KR20050040912A - 플라비비리다에 감염 치료용의 비사이클로[4.2.1]노난시스템을 가지는 화합물 - Google Patents

플라비비리다에 감염 치료용의 비사이클로[4.2.1]노난시스템을 가지는 화합물 Download PDF

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KR20050040912A
KR20050040912A KR1020057001868A KR20057001868A KR20050040912A KR 20050040912 A KR20050040912 A KR 20050040912A KR 1020057001868 A KR1020057001868 A KR 1020057001868A KR 20057001868 A KR20057001868 A KR 20057001868A KR 20050040912 A KR20050040912 A KR 20050040912A
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lower alkyl
hydrogen
aryl
alkenyl
compound
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왕페이유안
스투이버리벤제이.
와타나베교이치에이.
하산압달라
천병관
홀레커롤랑
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파마셋 인코포레이티드
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    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
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    • A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
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    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
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    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
    • A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
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    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
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    • C07H9/06—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical the hetero ring containing nitrogen as ring hetero atoms

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KR1020057001868A 2002-08-01 2003-08-01 플라비비리다에 감염 치료용의 비사이클로[4.2.1]노난시스템을 가지는 화합물 Ceased KR20050040912A (ko)

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US45371602P 2002-08-01 2002-08-01
US60/453,716 2002-08-01

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US (1) US8093380B2 (enExample)
EP (1) EP1545545A4 (enExample)
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KR (1) KR20050040912A (enExample)
AU (1) AU2003257157C1 (enExample)
BR (1) BR0313164A (enExample)
CA (1) CA2494340C (enExample)
IL (1) IL166640A0 (enExample)
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