inflammatory activity

Publications (1)

Publication Number Publication Date
NO20080377L true NO20080377L (no) 2008-02-01

Family

ID=37420844

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20080377A NO20080377L (no) 2005-07-22 2008-01-21 Tiokochikosidanaloger med myorelakserende og antiinflammatorisk aktivitet

Country Status (14)

Country Link
EP (1) EP1907405A1 (es)
JP (1) JP2009502755A (es)
KR (1) KR20080036585A (es)
CN (1) CN101228175A (es)
AU (1) AU2006271923A1 (es)
BR (1) BRPI0613680A2 (es)
CA (1) CA2615860A1 (es)
IL (1) IL188900A0 (es)
IT (1) ITMI20051418A1 (es)
MX (1) MX2008000968A (es)
NO (1) NO20080377L (es)
NZ (1) NZ565265A (es)
RU (1) RU2008102251A (es)
WO (1) WO2007009772A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8421747B2 (en) * 2008-09-24 2013-04-16 Microsoft Corporation Object detection and user settings
WO2010138670A2 (en) * 2009-05-27 2010-12-02 Mutual Pharmaceutical Company, Inc. Thiocolchicine derivatives, method of making and methods of use thereof
CN102741223A (zh) * 2010-01-22 2012-10-17 共有药物有限公司 硫代秋水仙碱和秋水仙碱类似物、其制备方法和使用方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1291550B1 (it) * 1997-04-11 1999-01-11 Indena Spa Derivati della colchicina e della tiocolchicina ad attivita' antinfiammatoria e miorilassante
ITMI20031144A1 (it) * 2003-06-06 2004-12-07 Indena Spa Analoghi del colchicoside.

Also Published As

Publication number Publication date
RU2008102251A (ru) 2009-07-27
JP2009502755A (ja) 2009-01-29
BRPI0613680A2 (pt) 2011-01-25
ITMI20051418A1 (it) 2007-01-23
MX2008000968A (es) 2008-03-26
EP1907405A1 (en) 2008-04-09
KR20080036585A (ko) 2008-04-28
AU2006271923A1 (en) 2007-01-25
CN101228175A (zh) 2008-07-23
WO2007009772A1 (en) 2007-01-25
CA2615860A1 (en) 2007-01-25
NZ565265A (en) 2010-01-29
IL188900A0 (en) 2008-04-13

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application