KR20060130697A - 신규한 아미도-치환 히드록시-6-페닐페난트리딘 및 ｐｄｅ4억제제로서의 이의 용도 - Google Patents

신규한 아미도-치환 히드록시-6-페닐페난트리딘 및 ｐｄｅ4억제제로서의 이의 용도 Download PDF

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Publication number
KR20060130697A
KR20060130697A KR1020067020318A KR20067020318A KR20060130697A KR 20060130697 A KR20060130697 A KR 20060130697A KR 1020067020318 A KR1020067020318 A KR 1020067020318A KR 20067020318 A KR20067020318 A KR 20067020318A KR 20060130697 A KR20060130697 A KR 20060130697A
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South Korea
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alkyl
hydrogen
methoxy
hydroxy
hexahydro
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KR1020067020318A
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Korean (ko)
Inventor
베아테 슈미트
디터 플로커치
아르민 하첼만
크리스토프 치트
요하네스 바르지히
데겐하르트 막스
한스-페터 클라이
울리히 카우츠
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알타나 파마 아게
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/10—Aza-phenanthrenes
    • C07D221/12—Phenanthridines
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Diabetes (AREA)
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  • Pain & Pain Management (AREA)
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  • Virology (AREA)
  • Urology & Nephrology (AREA)
  • Psychiatry (AREA)
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  • Tropical Medicine & Parasitology (AREA)
  • Ophthalmology & Optometry (AREA)
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KR1020067020318A 2004-03-10 2005-03-09 신규한 아미도-치환 히드록시-6-페닐페난트리딘 및 ｐｄｅ4억제제로서의 이의 용도 Ceased KR20060130697A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP04100990.3 2004-03-10
EP04100990 2004-03-10
EP04106677 2004-12-17
EP04106677.0 2004-12-17

Publications (1)

Publication Number Publication Date
KR20060130697A true KR20060130697A (ko) 2006-12-19

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KR1020067020318A Ceased KR20060130697A (ko) 2004-03-10 2005-03-09 신규한 아미도-치환 히드록시-6-페닐페난트리딘 및 ｐｄｅ4억제제로서의 이의 용도

Country Status (15)

Country Link
US (1) US20070185149A1 (https=)
EP (1) EP1725534A1 (https=)
JP (1) JP2007527901A (https=)
KR (1) KR20060130697A (https=)
CN (1) CN1926113B (https=)
AR (1) AR049324A1 (https=)
AU (1) AU2005221832A1 (https=)
BR (1) BRPI0508481A (https=)
CA (1) CA2558391A1 (https=)
IL (1) IL177496A0 (https=)
MX (1) MXPA06009892A (https=)
NO (1) NO20064415L (https=)
NZ (1) NZ549254A (https=)
TW (1) TW200600499A (https=)
WO (1) WO2005087745A1 (https=)

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PL2589599T4 (pl) 2004-03-03 2015-06-30 Takeda Gmbh Nowe hydroksy-6-heteroarylofenantrydyny i ich zastosowanie jako inhibitorów PDE4
EP1791847A2 (en) 2004-09-08 2007-06-06 Altana Pharma AG Novel 3-thia-10-aza-phenanthrene derivatives
ATE508130T1 (de) 2004-09-08 2011-05-15 Nycomed Gmbh 3-oxa-10-aza-phenanthrene als pde4- oder pde3/4- inhibitoren
PL1856093T3 (pl) * 2005-03-02 2010-05-31 Takeda Gmbh Chlorowodorek (2R,4aR,10bR)-6-(2,6-dimetoksy-pirydyn-3-ylo)-9-etoksy-8-metoksy-1,2,3,4,4a,10b-heksahydrofenantrydyn-2-olu
GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
JP2010508315A (ja) 2006-10-30 2010-03-18 ノバルティス アーゲー 抗炎症剤としてのヘテロ環式化合物
ES2460897T3 (es) 2007-10-04 2014-05-14 F. Hoffmann-La Roche Ag Derivados de ciclopropil aril amida y usos de los mismos
AU2009203693B2 (en) 2008-01-11 2012-06-07 Novartis Ag Pyrimidines as kinase inhibitors
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CN1926113A (zh) 2007-03-07
WO2005087745A8 (en) 2006-10-26
MXPA06009892A (es) 2007-03-01
JP2007527901A (ja) 2007-10-04
BRPI0508481A (pt) 2007-07-31
NZ549254A (en) 2010-06-25
CA2558391A1 (en) 2005-09-22
NO20064415L (no) 2006-10-10
CN1926113B (zh) 2010-06-23
AR049324A1 (es) 2006-07-19
IL177496A0 (en) 2006-12-10
US20070185149A1 (en) 2007-08-09
AU2005221832A1 (en) 2005-09-22
EP1725534A1 (en) 2006-11-29

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